(Q43732266)

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Benzamide bioisosteres incorporating dihydroheteroazole substructures: EPC synthesis and SAR leading to a selective dopamine D4 receptor partial agonist (FAUC 179).

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Europe PubMed Central

PubMed publication ID

26 November 2017

Benzamide bioisosteres incorporating dihydroheteroazole substructures: EPC synthesis and SAR leading to a selective dopamine D4 receptor partial agonist (FAUC 179). (English)

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Europe PubMed Central

PubMed publication ID

26 November 2017

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3

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26 November 2017

author name string

Einsiedel J

1

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26 November 2017

Hübner H

2

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26 November 2017

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publication date

1 September 2001

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26 November 2017

Bioorganic & Medicinal Chemistry Letters

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26 November 2017

11

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26 November 2017

18

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26 November 2017

2533-2536

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26 November 2017

Cloning of the gene for a human dopamine D4 receptor with high affinity for the antipsychotic clozapine

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Evidence for linkage of a tandem duplication polymorphism upstream of the dopamine D4 receptor gene (DRD4) with attention deficit hyperactivity disorder (ADHD).

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A hypervariable segment in the human dopamine receptor D4 (DRD4) gene.

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Substituted [(4-phenylpiperazinyl)-methyl]benzamides: selective dopamine D4 agonists

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Cyanoindole derivatives as highly selective dopamine D(4) receptor partial agonists: solid-phase synthesis, binding assays, and functional experiments

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2-Phenyl-4(5)-[[4-(pyrimidin-2-yl)piperazin-1-yl]methyl]imidazole. A highly selective antagonist at cloned human D4 receptors

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NGD 94-1 as an agonist at human recombinant dopamine D4.4 receptors expressed in HEK293 cells

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Current and novel approaches to the drug treatment of schizophrenia

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Receptor density as a factor governing the efficacy of the dopamine D4 receptor ligands, L-745,870 and U-101958 at human recombinant D4.4 receptors expressed in CHO cells

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Phenyloxazoles and phenylthiazoles as benzamide bioisosteres: synthesis and dopamine receptor binding profiles

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The reactions of an N-sulfonylamine inner salt

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Indole Grignard reaction. III. Synthesis, crystal structure, and analgesic activity of (R)- and (S)-3-amino-2,3,4,9-tetrahydrothiopyrano[2,3-b]indoles

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Aryloxyacetamidines and 2-(aryloxymethyl)-imidazolines

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Pharmacology of human dopamine D3 receptor expressed in a mammalian cell line: comparison with D2 receptor

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Conjugated enynes as nonaromatic catechol bioisosteres: synthesis, binding experiments, and computational studies of novel dopamine receptor agonists recognizing preferentially the D(3) subtype

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Identifiers

10.1016/S0960-894X(01)00484-X

1 reference

Europe PubMed Central

PubMed publication ID

26 November 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

26 November 2017

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