(Q44082415)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12147298%20AND%20SRC:MED&resulttype=core&format=json

11 November 2019

title

Substrate-dependent, non-hyperbolic kinetics of pig brain prolyl oligopeptidase and its tight binding inhibition by JTP-4819 (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12147298%20AND%20SRC:MED&resulttype=core&format=json

11 November 2019

5

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12147298%20AND%20SRC:MED&resulttype=core&format=json

11 November 2019

Markus M Forsberg

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12147298%20AND%20SRC:MED&resulttype=core&format=json

11 November 2019

Arturo García-Horsman

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12147298%20AND%20SRC:MED&resulttype=core&format=json

11 November 2019

Erik A A Wallén

6

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12147298%20AND%20SRC:MED&resulttype=core&format=json

11 November 2019

Pekka T. Männistö

8

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12147298%20AND%20SRC:MED&resulttype=core&format=json

11 November 2019

author name string

Jarkko I Venäläinen

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12147298%20AND%20SRC:MED&resulttype=core&format=json

11 November 2019

Risto O Juvonen

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12147298%20AND%20SRC:MED&resulttype=core&format=json

11 November 2019

Jukka Gynther

7

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12147298%20AND%20SRC:MED&resulttype=core&format=json

11 November 2019

language of work or name

English

0 references

publication date

1 August 2002

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12147298%20AND%20SRC:MED&resulttype=core&format=json

11 November 2019

published in

Biochemical Pharmacology

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12147298%20AND%20SRC:MED&resulttype=core&format=json

11 November 2019

volume

64

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12147298%20AND%20SRC:MED&resulttype=core&format=json

11 November 2019

issue

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12147298%20AND%20SRC:MED&resulttype=core&format=json

11 November 2019

page(s)

463-471

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12147298%20AND%20SRC:MED&resulttype=core&format=json

Proline specific peptidases

11 November 2019

cites work

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2802%2901184-X

cDNA cloning of porcine brain prolyl endopeptidase and identification of the active-site seryl residue

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2802%2901184-X

In vitro and in vivo inhibition of prolyl endopeptidase

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2802%2901184-X

Effect of a novel prolyl endopeptidase inhibitor, JTP-4819, on spatial memory and central cholinergic neurons in aged rats.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2802%2901184-X

Substrate- and pH-dependent contribution of oxyanion binding site to the catalysis of prolyl oligopeptidase, a paradigm of the serine oligopeptidase family

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2802%2901184-X

7 January 2021

Prolyl Oligopeptidase

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2802%2901184-X

Structures of prolyl oligopeptidase substrate/inhibitor complexes. Use of inhibitor binding for titration of the catalytic histidine residue

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2802%2901184-X

A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2802%2901184-X

Tight-binding inhibitors-I. Kinetic behavior

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2802%2901184-X

Automated docking using a Lamarckian genetic algorithm and an empirical binding free energy function

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2802%2901184-X

7 January 2021

Prolyl oligopeptidases

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2802%2901184-X

pH-dependent mechanism in the catalysis of prolyl endopeptidase from pig muscle

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2802%2901184-X

Changes in Prolyl Endopeptidase During Maturation of Rat Brain and Hydrolysis of Substance P by the Purified Enzyme

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2802%2901184-X

Prolyl endopeptidase from bovine testis: purification, characterization and comparison with the enzymes from other tissues

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2802%2901184-X

Oligopeptidase B: a new type of serine peptidase with a unique substrate-dependent temperature sensitivity

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2802%2901184-X

A Novel Prolyl Endopeptidase Inhibitor, JTP-4819 - Its Behavioral and Neurochemical Properties for the Treatment of Alzheimer's Disease

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2802%2901184-X

Slow tight-binding inhibition of prolyl endopeptidase by benzyloxycarbonyl-prolyl-prolinal

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2802%2901184-X

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0006-2952%2802%2901184-X

10.1016/S0006-2952(02)01184-X

7 January 2021

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12147298%20AND%20SRC:MED&resulttype=core&format=json

11 November 2019

1 reference