(Q41540958)

2 October 2017

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title

Prodrug strategies based on intramolecular cyclization reactions (English)

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2 October 2017

Shan D

1

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2 October 2017

Nicolaou MG

series ordinal

2

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2 October 2017

Borchardt RT

series ordinal

3

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2 October 2017

Wang B

series ordinal

4

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2 October 2017

language of work or name

English

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publication date

1 July 1997

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Journal of Pharmaceutical Sciences

2 October 2017

published in

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2 October 2017

volume

86

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2 October 2017

issue

7

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2 October 2017

page(s)

765-767

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Pilocarpine prodrugs. II. Synthesis, stability, bioconversion, and physicochemical properties of sequentially labile pilocarpine acid diesters

2 October 2017

cites work

1 reference

7 January 2021

Potent in vitro and in vivo inhibitors of platelet aggregation based upon the Arg-Gly-Asp-Phe sequence of fibrinogen. A proposal on the nature of the binding interaction between the Arg-guanidine of RGDX mimetics and the platelet GP IIb-IIIa recepto

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7 January 2021

Discovery of an orally active non-peptide fibrinogen receptor antagonist

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7 January 2021

Prodrugs of peptides. 18. Synthesis and evaluation of various esters of desmopressin (dDAVP).

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7 January 2021

Prodrugs of peptides and proteins for improved formulation and delivery

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7 January 2021

Cyclization-activated prodrugs. Basic esters of 5-bromo-2'-deoxyuridine

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7 January 2021

Cyclization-activated prodrugs. Basic carbamates of 4-hydroxyanisole

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7 January 2021

Relationships between structure and kinetics of cyclization of 2-aminoaryl amides: potential prodrugs of cyclization-activated aromatic mustards

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7 January 2021

Cyclization-activated prodrugs: N-(substituted 2-hydroxyphenyl and 2-hydroxypropyl)carbamates based on ring-opened derivatives of active benzoxazolones and oxazolidinones as mutual prodrugs of acetaminophen.

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7 January 2021

Stereopopulation control. I. Rate enhancement in the lactonizations of o-hydroxyhydrocinnamic acids

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7 January 2021

Amine prodrugs which utilize hydroxy amide lactonization. I. A potential redox-sensitive amide prodrug

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7 January 2021

Amine prodrugs which utilize hydroxy amide lactonization. II. A potential esterase-sensitive amide prodrug

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7 January 2021

Synthesis of a Novel Esterase-Sensitive Cyclic Prodrug System for Peptides That Utilizes a “Trimethyl Lock”-Facilitated Lactonization Reaction

1 reference

7 January 2021

Esterase-sensitive cyclic prodrugs of peptides: evaluation of a phenylpropionic acid promoiety in a model hexapeptide.

1 reference

7 January 2021

Facilitated Intramolecular Conjugate Addition of Amides of 3-(3',6'-Dioxo-2',4'-dimethyl-1',4'-cyclohexadienyl)-3,3-dimethylpropionic Acid. 2. Kinetics of Degradation

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7 January 2021

Orally active water-soluble N,O-acyl transfer products of a beta,gamma-bishydroxyl amide containing renin inhibitor

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7 January 2021

The importance of structural factors on the rate and the extent of N,O-acyl migration in cyclic and linear peptides

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7 January 2021

Chemical feasibility studies of a potential coumarin-based prodrug system

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7 January 2021

Coumarin-based prodrugs 2. Synthesis and bioreversibility studies of an esterase-sensitive cyclic prodrug of dadle, an opioid peptide

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7 January 2021

Identification of two related pentapeptides from the brain with potent opiate agonist activity

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7 January 2021

Identifiers

DOI

10.1021/JS970069D

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2 October 2017

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