(Q43962766)

English

Dermorphin and deltorphin heptapeptide analogues: replacement of Phe residue by Dmp greatly improves opioid receptor affinity and selectivity

scientific article published in March 2002

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scholarly article

1 reference

Europe PubMed Central

PubMed publication ID

28 November 2017

Dermorphin and deltorphin heptapeptide analogues: replacement of Phe residue by Dmp greatly improves opioid receptor affinity and selectivity (English)

1 reference

Europe PubMed Central

PubMed publication ID

28 November 2017

author name string

Akihiro Ambo

1

1 reference

Europe PubMed Central

PubMed publication ID

28 November 2017

Harumi Murase

2

1 reference

Europe PubMed Central

PubMed publication ID

28 November 2017

Hideko Niizuma

3

1 reference

Europe PubMed Central

PubMed publication ID

28 November 2017

Hidekazu Ouchi

4

1 reference

Europe PubMed Central

PubMed publication ID

28 November 2017

Yutaka Yamamoto

5

1 reference

Europe PubMed Central

PubMed publication ID

28 November 2017

Yusuke Sasaki

6

1 reference

Europe PubMed Central

PubMed publication ID

28 November 2017

language of work or name

0 references

publication date

1 March 2002

1 reference

Europe PubMed Central

PubMed publication ID

28 November 2017

Bioorganic & Medicinal Chemistry Letters

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Europe PubMed Central

PubMed publication ID

28 November 2017

12

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Europe PubMed Central

PubMed publication ID

28 November 2017

6

1 reference

Europe PubMed Central

PubMed publication ID

28 November 2017

879-881

1 reference

Europe PubMed Central

PubMed publication ID

28 November 2017

Recent developments in the design of receptor specific opioid peptides

1 reference

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Preparation and opioid activity of analogues of the analgesic dipeptide 2,6-dimethyl-L-tyrosyl-N-(3-phenylpropyl)-D-alaninamide

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2802%2900035-5

7 January 2021

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Systemic analgesic activity and delta-opioid selectivity in [2,6-dimethyl-Tyr1,D-Pen2,D-Pen5]enkephalin

1 reference

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7 January 2021

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Enkephalin Analogs as Systemically Active Antinociceptive Agents: O- and N-Alkylated Derivatives of the Dipeptide Amide L-2,6-Dimethyltyrosyl-N-(3-phenylpropyl)-D-alaninamide

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2802%2900035-5

7 January 2021

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Delta opioidmimetic antagonists: prototypes for designing a new generation of ultraselective opioid peptides.

1 reference

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7 January 2021

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Opioid receptor selectivity alteration by single residue replacement: synthesis and activity profile of [Dmt1]deltorphin B.

1 reference

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7 January 2021

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Evolution of the Dmt-Tic pharmacophore: N-terminal methylated derivatives with extraordinary delta opioid antagonist activity

1 reference

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7 January 2021

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Design of a high affinity peptidomimetic opioid agonist from peptide pharmacophore models.

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

The opioid mu agonist/delta antagonist DIPP-NH(2)[Psi] produces a potent analgesic effect, no physical dependence, and less tolerance than morphine in rats

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

Dmt-Tic-OH a highly selective and potent delta-opioid dipeptide receptor antagonist after systemic administration in the mouse

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

New delta-opioid antagonists as pharmacological probes.

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

Further studies on the Dmt-Tic pharmacophore: hydrophobic substituents at the C-terminus endow delta antagonists to manifest mu agonism or mu antagonism.

1 reference

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7 January 2021

based on heuristic

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Biological properties of opioid peptides replacing Tyr at position 1 by 2,6-dimethyl-Tyr

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

Enkephalin analogues with 2',6'-dimethylphenylalanine replacing phenylalanine in position 4.

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

AMINO ACID COMPOSITION AND SEQUENCE OF DERMORPHIN, A NOVEL OPIATE-LIKE PEPTIDE FROM THE SKIN OF PHYLLOMEDUSA SAUVAGEI

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2802%2900035-5

7 January 2021

based on heuristic

inferred from DOI database lookup

Deltorphins: a family of naturally occurring peptides with high affinity and selectivity for delta opioid binding sites

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2802%2900035-5

7 January 2021

based on heuristic

inferred from DOI database lookup

[D-Ala2]deltorphin II analogs with high affinity and selectivity for delta-opioid receptor

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2802%2900035-5

7 January 2021

based on heuristic

inferred from DOI database lookup

Structure-activity relationships of cyclic opioid peptide analogues containing a phenylalanine residue in the 3-position

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2802%2900035-5

7 January 2021

based on heuristic

inferred from DOI database lookup

Modification of the Phe3 aromatic moiety in delta receptor-selective dermorphin/deltorphin-related tetrapeptides. Effects on opioid receptor binding

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2802%2900035-5

7 January 2021

based on heuristic

inferred from DOI database lookup

What peptides these deltorphins be.

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2802%2900035-5

7 January 2021

based on heuristic

inferred from DOI database lookup

Identifiers

10.1016/S0960-894X(02)00035-5

1 reference

Europe PubMed Central

PubMed publication ID

28 November 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

28 November 2017

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