(Q43964144)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11960662%20AND%20SRC:MED&resulttype=core&format=json

9 December 2019

title

Active conformation of some arylpiperazine postsynaptic 5-HT(1A) receptor antagonists (English)

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9 December 2019

2

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9 December 2019

Anna Wesołowska

series ordinal

4

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9 December 2019

author name string

Maria Halina Paluchowska

series ordinal

1

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9 December 2019

Sijka Charakchieva-Minol

series ordinal

3

1 reference

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9 December 2019

publication date

1 April 2002

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European Journal of Medicinal Chemistry

9 December 2019

published in

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9 December 2019

volume

37

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9 December 2019

issue

4

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9 December 2019

page(s)

273-283

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Arylpiperazine derivatives as high-affinity 5-HT1A serotonin ligands

9 December 2019

cites work

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

A series of N4-imidoethyl derivatives of 1-(2,3-dihydro-1,4-benzodioxin-5-yl)piperazine as 5-HT1A receptor ligands: synthesis and structure-affinity relationships

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

Structure-activity relationship studies of CNS agents, Part 22. A search for new trazodone-like antidepressants: synthesis and preliminary receptor binding studies

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

Structure-activity relationship studies of CNS agents, Part 31: Analogs of MP 3022 with a different number of nitrogen atoms in the heteroaromatic fragment--new 5-HT1A receptor ligands

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

Synthesis and structure-activity relationships of a new model of arylpiperazines. 1. 2-[[4-(o-methoxyphenyl)piperazin-1-yl]methyl]-1, 3-dioxoperhydroimidazo[1,5-alpha]pyridine: a selective 5-HT1A receptor agonist.

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

Structure-affinity relationship studies on 5-HT1A receptor ligands. 1. Heterobicyclic phenylpiperazines with N4-alkyl substituents

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

Structure-activity relationship studies of CNS agents, XIX: Quantitative analysis of the alkyl chain effects on the 5-HT1A and 5-HT2 receptor affinities of 4-alkyl-1-arylpiperazines and their analogs

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

Structure—affinity relationship studies on benzotriazole derivatives binding to 5-HT receptor subtypes

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

[[(Arylpiperazinyl)alkyl]thio]thieno[2,3-d]pyrimidinone derivatives as high-affinity, selective 5-HT1A receptor ligands

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

1-aryl-4-[(1-tetralinyl)alkyl]piperazines: alkylamido and alkylamino derivatives. Synthesis, 5-HT1A receptor affinity, and selectivity. 3

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

High potent and selective arylpiperazine derivatives as ligands for the 5-HT1A receptor

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

Structure-affinity relationship studies on 5-HT1A receptor ligands. 2. Heterobicyclic phenylpiperazines with N4-aralkyl substituents

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

New (2-methoxyphenyl)piperazine derivatives as 5-HT1A receptor ligands with reduced alpha 1-adrenergic activity. Synthesis and structure-affinity relationships

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

5-HT1A- versus D2-Receptor Selectivity of Flesinoxan and AnalogousN 4-SubstitutedN 1-Arylpiperazines

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

Synthesis and SAR of adatanserin: novel adamantyl aryl- and heteroarylpiperazines with dual serotonin 5-HT(1A) and 5-HT(2) activity as potential anxiolytic and antidepressant agents

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

Effect of linking bridge modifications on the antipsychotic profile of some phthalimide and isoindolinone derivatives

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

10-substituted 11-oxygenated (R)-aporphines: synthesis, pharmacology, and modeling of 5-HT1A receptor interactions

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

Three-dimensional quantitative structure-activity relationships of 5-HT receptor binding data for tetrahydropyridinylindole derivatives: a comparison of the Hansch and CoMFA methods

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

A 3-D model for 5-HT1A-receptor agonists based on stereoselective methyl-substituted and conformationally restricted analogues of 8-hydroxy-2-(dipropylamino)tetralin

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

Comparison of 5-HT1A and dopamine D2 pharmacophores. X-ray structures and affinities of conformationally constrained ligands

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

Development of 5-HT1A receptor antagonists

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

Structure-activity relationship studies of central nervous system agents. 13. 4-[3-(Benzotriazol-1-yl)propyl]-1-(2-methoxyphenyl)piperazine, a new putative 5-HT1A receptor antagonist, and its analogs

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

On the bioactive conformation of NAN-190 (1) and MP3022 (2), 5-HT(1A) receptor antagonists

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

Analogs of the 5-HT1A serotonin antagonist 1-(2-methoxyphenyl)-4-[4-(2-phthalimido)butyl]piperazine with reduced .alpha.1-adrenergic affinity

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

1,2,3,4-tetrahydroisoquinoline derivatives: a new class of 5-HT1A receptor ligands

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

8-[4-[2-(1,2,3,4-Tetrahydroisoquinolinyl]butyl-8-azaspiro[4.5]decane-7,9-dione: a new 5-HT1A receptor ligand with the same activity profile as buspirone.

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

The involvement of subtypes of the 5-HT1 receptor and of catecholaminergic systems in the behavioural response to 8-hydroxy-2-(di-n-propylamino)tetralin in the rat.

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

Selective activation of 5HT1A receptors induces lower lip retraction in the rat.

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2801%2901312-5

7 January 2021

10.1016/S0223-5234(01)01312-5

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11960662%20AND%20SRC:MED&resulttype=core&format=json

9 December 2019

1 reference