(Q41243374)

28 September 2017

title

Pharmacological properties of recombinant "diazepam-insensitive" GABAA receptors (English)

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28 September 2017

0 references

Gunnersen D

1

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28 September 2017

Kaufman CM

series ordinal

2

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28 September 2017

Skolnick P

series ordinal

3

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28 September 2017

publication date

1 January 1996

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28 September 2017

number of pages

8

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based on heuristic

inferred from page(s)

published in

Neuropharmacology

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28 September 2017

volume

35

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28 September 2017

issue

9-10

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28 September 2017

page(s)

1307-1314

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Beta-carbolines: synthesis and neurochemical and pharmacological actions on brain benzodiazepine receptors

28 September 2017

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Triazolam is more efficacious than diazepam in a broad spectrum of recombinant GABAA receptors

7 January 2021

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Synthesis and evaluation of imidazo[1,5-a][1,4]benzodiazepine esters with high affinities and selectivities at "diazepam-insensitive" benzodiazepine receptors

7 January 2021

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Contribution of "diazepam-insensitive" GABAA receptors to the alcohol antagonist properties of Ro 15-4513 and related imidazobenzodiazepines

7 January 2021

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Characterization of diazepam-insensitive [3H]Ro 15-4513 binding in rodent brain and cultured cerebellar neuronal cells

7 January 2021

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Novel GABAA receptor alpha subunit is expressed only in cerebellar granule cells

7 January 2021

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The subunit composition of a GABAA/benzodiazepine receptor from rat cerebellum.

7 January 2021

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Current potentiation by diazepam but not GABA sensitivity is determined by a single histidine residue.

7 January 2021

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Natural mutation of GABAA receptor alpha 6 subunit alters benzodiazepine affinity but not allosteric GABA effects

7 January 2021

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Substrate specificity of diazepan-insensitive cerebellar [3H] Ro 15-4513 binding sites

7 January 2021

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Benzodiazepine-induced motor impairment linked to point mutation in cerebellar GABAA receptor.

7 January 2021

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Antagonism of the intoxicating effects of ethanol by the potent benzodiazepine receptor ligand Ro 19-4603

7 January 2021

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Cerebellar GABAA receptor selective for a behavioural alcohol antagonist

7 January 2021

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Diazepam-insensitive [3H]Ro 15-4513 binding in intact cultured cerebellar granule cells.

7 January 2021

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Importance of a novel GABAA receptor subunit for benzodiazepine pharmacology

7 January 2021

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Photoaffinity labeling of benzodiazepine receptor proteins with the partial inverse agonist [3H]Ro 15-4513: a biochemical and autoradiographic study

7 January 2021

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7 January 2021

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Ethanol stimulates gamma-aminobutyric acid receptor-mediated chloride transport in rat brain synaptoneurosomes

7 January 2021

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Ro15-4513 differentially affects ethanol-induced hypnosis and hypothermia.

7 January 2021

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Diazepam sensitivity of the binding of an imidazobenzodiazepine, [3H]Ro 15-4513, in cerebellar membranes from two rat lines developed for high and low alcohol sensitivity

7 January 2021

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Functional properties of recombinant rat GABAA receptors depend upon subunit composition

7 January 2021

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Four amino acid exchanges convert a diazepam-insensitive, inverse agonist-preferring GABAA receptor into a diazepam-preferring GABAA receptor

7 January 2021

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Cloning, pharmacological characteristics and expression pattern of the rat GABAA receptor alpha 4 subunit

7 January 2021

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The distribution of 13 GABAA receptor subunit mRNAs in the rat brain. I. Telencephalon, diencephalon, mesencephalon

7 January 2021

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High affinity ligands for ‘diazepam-insensitive’ benzodiazepine receptors

7 January 2021

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Ro 15-4513 binding to GABAA receptors: subunit composition determines ligand efficacy

7 January 2021

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Labelling of diazepam-sensitive and -insensitive benzodiazepine receptors with [3H]tert-butyl-8-chloro-5,6-dihydro-5-methyl-6-oxo-4H-imidazo [1,5-a][1,4]benzodiazepine 3-carboxylate (ZG-63).

7 January 2021

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Synthetic and computer-assisted analysis of the structural requirements for selective, high-affinity ligand binding to diazepam-insensitive benzodiazepine receptors.

7 January 2021

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Cloning and characterization of the human GABAA receptor alpha 4 subunit: identification of a unique diazepam-insensitive binding site

7 January 2021

1 reference

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Sequence and expression of a novel GABAA receptor alpha subunit

7 January 2021

1 reference

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Synthesis of novel imidazobenzodiazepines as probes of the pharmacophore for "diazepam-insensitive" GABAA receptors

7 January 2021

1 reference

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10.1016/S0028-3908(96)00054-8

7 January 2021

Identifiers

DOI

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release_tg6xj6kak5ah3cl6cdspxfejl4

28 September 2017

Fatcat ID

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Fatcat

https://api.fatcat.wiki/v0/release/tg6xj6kak5ah3cl6cdspxfejl4

mapped directly with Wikidata item

24 November 2022

based on heuristic

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