(Q39846240)

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Synthesis, molecular docking and biological evaluation as HDAC inhibitors of cyclopeptide mimetics by a tandem three-component reaction and intramolecular [3+2] cycloaddition.

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scholarly article

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29 January 2020

Synthesis, molecular docking and biological evaluation as HDAC inhibitors of cyclopeptide mimetics by a tandem three-component reaction and intramolecular [3+2] cycloaddition (English)

1 reference

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29 January 2020

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Armando A. Genazzani

7

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29 January 2020

Giuseppe Bifulco

6

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29 January 2020

author name string

Tracey Pirali

1

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29 January 2020

Valeria Faccio

2

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29 January 2020

Riccardo Mossetti

3

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29 January 2020

Ambra A Grolla

4

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29 January 2020

Simone Di Micco

5

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29 January 2020

Gian Cesare Tron

8

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29 January 2020

publication date

28 May 2009

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29 January 2020

Molecular Diversity

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29 January 2020

14

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29 January 2020

1

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29 January 2020

109-121

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29 January 2020

https://scigraph.springernature.com/pub.10.1007/s11030-009-9153-9

0 references

Structural snapshots of human HDAC8 provide insights into the class I histone deacetylases

1 reference

https://pubmed.ncbi.nlm.nih.gov/19475493

12 December 2020

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The exploration of macrocycles for drug discovery--an underexploited structural class

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Homology modeling, force field design, and free energy simulation studies to optimize the activities of histone deacetylase inhibitors

1 reference

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Development of a scintillation proximity assay for histone deacetylase using a biotinylated peptide derived from histone-H4

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Solution-phase parallel synthesis and biological evaluation of combretatriazoles

1 reference

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One-pot synthesis of macrocycles by a tandem three-component reaction and intramolecular [3+2] cycloaddition

1 reference

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A chemical switch for the modulation of the functional activity of higher homologues of histamine on the human histamine H3 receptor: effect of various substitutions at the primary amino function

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Ammonium chloride-promoted four-component synthesis of pyrrolo[3,4-b]pyridin-5-one

1 reference

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Histone deacetylase inhibitors: from bench to clinic

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Molecular modeling studies toward the structural optimization of new cyclopeptide-based HDAC inhibitors modeled on the natural product FR235222.

1 reference

https://pubmed.ncbi.nlm.nih.gov/19475493

12 December 2020

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Epigenetics--an epicenter of gene regulation: histones and histone-modifying enzymes

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Structures of a histone deacetylase homologue bound to the TSA and SAHA inhibitors

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Total synthesis of the eight diastereomers of the syn-anti-syn phytoprostanes F1 types I and II

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Toward selective histone deacetylase inhibitor design: homology modeling, docking studies, and molecular dynamics simulations of human class I histone deacetylases

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Zinc binding in proteins and solution: a simple but accurate nonbonded representation

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https://pubmed.ncbi.nlm.nih.gov/19475493

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Reduced surface: an efficient way to compute molecular surfaces

1 reference

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Synthesis of 7200 small molecules based on a substructural analysis of the histone deacetylase inhibitors trichostatin and trapoxin

1 reference

https://pubmed.ncbi.nlm.nih.gov/19475493

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