(Q39766088)

English

Lead optimization of N-3-substituted 7-morpholinotriazolopyrimidines as dual phosphoinositide 3-kinase/mammalian target of rapamycin inhibitors: discovery of PKI-402.

scientific article

Statements

Lead optimization of N-3-substituted 7-morpholinotriazolopyrimidines as dual phosphoinositide 3-kinase/mammalian target of rapamycin inhibitors: discovery of PKI-402. (English)
Christoph M Dehnhardt
Aranapakam M Venkatesan
Efren Delos Santos
Zecheng Chen
Osvaldo Santos
Semiramis Ayral-Kaloustian
Natasja Brooijmans
Robert Mallon
Irwin Hollander
Larry Feldberg
Judy Lucas
Inder Chaudhary
Ker Yu
Jay Gibbons
Robert Abraham
Tarek S Mansour
1 January 2010
798-810

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