(Q43797338)

26 November 2017

title

Morphine-6beta-glucuronide and morphine-3-glucuronide, opioid receptor agonists with different potencies (English)

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26 November 2017

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C Ulens

1

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26 November 2017

L Baker

2

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26 November 2017

A Ratka

3

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26 November 2017

D Waumans

4

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26 November 2017

J Tytgat

5

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26 November 2017

language of work or name

English

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publication date

1 November 2001

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26 November 2017

published in

Biochemical Pharmacology

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26 November 2017

volume

62

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26 November 2017

issue

9

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26 November 2017

page(s)

1273-1282

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Morphine-6-glucuronide: analgesic effects and receptor binding profile in rats

26 November 2017

cites work

1 reference

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Morphine-6-glucuronide, a potent mu agonist.

7 January 2021

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Morphine-6-glucuronide has high affinity for the opioid receptor

7 January 2021

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Enhanced binding of morphine and nalorphine to opioid delta receptor by glucuronate and sulfate conjugations at the 6-position

7 January 2021

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Properties of Opiate-Receptor Binding in Rat Brain

7 January 2021

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Mu receptor binding of some commonly used opioids and their metabolites

7 January 2021

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Affinity profiles of morphine, codeine, dihydrocodeine and their glucuronides at opioid receptor subtypes

7 January 2021

1 reference

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The disposition of morphine and its 3- and 6-glucuronide metabolites in humans and animals, and the importance of the metabolites to the pharmacological effects of morphine.

7 January 2021

1 reference

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Effects of morphine and its metabolites on opiate receptor binding, cAMP formation and [3H]noradrenaline release from SH-SY5Y cells

7 January 2021

1 reference

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the apparent affinity of morphine-3-glucuronide at μ1-opioid receptors results from morphine contamination: demonstration using HPLC and radioligand binding

7 January 2021

1 reference

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Morphine-6-O-beta-D-glucuronide but not morphine-3-O-beta-D-glucuronide binds to mu-, delta- and kappa- specific opioid binding sites in cerebral membranes

7 January 2021

1 reference

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Differential blockade of morphine and morphine-6 beta-glucuronide analgesia by antisense oligodeoxynucleotides directed against MOR-1 and G-protein alpha subunits in rats

7 January 2021

1 reference

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Antisense mapping the MOR-1 opioid receptor: evidence for alternative splicing and a novel morphine-6 beta-glucuronide receptor

7 January 2021

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Novel receptor mechanisms for heroin and morphine-6 beta-glucuronide analgesia.

7 January 2021

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Cloning of a delta opioid receptor by functional expression

7 January 2021

1 reference

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The delta-opioid receptor: isolation of a cDNA by expression cloning and pharmacological characterization

7 January 2021

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mu opiate receptor: cDNA cloning and expression

7 January 2021

1 reference

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Cloning and pharmacological characterization of a rat mu opioid receptor

7 January 2021

1 reference

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Cloning and functional comparison of kappa and delta opioid receptors from mouse brain

7 January 2021

1 reference

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Blockade of morphine analgesia by an antisense oligodeoxynucleotide against the mu receptor

7 January 2021

1 reference

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Blockade of U50,488H analgesia by antisense oligodeoxynucleotides to a kappa-opioid receptor

7 January 2021

1 reference

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Selective loss of delta opioid analgesia and binding by antisense oligodeoxynucleotides to a delta opioid receptor

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2801%2900761-4

Changes in GIRK1/GIRK2 deactivation kinetics and basal activity in the presence and absence of RGS4.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2801%2900761-4

Evidence that neuronal G-protein-gated inwardly rectifying K+ channels are activated by G beta gamma subunits and function as heteromultimers

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2801%2900761-4

Mu and delta receptors belong to a family of receptors that are coupled to potassium channels

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2801%2900761-4

Opioids activate both an inward rectifier and a novel voltage-gated potassium conductance in the hippocampal formation

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2801%2900761-4

Inhibition of G-protein-mediated MAP kinase activation by a new mammalian gene family

7 January 2021

1 reference

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RGS proteins reconstitute the rapid gating kinetics of gbetagamma-activated inwardly rectifying K+ channels

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2801%2900761-4

Opioid receptor three-dimensional structures from distance geometry calculations with hydrogen bonding constraints

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2801%2900761-4

Molecular cloning of a mouse G-protein-activated K+ channel (mGIRK1) and distinct distributions of three GIRK (GIRK1, 2 and 3) mRNAs in mouse brain

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2801%2900761-4

Functional messenger RNAs are produced by SP6in vitrotranscription of cloned cDNAs

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2801%2900761-4

Cloning of a human kappa opioid receptor from the brain

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2801%2900761-4

Identification of a human delta opioid receptor: cloning and expression

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2801%2900761-4

Subunit stoichiometry of a mammalian K+ channel determined by construction of multimeric cDNAs.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2801%2900761-4

Comparative binding of mu and delta selective ligands in whole brain and pons/medulla homogenates from rat: affinity profiles of fentanyl derivatives

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2801%2900761-4

Identification and characterization of three new alternatively spliced mu-opioid receptor isoforms.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2801%2900761-4

Retention of heroin and morphine-6 beta-glucuronide analgesia in a new line of mice lacking exon 1 of MOR-1.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2801%2900761-4

Effects of morphine glucuronides on the function of opioid receptors in human SK-N-SH cells

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2801%2900761-4

10.1016/S0006-2952(01)00761-4

7 January 2021

Identifiers

DOI

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release_gsffvum3tva3rkvlgep7tgiupu

26 November 2017

Fatcat ID

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Fatcat

https://api.fatcat.wiki/v0/release/gsffvum3tva3rkvlgep7tgiupu

mapped directly with Wikidata item

24 November 2022

based on heuristic

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