(Q43264679)

English

5-HT(1A) receptor agonist-antagonist binding affinity difference as a measure of intrinsic activity in recombinant and native tissue systems

scientific article published in July 2000

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scholarly article

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

5-HT(1A) receptor agonist-antagonist binding affinity difference as a measure of intrinsic activity in recombinant and native tissue systems (English)

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

author name string

J Watson

1

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

L Collin

2

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

M Ho

3

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

G Riley

4

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

C Scott

5

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

J V Selkirk

6

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

G W Price

7

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

language of work or name

0 references

publication date

1 July 2000

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

British Journal of Pharmacology

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

130

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

5

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

1108-1114

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

Relationships between ligand affinities for the cerebellar cannabinoid receptor CB1 and the induction of GDP/GTP exchange.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1572157

25 May 2018

High-affinity agonist binding correlates with efficacy (intrinsic activity) at the human serotonin 5-HT2A and 5-HT2C receptors: evidence favoring the ternary complex and two-state models of agonist action

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1572157

25 May 2018

Functional effects of the muscarinic receptor agonist, xanomeline, at 5-HT1 and 5-HT2 receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1572157

25 May 2018

SB 202026: a novel muscarinic partial agonist with functional selectivity for M1 receptors.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1572157

25 May 2018

Human 5-HT1 receptor subtypes exhibit distinct G protein coupling behaviors in membranes from Sf9 cells

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1572157

25 May 2018

New 5-HT1A receptor antagonist: [3H]p-MPPF.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1572157

25 May 2018

A mutation-induced activated state of the beta 2-adrenergic receptor. Extending the ternary complex model

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1572157

25 May 2018

The two-state model of receptor activation

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1572157

25 May 2018

Differential regulation of high-affinity agonist binding to muscarinic sites in the rat heart, cerebellum, and cerebral cortex.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1572157

25 May 2018

A ternary complex model explains the agonist-specific binding properties of the adenylate cyclase-coupled beta-adrenergic receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1572157

25 May 2018

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1572157

25 May 2018

Relative affinities of drugs acting at cholinoceptors in displacing agonist and antagonist radioligands: the NMS/Oxo-M ratio as an index of efficacy at cortical muscarinic receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1572157

25 May 2018

A1 adenosine receptor-G protein coupling in bovine brain membranes: effects of guanine nucleotides, salt, and solubilization

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1572157

25 May 2018

Species differences in the distribution of central 5-HT1 binding sites: a comparative autoradiographic study between rat and guinea pig

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1572157

25 May 2018

Intrinsic activity determinations at the dopamine D2 guanine nucleotide-binding protein-coupled receptor: utilization of receptor state binding affinities

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1572157

25 May 2018

The binding of agonists to brain muscarinic receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1572157

25 May 2018

Evaluation of an agonist index: affinity ratio for compounds active on muscarinic cholinergic M2 receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1572157

15 August 2018

Differential receptor-G-protein coupling evoked by dissimilar cannabinoid receptor agonists.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1572157

15 August 2018

Evidence for the stabilisation of the high-affinity state of beta-adrenoceptors by an endogenous factor in rat brain

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1572157

15 August 2018

Correlation between low/high affinity ratios for 5-HT(1A) receptors and intrinsic activity

1 reference

https://pubmed.ncbi.nlm.nih.gov/10882396

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The character of the muscarinic receptors in different regions of the rat brain

1 reference

https://pubmed.ncbi.nlm.nih.gov/10882396

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Pharmacological characterisation of the 5-HT1A serotonin receptor using the agonist [3H]8-OH-DPAT, and the antagonist [3H]spiperone

1 reference

https://pubmed.ncbi.nlm.nih.gov/10882396

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Species differences in A1 adenosine receptor/G protein coupling: identification of a membrane protein that stabilizes the association of the receptor/G protein complex

1 reference

https://pubmed.ncbi.nlm.nih.gov/10882396

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1038/SJ.BJP.0703394

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

release_6mxulr3sybfahfzokudje5v2oq

1 reference

https://api.fatcat.wiki/v0/release/6mxulr3sybfahfzokudje5v2oq

24 November 2022

based on heuristic

mapped directly with Wikidata item

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

ResearchGate publication ID

0 references

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