(Q40632233)

22 September 2017

title

4-(2-pyridyl)piperazine-1-carboxamides: potent vanilloid receptor 1 antagonists (English)

1 reference

22 September 2017

4-(2-Pyridyl)piperazine-1-carboxamides: potent vanilloid receptor 1 antagonists (English)

1 reference

https://api.crossref.org/works/10.1016/S0960-894X(03)00759-5

13 March 2024

1 reference

https://api.crossref.org/works/10.1016/S0960-894X(03)00759-5

13 March 2024

pharmaceutical science

1 reference

https://api.crossref.org/works/10.1016/S0960-894X(03)00759-5

13 March 2024

1 reference

https://api.crossref.org/works/10.1016/S0960-894X(03)00759-5

13 March 2024

1 reference

https://api.crossref.org/works/10.1016/S0960-894X(03)00759-5

13 March 2024

author name string

Qun Sun

1

1 reference

22 September 2017

Laykea Tafesse

2

1 reference

22 September 2017

Khondaker Islam

3

1 reference

22 September 2017

Xiaoming Zhou

4

1 reference

22 September 2017

Chongwu Zhang

6

1 reference

22 September 2017

Mohamed Hachicha

7

1 reference

22 September 2017

Aniket Patel

9

1 reference

22 September 2017

Yakov Rotshteyn

10

1 reference

22 September 2017

Sam F. Victory

5

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A14505681

13 March 2024

Lori A. Schmid

8

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A14505681

13 March 2024

Kenneth J. Valenzano

11

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A14505681

13 March 2024

Donald J. Kyle

12

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A14505681

13 March 2024

language of work or name

English

0 references

publication date

1 October 2003

1 reference

22 September 2017

20 October 2003

1 reference

National Center for Biotechnology Information

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/esummary.fcgi?db=pubmed&retmode=json&id=14505681

full work available at URL

13 March 2024

https://api.elsevier.com/content/article/PII:S0960894X03007595?httpAccept=text/xml

1 reference

https://api.crossref.org/works/10.1016/S0960-894X(03)00759-5

https://api.elsevier.com/content/article/PII:S0960894X03007595?httpAccept=text/plain

13 March 2024

1 reference

https://api.crossref.org/works/10.1016/S0960-894X(03)00759-5

Bioorganic & Medicinal Chemistry Letters

13 March 2024

published in

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22 September 2017

volume

13

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22 September 2017

issue

20

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22 September 2017

page(s)

3611-3616

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Vanilloid and TRP channels: a family of lipid-gated cation channels.

22 September 2017

cites work

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900759-5

7 January 2021

The capsaicin receptor: a heat-activated ion channel in the pain pathway

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900759-5

7 January 2021

The cloned capsaicin receptor integrates multiple pain-producing stimuli

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900759-5

7 January 2021

Cloning and functional expression of a human orthologue of rat vanilloid receptor-1.

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900759-5

7 January 2021

The ligand that came from within

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900759-5

7 January 2021

Impaired nociception and pain sensation in mice lacking the capsaicin receptor

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900759-5

7 January 2021

Vanilloid receptor-1 is essential for inflammatory thermal hyperalgesia

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900759-5

7 January 2021

Characterization using FLIPR of rat vanilloid receptor (rVR1) pharmacology

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900759-5

7 January 2021

Characterisation using FLIPR of human vanilloid VR1 receptor pharmacology

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900759-5

7 January 2021

The discovery of capsazepine, the first competitive antagonist of the sensory neuron excitants capsaicin and resiniferatoxin

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900759-5

7 January 2021

Attenuation of thermal nociception and hyperalgesia by VR1 blockers

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900759-5

7 January 2021

N-(3-acyloxy-2-benzylpropyl)-N'-dihydroxytetrahydrobenzazepine and tetrahydroisoquinoline thiourea analogues as vanilloid receptor ligands

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900759-5

7 January 2021

N-(4-Tertiarybutylphenyl)-4-(3-chloropyridin-2-yl)tetrahydropyrazine -1(2H)-carbox-amide (BCTC), a Novel, Orally Effective Vanilloid Receptor 1 Antagonist with Analgesic Properties: I. In Vitro Characterization and Pharmacokinetic Properties

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900759-5

7 January 2021

N-(4-Tertiarybutylphenyl)-4-(3-cholorphyridin-2-yl)tetrahydropyrazine -1(2H)-carbox-amide (BCTC), a novel, orally effective vanilloid receptor 1 antagonist with analgesic properties: II. in vivo characterization in rat models of inflammatory and neu

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900759-5

7 January 2021

Identifiers

1 reference

22 September 2017

1 reference