(Q40801922)

23 September 2017

title

Action of bicyclic isoxazole GABA analogues on GABA transporters and its relation to anticonvulsant activity (English)

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23 September 2017

Bolvig T

1

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23 September 2017

Larsson OM

2

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23 September 2017

Pickering DS

3

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23 September 2017

Nelson N

4

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23 September 2017

Falch E

5

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23 September 2017

Krogsgaard-Larsen P

6

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23 September 2017

Schousboe A

7

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23 September 2017

language of work or name

English

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publication date

1 June 1999

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European Journal of Pharmacology

23 September 2017

published in

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23 September 2017

volume

375

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23 September 2017

issue

1-3

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23 September 2017

page(s)

367-374

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Orally active and potent inhibitors of gamma-aminobutyric acid uptake

23 September 2017

cites work

1 reference

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GABA transporter heterogeneity: pharmacology and cellular localization

7 January 2021

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Tiagabine, SK&F 89976-A, CI-966, and NNC-711 are selective for the cloned GABA transporter GAT-1.

7 January 2021

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(R)-N-[4,4-bis(3-methyl-2-thienyl)but-3-en-1-yl]nipecotic acid binds with high affinity to the brain gamma-aminobutyric acid uptake carrier

7 January 2021

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High-efficiency transformation of mammalian cells by plasmid DNA

7 January 2021

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Anticonvulsant activity of GABA uptake inhibitors and their prodrugs following central or systemic administration

7 January 2021

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Design, synthesis and evaluation of substituted triarylnipecotic acid derivatives as GABA uptake inhibitors: identification of a ligand with moderate affinity and selectivity for the cloned human GABA transporter GAT-3.

7 January 2021

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Anticonvulsant activity of intracerebroventricularly administered glial GABA uptake inhibitors and other GABAmimetics in chemical seizure models

7 January 2021

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Anticonvulsant activity of the glial GABA uptake inhibitor, THAO, in chemical seizures

7 January 2021

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Inhibition of the uptake of GABA and related amino acids in rat brain slices by the optical isomers of nipecotic acid

7 January 2021

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Differential effects of nipecotic acid and 4,5,6,7-tetrahydroisoxazolo[4,5-c]pyridin-3-ol on extracellular gamma-aminobutyrate levels in rat thalamus.

7 January 2021

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GABA uptake inhibitors: relevance to antiepileptic drug research

7 January 2021

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GABAA receptor agonists, partial agonists, and antagonists. Design and therapeutic prospects

7 January 2021

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Comparison between (RS)-nipecotic acid and GABA transport in cultured astrocytes: Coupling with two sodium ions

7 January 2021

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Ion dependency of uptake and release of GABA and (RS)-nipecotic acid studied in cultured mouse brain cortex neurons

7 January 2021

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Ontogenetic development of glutamate and GABA metabolizing enzymes in cultured cerebral cortex interneurons and in cerebral cortex in vivo.

7 January 2021

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Uptake of GABA and nipecotic acid in astrocytes and neurons in primary cultures: changes in the sodium coupling ratio during differentiation.

7 January 2021

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A family of genes encoding neurotransmitter transporters

7 January 2021

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Characterization of tiagabine (NO-328), a new potent and selective GABA uptake inhibitor

7 January 2021

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Transient expression shows ligand gating and allosteric potentiation of GABAA receptor subunits

7 January 2021

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Uptake and metabolism of GABA in astrocytes cultured from dissociated mouse brain hemispheres

7 January 2021

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Tissue distribution, metabolism, anticonvulsant efficacy and effect on brain amino acid levels of the glia-selective gamma-aminobutyric acid transport inhibitor 4,5,6,7-tetrahydroisoxazolo[4,5-c]pyridin-3-ol in mice and chicks.

7 January 2021

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1-(3-(9H-carbazol-9-yl)-1-propyl)-4-(2-methoxyphenyl)-4-piperidinol, a novel subtype selective inhibitor of the mouse type II GABA-transporter

7 January 2021

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Transporter explosion: update on uptake

7 January 2021

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Anticonvulsant activity of the gamma-aminobutyric acid uptake inhibitor N-4,4-diphenyl-3-butenyl-4,5,6,7-tetrahydroisoxazolo[4,5-c]pyridin-3-ol

7 January 2021

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Transport and Metabolism of Glutamate and Gaba in Neurons and Glial Cells

7 January 2021

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inferred from DOI database lookup

7 January 2021

based on heuristic

Identifiers

DOI

10.1016/S0014-2999(99)00263-0

1 reference

23 September 2017

1 reference