(Q40816595)

24 September 2017

Ivermectin, an unconventional agonist of the glycine receptor chloride channel (English)

1 reference

24 September 2017

0 references

Shan Q

1

1 reference

24 September 2017

Haddrill JL

series ordinal

2

1 reference

24 September 2017

Lynch JW

series ordinal

3

1 reference

24 September 2017

language of work or name

English

0 references

publication date

18 January 2001

1 reference

Journal of Biological Chemistry

24 September 2017

1 reference

24 September 2017

276

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24 September 2017

16

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24 September 2017

12556-12564

1 reference

The Chemistry and Pharmacology of Avermectins

24 September 2017

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Treatment of onchocerciasis

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

The role of albendazole in programmes to eliminate lymphatic filariasis

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Cloning of an avermectin-sensitive glutamate-gated chloride channel from Caenorhabditis elegans

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Identification of a Drosophila melanogaster glutamate-gated chloride channel sensitive to the antiparasitic agent avermectin

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Genetic and biochemical evidence for a novel avermectin-sensitive chloride channel in Caenorhabditis elegans. Isolation and characterization.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Drug-resistant Drosophila indicate glutamate-gated chloride channels are targets for the antiparasitics nodulisporic acid and ivermectin.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Anticonvulsant effects of ivermectin in genetically-epileptic chickens.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

The strychnine-binding subunit of the glycine receptor shows homology with nicotinic acetylcholine receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Sequence and functional expression of the GABA A receptor shows a ligand-gated receptor super-family.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Primary structure and functional expression of the 5HT3 receptor, a serotonin-gated ion channel

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Evolutionary relationship of the ligand-gated ion channels and the avermectin-sensitive, glutamate-gated chloride channels.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Effect of ivermectin on gamma-aminobutyric acid-induced chloride currents in mouse hippocampal embryonic neurones.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Actions of anaesthetics and avermectin on GABAA chloride channels in mammalian dorsal root ganglion neurones

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Activation of rat recombinant alpha(1)beta(2)gamma(2S) GABA(A) receptor by the insecticide ivermectin.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Avermectin B1a inhibits the binding of strychnine to the glycine receptor of rat spinal cord

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

High-efficiency transformation of mammalian cells by plasmid DNA

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Conserved quaternary structure of ligand-gated ion channels: the postsynaptic glycine receptor is a pentamer

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Strychnine binding associated with glycine receptors of the central nervous system

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Antagonism of ligand-gated ion channel receptors: two domains of the glycine receptor alpha subunit form the strychnine-binding site

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Distinct agonist- and antagonist-binding sites on the glycine receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Mutations affecting the glycine receptor agonist transduction mechanism convert the competitive antagonist, picrotoxin, into an allosteric potentiator.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Modulation by zinc ions of native rat and recombinant human inhibitory glycine receptors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

A single amino acid exchange alters the pharmacology of neonatal rat glycine receptor subunit.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Mutation of glycine receptor subunit creates beta-alanine receptor responsive to GABA.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Mutations in the alpha 1 subunit of the inhibitory glycine receptor cause the dominant neurologic disorder, hyperekplexia

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Mutation of an arginine residue in the human glycine receptor transforms beta-alanine and taurine from agonists into competitive antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Identification of intracellular and extracellular domains mediating signal transduction in the inhibitory glycine receptor chloride channel

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

Mild KCC2 Hypofunction Causes Inconspicuous Chloride Dysregulation that Degrades Neural Coding

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M011264200

21 January 2018

Identifiers

DOI

10.1074/JBC.M011264200

1 reference

24 September 2017

1 reference