(Q39830106)

English

Engineering galanin analogues that discriminate between GalR1 and GalR2 receptor subtypes and exhibit anticonvulsant activity following systemic delivery

scientific article

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scholarly article

1 reference

Europe PubMed Central

PMC publication ID

15 September 2017

Engineering galanin analogues that discriminate between GalR1 and GalR2 receptor subtypes and exhibit anticonvulsant activity following systemic delivery (English)

1 reference

Europe PubMed Central

PMC publication ID

15 September 2017

author name string

Charles R Robertson

1

1 reference

Europe PubMed Central

PMC publication ID

15 September 2017

Erika Adkins Scholl

2

1 reference

Europe PubMed Central

PMC publication ID

15 September 2017

Timothy H Pruess

3

1 reference

Europe PubMed Central

PMC publication ID

15 September 2017

Brad R Green

4

1 reference

Europe PubMed Central

PMC publication ID

15 September 2017

H Steve White

5

1 reference

Europe PubMed Central

PMC publication ID

15 September 2017

Grzegorz Bulaj

6

1 reference

Europe PubMed Central

PMC publication ID

15 September 2017

language of work or name

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publication date

1 February 2010

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Europe PubMed Central

PMC publication ID

15 September 2017

number of pages

5

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inferred from page(s)

Journal of Medicinal Chemistry

1 reference

Europe PubMed Central

PMC publication ID

15 September 2017

53

1 reference

Europe PubMed Central

PMC publication ID

15 September 2017

4

1 reference

Europe PubMed Central

PMC publication ID

15 September 2017

1871-1875

1 reference

Europe PubMed Central

PMC publication ID

15 September 2017

A novel GalR2-specific peptide agonist

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2846716

22 September 2017

IC50-to-Ki: a web-based tool for converting IC50 to Ki values for inhibitors of enzyme activity and ligand binding

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2846716

22 September 2017

Developing novel antiepileptic drugs: characterization of NAX 5055, a systemically-active galanin analog, in epilepsy models

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2846716

22 September 2017

Structural requirements for a lipoamino acid in modulating the anticonvulsant activities of systemically active galanin analogues

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2846716

22 September 2017

Design, synthesis, and characterization of high-affinity, systemically-active galanin analogues with potent anticonvulsant activities

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2846716

22 September 2017

Galanin, galanin receptors and drug targets

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2846716

22 September 2017

Galanin and spinal pain mechanisms: where do we stand in 2008?

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2846716

22 September 2017

Regulation of kindling epileptogenesis by hippocampal galanin type 1 and type 2 receptors: The effects of subtype-selective agonists and the role of G-protein-mediated signaling

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2846716

22 September 2017

Galmic, a nonpeptide galanin receptor agonist, affects behaviors in seizure, pain, and forced-swim tests

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2846716

22 September 2017

Anticonvulsant activity of a nonpeptide galanin receptor agonist

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2846716

22 September 2017

Pharmacological characterization of the 6 Hz psychomotor seizure model of partial epilepsy

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2846716

22 September 2017

Receptor subtype-specific pronociceptive and analgesic actions of galanin in the spinal cord: selective actions via GalR1 and GalR2 receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2846716

22 September 2017

Cloning and characterization of the human galanin GALR2 receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2846716

22 September 2017

Pharmacological and biochemical characterization of a recombinant human galanin GALR1 receptor: agonist character of chimeric galanin peptides

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2846716

22 September 2017

Cloning and expression of the human galanin receptor GalR2

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2846716

22 September 2017

Mutagenesis and ligand modification studies on galanin binding to its GTP-binding-protein-coupled receptor GalR1.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2846716

25 September 2017

Linear and cyclic N-terminal galanin fragments and analogs as ligands at the hypothalamic galanin receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2846716

17 June 2018

Important pharmacophores for binding to galanin receptor 2.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2846716

20 August 2018

Molecular modelling and site-directed mutagenesis of human GALR1 galanin receptor defines determinants of receptor subtype specificity

1 reference

https://pubmed.ncbi.nlm.nih.gov/20121116

12 December 2020

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inferred from PubMed ID database lookup

Identifiers

10.1021/JM9018349

1 reference

Europe PubMed Central

PMC publication ID

15 September 2017

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

15 September 2017

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

15 September 2017

ResearchGate publication ID

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