(Q39660148)

13 September 2017

title

Discovery and structure-activity relationship of a novel spirocarbamate series of NPY Y5 antagonists (English)

1 reference

13 September 2017

Discovery and structure–activity relationship of a novel spirocarbamate series of NPY Y5 antagonists (English)

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

5 July 2024

author name string

Jonathan Bentley

2

1 reference

13 September 2017

Matteo Biagetti

3

1 reference

13 September 2017

Stefania Contini

4

1 reference

13 September 2017

Romano Di Fabio

5

1 reference

13 September 2017

Daniele Donati

6

1 reference

13 September 2017

Thorsten Genski

7

1 reference

13 September 2017

Sebastien Guery

8

1 reference

13 September 2017

Angelica Mazzali

9

1 reference

13 September 2017

Giancarlo Merlo

10

1 reference

13 September 2017

Fabiola Sacco

12

1 reference

13 September 2017

Catia Seri

13

1 reference

13 September 2017

Michela Tessari

14

1 reference

13 September 2017

Laura Zonzini

15

1 reference

13 September 2017

Laura Caberlotto

16

1 reference

13 September 2017

Colin P. Leslie

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20813523

5 July 2024

Domenica A. Pizzi

11

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20813523

5 July 2024

language of work or name

English

0 references

publication date

12 August 2010

1 reference

full work available at URL

13 September 2017

number of pages

5

1 reference

based on heuristic

inferred from page(s)

https://api.elsevier.com/content/article/PII:S0960894X10011649?httpAccept=text/xml

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

https://api.elsevier.com/content/article/PII:S0960894X10011649?httpAccept=text/plain

5 July 2024

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

Bioorganic & Medicinal Chemistry Letters

5 July 2024

published in

1 reference

13 September 2017

volume

20

1 reference

13 September 2017

issue

20

1 reference

13 September 2017

page(s)

6103-6107

1 reference

Neuropeptide Y--a novel brain peptide with structural similarities to peptide YY and pancreatic polypeptide

13 September 2017

cites work

1

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

Neuropeptide Y and peptide YY neuronal and endocrine systems

5 July 2024

2

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

Synthesis of receptor antagonists of neuropeptide Y

5 July 2024

3

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

Neuropeptide Y injected in the paraventricular hypothalamus: a powerful stimulant of feeding behavior

5 July 2024

4

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

Evidence for neuropeptide Y mediation of eating produced by food deprivation and for a variant of the Y1 receptor mediating this peptide's effect

5 July 2024

5

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

Y-receptor subtypes--how many more?

5 July 2024

6

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

Neuropeptide y receptor selective ligands in the treatment of obesity

5 July 2024

7

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

Regulation of maternal food intake and mother-pup interactions by the Y5 receptor

5 July 2024

8

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

NPY receptors as drug targets for the central regulation of body weight

5 July 2024

9

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

Role of the Y5 neuropeptide Y receptor in feeding and obesity

5 July 2024

10

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

A receptor subtype involved in neuropeptide-Y-induced food intake

5 July 2024

11

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

Effects of a novel Y5 antagonist in obese mice: combination with food restriction or sibutramine

5 July 2024

12

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

Discovery of novel orally active ureido NPY Y5 receptor antagonists

5 July 2024

13

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

The Novel Neuropeptide Y Y5 Receptor Antagonist Lu AA33810 [N-[[trans-4-[(4,5-Dihydro[1]benzothiepino[5,4-d]thiazol-2-yl)amino]cyclohexyl]methyl]-methanesulfonamide] Exerts Anxiolytic- and Antidepressant-Like Effects in Rat Models of Stress …

5 July 2024

15

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

Neuropeptide Y5 receptor antagonism does not induce clinically meaningful weight loss in overweight and obese adults

5 July 2024

16

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

Aminothiazole derivatives as neuropeptide Y5 receptor ligands: finding the balance between affinity and physicochemical properties

5 July 2024

18

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

Discovery and SAR of potent, orally available and brain-penetrable 5,6-dihydro-4H-3-thia-1-aza-benzo[e]azulen- and 4,5-dihydro-6-oxa-3-thia-1-aza-benzo[e]azulen derivatives as neuropeptide Y Y5 receptor antagonists

5 July 2024

19

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

Aryl urea derivatives of spiropiperidines as NPY Y5 receptor antagonists.

5 July 2024

20

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

Identification of novel and orally active spiroindoline NPY Y5 receptor antagonists

5 July 2024

21

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

Novel orally active NPY Y5 receptor antagonists: Synthesis and structure-activity relationship of spiroindoline class compounds.

5 July 2024

22

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

Design, syntheses, and structure-activity relationships of novel NPY Y5 receptor antagonists: 2-{3-Oxospiro[isobenzofuran-1(3H),4'-piperidin]-1'-yl}benzimidazole derivatives

5 July 2024

23

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

Dimethyloxosulfonium Methylide ((CH3)2SOCH2) and Dimethylsulfonium Methylide ((CH3)2SCH2). Formation and Application to Organic Synthesis

5 July 2024

24

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.041

5 July 2024

Identifiers

1 reference

13 September 2017

1 reference