(Q44244370)

1 December 2017

title

Plasmepsin inhibitors: design, synthesis, inhibitory studies and crystal structure analysis (English)

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1 December 2017

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Kesavulu MM

1

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1 December 2017

Prakasha Gowda AS

2

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1 December 2017

Ramya TN

3

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1 December 2017

Surolia N

4

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1 December 2017

Suguna K

5

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1 December 2017

publication date

1 October 2005

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Chemical Biology and Drug Design

1 December 2017

published in

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1 December 2017

volume

66

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1 December 2017

issue

4

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1 December 2017

page(s)

211-219

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Drug resistance in malaria

1 December 2017

cites work

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https://api.crossref.org/works/10.1111%2FJ.1399-3011.2005.00288.X

New class of small nonpeptidyl compounds blocks Plasmodium falciparum development in vitro by inhibiting plasmepsins

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1399-3011.2005.00288.X

Identification and characterization of falcilysin, a metallopeptidase involved in hemoglobin catabolism within the malaria parasite Plasmodium falciparum

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1399-3011.2005.00288.X

A distinct member of the aspartic proteinase gene family from the human malaria parasite Plasmodium falciparum

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1399-3011.2005.00288.X

Four plasmepsins are active in the Plasmodium falciparum food vacuole, including a protease with an active-site histidine

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1399-3011.2005.00288.X

Aspartic proteases of Plasmodium falciparum and other parasitic protozoa as drug targets.

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1399-3011.2005.00288.X

Design and synthesis of plasmepsin I and plasmepsin II inhibitors with activity in Plasmodium falciparum-infected cultured human erythrocytes

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1399-3011.2005.00288.X

Design and synthesis of potent inhibitors of plasmepsin I and II: X-ray crystal structure of inhibitor in complex with plasmepsin II.

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1399-3011.2005.00288.X

Novel uncomplexed and complexed structures of plasmepsin II, an aspartic protease from Plasmodium falciparum

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1399-3011.2005.00288.X

New inhibitors of the malaria aspartyl proteases plasmepsin I and II.

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1399-3011.2005.00288.X

Potent inhibitors of the Plasmodium falciparum enzymes plasmepsin I and II devoid of cathepsin D inhibitory activity

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1399-3011.2005.00288.X

Structure and inhibition of plasmepsin II, a hemoglobin-degrading enzyme from Plasmodium falciparum

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1399-3011.2005.00288.X

X-ray structure of plasmepsin II complexed with a potent achiral inhibitor

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1399-3011.2005.00288.X

10.1111/J.1399-3011.2005.00288.X

21 January 2018

Identifiers

DOI

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1 December 2017

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