(Q40665061)

English

Tibolone is not converted by human aromatase to 7alpha-methyl-17alpha-ethynylestradiol (7alpha-MEE): analyses with sensitive bioassays for estrogens and androgens and with LC-MSMS.

scientific article published on March 2003

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scholarly article

1 reference

Europe PubMed Central

PubMed publication ID

22 September 2017

Tibolone is not converted by human aromatase to 7alpha-methyl-17alpha-ethynylestradiol (7alpha-MEE): analyses with sensitive bioassays for estrogens and androgens and with LC-MSMS. (English)

1 reference

Europe PubMed Central

PubMed publication ID

22 September 2017

1 reference

based on heuristic

inferred from title

author name string

Marcel E de Gooyer

1

1 reference

Europe PubMed Central

PubMed publication ID

22 September 2017

Hendrika M Oppers-Tiemissen

2

1 reference

Europe PubMed Central

PubMed publication ID

22 September 2017

Dirk Leysen

3

1 reference

Europe PubMed Central

PubMed publication ID

22 September 2017

Herman A M Verheul

4

1 reference

Europe PubMed Central

PubMed publication ID

22 September 2017

Helenius J Kloosterboer

5

1 reference

Europe PubMed Central

PubMed publication ID

22 September 2017

publication date

1 March 2003

1 reference

Europe PubMed Central

PubMed publication ID

22 September 2017

1 reference

Europe PubMed Central

PubMed publication ID

22 September 2017

68

1 reference

Europe PubMed Central

PubMed publication ID

22 September 2017

3

1 reference

Europe PubMed Central

PubMed publication ID

22 September 2017

235-243

1 reference

Europe PubMed Central

PubMed publication ID

22 September 2017

Tibolone: a steroid with a tissue-specific mode of action

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Effects of tibolone and continuous combined hormone replacement therapy on mammographic breast density

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Human endometrial 3 beta-hydroxysteroid dehydrogenase/isomerase can locally reduce intrinsic estrogenic/progestagenic activity ratios of a steroidal drug (Org OD 14)

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Mammographic changes associated with raloxifene and tibolone therapy in postmenopausal women: a prospective study

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Clinical profile of Org OD 14

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The in vivo metabolism of tibolone in animal species

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The in vivo human metabolism of tibolone

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Receptor profiling and endocrine interactions of tibolone

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Reassignment of the absolute configuration of 19-substituted 19-hydroxysteroids and stereomechanism of estrogen biosynthesis

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Studies on the mechanism of estrogen biosynthesis. VI. The stereochemistry of hydrogen elimination at C-2 during aromatization

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Aromatase--a brief overview

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Purification and reconstitution properties of human placental aromatase. A cytochrome P-450-type monooxygenase

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Aromatization of testosterone and 19-nortestosterone by a single enzyme from equine testicular microsomes. Differences from human placental aromatase

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Androgen and 19-norandrogen aromatization by equine and human placental microsomes

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Equine ovarian aromatase: evidence for a species specificity

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Formation and metabolism of 5(10)-estrene-3 beta,17 beta-diol, a novel 19-norandrogen produced by porcine granulosa cells from C19 aromatizable androgens

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Aromatization of 19-norandrogens by porcine Leydig cells

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Aromatization of 7α-Methyl-19-nortestosterone by human placental microsomes in vitro

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Synthesis and aromatization of 19-norandrogens in the stallion testis

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Inhibitor specificity of the placental microsomal oxidase system responsible for the aromatization of epitestosterone (17 alpha-hydroxy-4-androsten-3-one)

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Steroid modulation of aromatase activity in human cultured breast carcinoma cells

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7 January 2021

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In vivo conversion of norethisterone and norethisterone acetate to ethinyl etradiol in postmenopausal women

1 reference

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Formation of ethinylestradiol in postmenopausal women during continuous treatment with a combination of estradiol, estriol and norethisterone acetate

1 reference

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Selection of 19-(ethyldithio)-androst-4-ene-3,17-dione (ORG 30958): A potent aromatase inhibitor in vivo

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1 reference

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1 reference

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Plasma Levels of Adrenocorticotropin and Cortisol in Women Receiving Oral Contraceptive Steroid Treatment*

1 reference

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Differential effects on the androgen status of postmenopausal women treated with tibolone and continuous combined estradiol and norethindrone acetate replacement therapy

1 reference

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[Estrogenic effects after 14-days administration of 0.06 mg ethinyl estradiol in postmenopausal women]

1 reference

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Identifiers

10.1016/S0039-128X(02)00184-8

1 reference

Europe PubMed Central

PubMed publication ID

22 September 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

22 September 2017

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