(Q43967464)

English

Analogs of Substance P modified at the C-terminus which are both agonist and antagonist of the NK-1 receptor depending on the second messenger pathway.

scientific article published in May 2002

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scholarly article

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9 December 2019

Analogs of Substance P modified at the C-terminus which are both agonist and antagonist of the NK-1 receptor depending on the second messenger pathway (English)

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11966980%20AND%20SRC:MED&resulttype=core&format=json

9 December 2019

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Emmanuelle Sachon

1

1 reference

Europe PubMed Central

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9 December 2019

5

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9 December 2019

author name string

S Girault-Lagrange

2

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9 December 2019

G Chassaing

3

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9 December 2019

S Lavielle

4

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9 December 2019

publication date

1 May 2002

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9 December 2019

Chemical Biology and Drug Design

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9 December 2019

59

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9 December 2019

5

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9 December 2019

232-240

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9 December 2019

The mammalian tachykinin receptors

1 reference

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7 January 2021

based on heuristic

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Use of the chemical structure of peptides as the starting point to design nonpeptide agonists and antagonists at peptide receptors: examples with cholecystokinin and tachykinins

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

NK1 (substance P) receptor antagonists--why are they not analgesic in humans?

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

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A Potent Nonpeptide Antagonist of the Substance P (NK 1 ) Receptor

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

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Antinociceptive properties and inhibition of neurogenic inflammation with potent SP antagonists belonging to perhydroisoindolones

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Tachykinin receptors and tachykinin receptor antagonists

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Design and Synthesis of Effective Antagonists of Substance P

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Potent and highly selective neurokinin antagonists

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Highly potent substance P antagonists substituted with β-phenyl- or β-benzyl-proline at position 10

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Two related neurokinin-1 receptor antagonists have overlapping but different binding sites

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Synthesis of a substance P antagonist with a somatostatin scaffold: factors affecting agonism/antagonism at GPCRs and the role of pseudosymmetry

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Synthesis and biological activity of NK1 tachykinin antagonists not containing D-residues

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Synthesis of potent antagonists of substance P by modifying the methionyl and glutaminyl residues of its C-terminal hexapeptide and without using D-amino acids

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Model systems for the study of seven-transmembrane-segment receptors

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Septide and neurokinin A are high-affinity ligands on the NK-1 receptor: evidence from homologous versus heterologous binding analysis.

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

High affinity binding of [3H]propionyl-[Met(O2)11]substance P(7-11), a tritiated septide-like peptide, in Chinese hamster ovary cells expressing human neurokinin-1 receptors and in rat submandibular glands

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Further Delineation of the Two Binding Sites (R*n) Associated with Tachykinin Neurokinin-1 Receptors Using [3-Prolinomethionine11]SP Analogues

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Internalization of [3H]substance P analogues in NK-1 receptor transfected CHO cells.

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

The use of photolabelled peptides to localize the substance-P-binding site in the human neurokinin-1 tachykinin receptor

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Asymmetric synthesis of Boc- N -methyl- p -benzoyl-phenylalanine. preparation of a photoreactive antagonist of Substance P

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Synthesis and biological evaluation of cholecystokinin analogs in which the Asp-Phe-NH2 moiety has been replaced by a 3-amino-7-phenylheptanoic acid or a 3-amino-6-(phenyloxy)hexanoic acid

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

The design and synthesis of the high efficacy, non-peptide CCK 1 receptor agonist PD 170292

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Importance of the leucine side-chain to the spasmogenic activity and binding of Substance P analogues

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Further evidence for the presence of "septide-sensitive" tachykinin binding sites in tissues possessing solely NK(1) tachykinin receptors

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Differential contribution of substance P and neurokinin A to spinal cord neurokinin-1 receptor signaling in the rat.

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Direct evidence for the interaction of neurokinin A with the tachykinin NK(1) receptor in tissue

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Tachykinin NK-1 receptor probed with constrained analogues of substance P.

1 reference

https://api.crossref.org/works/10.1034%2FJ.1399-3011.2002.01977.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Identifiers

10.1034/J.1399-3011.2002.01977.X

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11966980%20AND%20SRC:MED&resulttype=core&format=json

9 December 2019

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11966980%20AND%20SRC:MED&resulttype=core&format=json

9 December 2019

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