(Q42239514)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27200176%20AND%20SRC:MED&resulttype=core&format=json

2 April 2020

title

Allosteric Glutaminase Inhibitors Based on a 1,4-Di(5-amino-1,3,4-thiadiazol-2-yl)butane Scaffold (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27200176%20AND%20SRC:MED&resulttype=core&format=json

2 April 2020

1 reference

8

1 reference

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2 April 2020

author name string

Sarah C Zimmermann

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27200176%20AND%20SRC:MED&resulttype=core&format=json

2 April 2020

Emily F Wolf

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27200176%20AND%20SRC:MED&resulttype=core&format=json

2 April 2020

Andrew Luu

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27200176%20AND%20SRC:MED&resulttype=core&format=json

2 April 2020

Ajit G Thomas

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27200176%20AND%20SRC:MED&resulttype=core&format=json

2 April 2020

Marigo Stathis

5

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27200176%20AND%20SRC:MED&resulttype=core&format=json

2 April 2020

Brad Poore

6

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27200176%20AND%20SRC:MED&resulttype=core&format=json

2 April 2020

Christopher Nguyen

7

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27200176%20AND%20SRC:MED&resulttype=core&format=json

2 April 2020

Camilo Rojas

9

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27200176%20AND%20SRC:MED&resulttype=core&format=json

2 April 2020

Barbara S Slusher

10

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27200176%20AND%20SRC:MED&resulttype=core&format=json

2 April 2020

Takashi Tsukamoto

11

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27200176%20AND%20SRC:MED&resulttype=core&format=json

2 April 2020

publication date

13 March 2016

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27200176%20AND%20SRC:MED&resulttype=core&format=json

ACS Medicinal Chemistry Letters

2 April 2020

published in

1 reference

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2 April 2020

volume

7

1 reference

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2 April 2020

issue

5

1 reference

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2 April 2020

page(s)

520-524

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27200176%20AND%20SRC:MED&resulttype=core&format=json

Targeted inhibition of tumor-specific glutaminase diminishes cell-autonomous tumorigenesis.

2 April 2020

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4868099

Antitumor activity of the glutaminase inhibitor CB-839 in triple-negative breast cancer

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4868099

Design, synthesis, and pharmacological evaluation of bis-2-(5-phenylacetamido-1,2,4-thiadiazol-2-yl)ethyl sulfide 3 (BPTES) analogs as glutaminase inhibitors.

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4868099

Glutaminase isoenzymes as key regulators in metabolic and oxidative stress against cancer.

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4868099

Analysis of glutamine dependency in non-small cell lung cancer: GLS1 splice variant GAC is essential for cancer cell growth

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4868099

Structural basis for the allosteric inhibitory mechanism of human kidney-type glutaminase (KGA) and its regulation by Raf-Mek-Erk signaling in cancer cell metabolism

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4868099

Dibenzophenanthridines as inhibitors of glutaminase C and cancer cell proliferation.

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4868099

Full-length human glutaminase in complex with an allosteric inhibitor

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4868099

Targeting mitochondrial glutaminase activity inhibits oncogenic transformation

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4868099

Novel mechanism of inhibition of rat kidney-type glutaminase by bis-2-(5-phenylacetamido-1,2,4-thiadiazol-2-yl)ethyl sulfide (BPTES)

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4868099

Regulation of glutaminase activity and glutamine metabolism

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4868099

Metabolism and action of amino acid analog anti-cancer agents

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4868099

Interactions of N-{[2-(4-phenyl-piperazin-1-yl)-ethyl]-phenyl}-2-aryl-2-yl-acetamides and 1-{[2-(4-phenyl-piperazin-1-yl)-ethyl]-phenyl}-3-aryl-2-yl-ureas with dopamine D2 and 5-hydroxytryptamine 5HT(1A) receptors.

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4868099

10.1021/ACSMEDCHEMLETT.6B00060

17 August 2018

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27200176%20AND%20SRC:MED&resulttype=core&format=json

release_4djves6elreyzfbmhjrhmafo6m

2 April 2020

Fatcat ID

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/4djves6elreyzfbmhjrhmafo6m

mapped directly with Wikidata item

24 November 2022

based on heuristic

1 reference

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2 April 2020

PubMed publication ID

27200176

1 reference