(Q44241682)

1 December 2017

title

Synthesis and pharmacological characterisation of 2,4-dicarboxy-pyrroles as selective non-competitive mGluR1 antagonists (English)

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1 December 2017

1

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1 December 2017

4

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6

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1 December 2017

11

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1 December 2017

Romano Di Fabio

2

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1 December 2017

Paolo Cavanni

3

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1 December 2017

Anna Maria Capelli

5

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1 December 2017

Mauro Corsi

7

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1 December 2017

Corrado Corti

8

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1 December 2017

Daniele Donati

9

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1 December 2017

Aldo Feriani

10

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1 December 2017

Micaela Maffeis

12

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1 December 2017

Andrea Missio

13

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1 December 2017

Emiliangelo Ratti

14

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1 December 2017

Alfredo Paio

15

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1 December 2017

Roberta Pachera

16

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1 December 2017

Mauro Quartaroli

17

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1 December 2017

Angelo Reggiani

18

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1 December 2017

Fabio Maria Sabbatini

19

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1 December 2017

David G Trist

20

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1 December 2017

Annarosa Ugolini

21

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1 December 2017

Giovanni Vitulli

22

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1 December 2017

language of work or name

English

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publication date

1 January 2003

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Bioorganic & Medicinal Chemistry

1 December 2017

published in

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1 December 2017

volume

11

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1 December 2017

issue

2

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1 December 2017

page(s)

171-183

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Substituted indole-2-carboxylates as in vivo potent antagonists acting as the strychnine-insensitive glycine binding site.

1 December 2017

cites work

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Cycloalkyl indole-2-carboxylates as useful tools for mapping the "north-eastern" region of the glycine binding site associated with the NMDA receptor

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Molecular diversity and functions of glutamate receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Cloned glutamate receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

The metabotropic glutamate receptors: structure and functions

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Metabotropic glutamate receptors: novel targets for drug development

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Pharmacology and functions of metabotropic glutamate receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

The ligand-binding domain in metabotropic glutamate receptors is related to bacterial periplasmic binding proteins

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Structural basis of glutamate recognition by a dimeric metabotropic glutamate receptor

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Cloning and characterization of an extracellular Ca(2+)-sensing receptor from bovine parathyroid

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Expression cloning of GABA(B) receptors uncovers similarity to metabotropic glutamate receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Olfactory receptors, vomeronasal receptors, and the organization of olfactory information

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Ligands for glutamate receptors: design and therapeutic prospects

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Pharmacological agents acting at subtypes of metabotropic glutamate receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Pharmacology of (S)-homoquisqualic acid and (S)-2-amino-5-phosphonopentanoic acid [(S)-AP5] at cloned metabotropic glutamate receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Phenylglycine derivatives discriminate between mGluR1- and mGluR5-mediated responses

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Analysis of agonist and antagonist activities of phenylglycine derivatives for different cloned metabotropic glutamate receptor subtypes

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

(S)-(+)-2-(3'-carboxybicyclo[1.1.1]pentyl)-glycine, a structurally new group I metabotropic glutamate receptor antagonist

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Competitive antagonism at metabotropic glutamate receptors by (S)-4-carboxyphenylglycine and (RS)-alpha-methyl-4-carboxyphenylglycine

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Synthesis and biological evaluation of 2-(3'-(1H-tetrazol-5-yl) bicyclo[1.1.1]pent-1-yl)glycine (S-TBPG), a novel mGlu1 receptor antagonist

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Neuroprotective and behavioral effects of the selective metabotropic glutamate mGlu(1) receptor antagonist BAY 36-7620.

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Metabotropic glutamate receptors: a new target for the therapy of neurodegenerative disorders?

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

1-Aminoindan-1,5-dicarboxylic acid and (S)-(+)-2-(3'-carboxybicyclo[1.1.1] pentyl)-glycine, two mGlu1 receptor-preferring antagonists, reduce neuronal death in in vitro and in vivo models of cerebral ischaemia

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Evidence for a role of metabotropic glutamate receptors in sustained nociceptive inputs to rat dorsal horn neurons

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Metabotropic glutamate receptor mRNA expression in rat spinal cord.

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Augmented motor activity and reduced striatal preprodynorphin mRNA induction in response to acute amphetamine administration in metabotropic glutamate receptor 1 knockout mice

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Knockdown of spinal metabotropic glutamate receptor 1 (mGluR(1)) alleviates pain and restores opioid efficacy after nerve injury in rats

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Pharmacophore models of group I and group II metabotropic glutamate receptor agonists. Analysis of conformational, steric, and topological parameters affecting potency and selectivity

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Modeling of amino-terminal domains of group I metabotropic glutamate receptors: structural motifs affecting ligand selectivity

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Competitive antagonism by phenylglycine derivatives at type I metabotropic glutamate receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Fluorescence measurement of changes in intracellular calcium induced by excitatory amino acids in cultured cortical astrocytes

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Synthetische Versuche mit dem Acetessigester. II. Mittheilung: Ueberführung des Diacetbernsteinsäureesters und des Acetessigesters in Pyrrolderivate

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Diversity in mammalian tachykinin peptidergic neurons: multiple peptides, receptors, and regulatory mechanisms

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Characterization of metabotropic glutamate receptor-stimulated phosphoinositide hydrolysis in rat cultured cerebellar granule cells.

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

The formalin test in mice: dissociation between inflammatory and non-inflammatory pain

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Effects of intraplantar morphine on paw edema and pain-related behaviour in a rat model of repeated acute inflammation

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Differential roles of NMDA and non-NMDA receptor activation in induction and maintenance of thermal hyperalgesia in rats with painful peripheral mononeuropathy

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Modulation of nociceptive transmission by NMDA/glycine site receptor in the ventroposterolateral nucleus of the thalamus

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Maturation in properties of motoneurons and their segmental input in the neonatal rat

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Expression and purification of the extracellular ligand binding region of metabotropic glutamate receptor subtype 1.

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Domains involved in the specificity of G protein activation in phospholipase C-coupled metabotropic glutamate receptors.

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Cloning and characterization of alternative mRNA forms for the rat metabotropic glutamate receptors mGluR7 and mGluR8

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Primary structure and functional expression of a rat G-protein-coupled muscarinic potassium channel

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

Cloning and functional expression of a rat heart KATP channel

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

General synthesis of hydrocarbon-soluble porphyrins

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900424-8

7 January 2021

10.1016/S0968-0896(02)00424-8

Identifiers

DOI

1 reference

1 December 2017

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