(Q41972819)

English

Characterization of the endothelin receptor selective agonist, BQ3020 and antagonists BQ123, FR139317, BQ788, 50235, Ro462005 and bosentan in the heart.

scientific article published on February 1996

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scholarly article

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8821534%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

Characterization of the endothelin receptor selective agonist, BQ3020 and antagonists BQ123, FR139317, BQ788, 50235, Ro462005 and bosentan in the heart (English)

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8821534%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

Anthony P Davenport

2

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8821534%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

author name string

M G Peter

1

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8821534%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

language of work or name

0 references

publication date

1 February 1996

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8821534%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

British Journal of Pharmacology

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8821534%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

117

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8821534%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

3

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8821534%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

455-462

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8821534%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

Distinct subdomains of human endothelin receptors determine their selectivity to endothelinA-selective antagonist and endothelinB-selective agonists

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

The human endothelin-B receptor gene. Structural organization and chromosomal assignment

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

The endothelin ETA receptor-specific effect of 50-235, a nonpeptide endothelin antagonist

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Stable expression of human endothelin receptors ETA and ETB by transfected baby hamster kidney cells

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Species differences in the binding characteristics of [125I]IRL-1620, a potent agonist specific for endothelin-B receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Evidence for heterogeneity of endothelin receptor distribution in human coronary artery

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Biochemical and pharmacological profile of a potent and selective endothelin B-receptor antagonist, BQ-788.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Is endothelin-induced vasoconstriction mediated only by ETA receptors in humans?

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Effect of a nonselective endothelin antagonist on vascular remodeling in deoxycorticosterone acetate-salt hypertensive rats. Evidence for a role of endothelin in vascular hypertrophy

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Pharmacological characterization of bosentan, a new potent orally active nonpeptide endothelin receptor antagonist

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Selectivity of [125I]-PD151242 for human, rat and porcine endothelin ETA receptors in the heart.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Role of endogenous endothelin in myocardial and coronary endothelial injury after ischaemia and reperfusion in rats: studies with bosentan, a mixed ETA-ETB antagonist

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Synergistic inhibition by BQ-123 and BQ-788 of endothelin-1-induced contractions of the rabbit pulmonary artery

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Pharmacological differences between rat and human endothelin B receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

ETA receptor-mediated constrictor responses to endothelin peptides in human blood vessels in vitro

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Endothelin ETA and ETB mRNA and receptors expressed by smooth muscle in the human vasculature: majority of the ETA sub-type

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Molecular and functional characterization of the non-isopeptide-selective ETB receptor in endothelial cells. Receptor coupling to nitric oxide synthase

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Human endothelin receptors characterized using reverse transcriptase-polymerase chain reaction, in situ hybridization, and subtype-selective ligands BQ123 and BQ3020: evidence for expression of ETB receptors in human vascular smooth muscle.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

LIGAND: A versatile computerized approach for characterization of ligand-binding systems

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Positive inotropic action of novel vasoconstrictor peptide endothelin on guinea pig atria

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Cardiovascular effects of endothelin in dogs: positive inotropic action in vivo

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Localization of endothelin-1 (ET-1), ET-2, and ET-3, mouse VIC, and sarafotoxin S6b binding sites in mammalian heart and kidney

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Cloning and characterization of cDNA encoding human a-type endothelin receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Tissue specificity of endothelin binding sites

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

[Ala1,3,11,15]endothelin-1 analogs with ETB agonistic activity.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Molecular cloning of a non-isopeptide-selective human endothelin receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

A novel radioligand [125I]BQ-3020 selective for endothelin (ETB) receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

A novel non-peptide endothelin antagonist isolated from bayberry, Myrica cerifera

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Molecular cloning and characterization of the major endothelin receptor subtype in porcine cerebellum

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Biological profiles of highly potent novel endothelin antagonists selective for the ETA receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

5 June 2018

Effects of an ET1-receptor antagonist, FR139317, on regional haemodynamic responses to endothelin-1 and [Ala11,15]Ac-endothelin-1 (6-21) in conscious rats.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

18 August 2018

An endothelin B receptor-selective antagonist: IRL 1038, [Cys11-Cys15]-endothelin-1(11-21)

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

18 August 2018

[125I]-PD151242: a selective radioligand for human ETA receptors

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1996.TB15212.X

21 January 2018

Davenport and Maguire reply

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1996.TB15212.X

21 January 2018

Effects of bosentan (Ro 47-0203), an ETA-, ETB-receptor antagonist, on regional haemodynamic responses to endothelins in conscious rats

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1996.TB15212.X

21 January 2018

Anatomical localization and pharmacological activity of mature endothelins and their precursors in human vascular tissue

2 references

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1996.TB15212.X

21 January 2018

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

3 November 2018

Novel ligands BQ123 and BQ3020 characterize endothelin receptor subtypes ETA and ETB in human kidney

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1996.TB15212.X

21 January 2018

Characterization and localization of endothelin receptor subtypes in the human atrioventricular conducting system and myocardium

2 references

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1996.TB15212.X

21 January 2018

https://pubmed.ncbi.nlm.nih.gov/8821534

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The endothelin receptor antagonist, BQ-123, inhibits angiotensin II-induced contractions in rabbit aorta

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1996.TB15212.X

21 January 2018

Characterization of endothelin isoforms in human heart: endothelin-2 demonstrated

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

3 November 2018

Autoradiographical localization of binding sites for porcine [125I]endothelin-1 in humans, pigs, and rats: functional relevance in humans

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909322

3 November 2018

Pathophysiological role of endothelin revealed by the first orally active endothelin receptor antagonist

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1996.TB15212.X

21 January 2018

Endothelin receptors in the human coronary artery, ventricle and atrium

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1996.TB15212.X

21 January 2018

Occurrence, specific binding sites and functional effects of endothelin in human cardiopulmonary tissue

1 reference

https://pubmed.ncbi.nlm.nih.gov/8821534

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Effects of endothelin on intracellular Ca2+ and contractility in single ventricular myocytes from the ferret and human

1 reference

https://pubmed.ncbi.nlm.nih.gov/8821534

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Endothelin receptors in cultured adult rat cardiac fibroblasts

1 reference

https://pubmed.ncbi.nlm.nih.gov/8821534

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

An endothelin B receptor-selective antagonist: IRL 1038, [Cys11- Cys15]-endothelin-1(11-21)

1 reference

https://pubmed.ncbi.nlm.nih.gov/8821534

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Cyclic hexapeptide endothelin receptor antagonists highly potent for both receptor subtypes ETA and ETB

1 reference

https://pubmed.ncbi.nlm.nih.gov/8821534

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Localization of endothelin immunoreactivity and demonstration of constrictory endothelin-A receptors in human coronary arteries and veins

1 reference

https://pubmed.ncbi.nlm.nih.gov/8821534

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Role of endothelin in the maintenance of blood pressure in conscious rats with chronic heart failure. Acute effects of the endothelin receptor antagonist Ro 47-0203 (bosentan)

1 reference

https://pubmed.ncbi.nlm.nih.gov/8821534

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

A practical computer-based approach to the analysis of radioligand binding experiments

1 reference

https://pubmed.ncbi.nlm.nih.gov/8821534

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Endothelin is a positive inotropic agent in human and rat heart in vitro

1 reference

https://pubmed.ncbi.nlm.nih.gov/8821534

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Endothelin ETA receptor antagonist, BQ-123, blocks the vasoconstriction induced by sarafotoxin 6b in the heart but not in other vascular beds

1 reference

https://pubmed.ncbi.nlm.nih.gov/8821534

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Endothelin receptors in human coronary arteries

1 reference

https://pubmed.ncbi.nlm.nih.gov/8821534

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Subtype selectivity of a novel endothelin antagonist, FR139317, for the two endothelin receptors in transfected Chinese hamster ovary cells

1 reference

https://pubmed.ncbi.nlm.nih.gov/8821534

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1111/J.1476-5381.1996.TB15212.X

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8821534%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8821534%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8821534%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

ResearchGate publication ID

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