(Q44346034)

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Identification of selective agonists and positive allosteric modulators for µ- and δ-opioid receptors from a single high-throughput screen

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scholarly article

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Europe PubMed Central

PubMed publication ID

2 December 2017

Identification of selective agonists and positive allosteric modulators for µ- and δ-opioid receptors from a single high-throughput screen (English)

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

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author name string

Neil T Burford

1

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Tom Wehrman

2

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Daniel Bassoni

3

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Jonathan O'Connell

4

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Martyn Banks

5

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Litao Zhang

6

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2 December 2017

Andrew Alt

7

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2 December 2017

publication date

21 July 2014

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Europe PubMed Central

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2 December 2017

Journal of Biomolecular Screening

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Europe PubMed Central

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2 December 2017

19

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Europe PubMed Central

PubMed publication ID

2 December 2017

9

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Europe PubMed Central

PubMed publication ID

2 December 2017

1255-1265

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Management of opioid side effects in cancer-related and chronic noncancer pain: a systematic review

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

Opioid receptors

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

Opioid receptor heteromers in analgesia

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

Mix and match: heterodimers and opioid tolerance

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

Strategies for the identification of allosteric modulators of G-protein-coupled receptors

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

Allosteric Modulation of G Protein–Coupled Receptors

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

Measurements of β-arrestin recruitment to activated seven transmembrane receptors using enzyme complementation

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

A homogeneous enzyme fragment complementation-based beta-arrestin translocation assay for high-throughput screening of G-protein-coupled receptors

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

Discovery of positive allosteric modulators and silent allosteric modulators of the μ-opioid receptor

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

A role for heterodimerization of mu and delta opiate receptors in enhancing morphine analgesia

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

Morphine-activated opioid receptors elude desensitization by beta-arrestin

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

Opioid receptors and their ligands

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

Understanding the effect of different assay formats on agonist parameters: a study using the µ-opioid receptor

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

Identification of a μ-δ opioid receptor heteromer-biased agonist with antinociceptive activity

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

A heterodimer-selective agonist shows in vivo relevance of G protein-coupled receptor dimers

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

6'-Guanidinonaltrindole (6'-GNTI) is a G protein-biased κ-opioid receptor agonist that inhibits arrestin recruitment

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

Comparison of the relative efficacy and potency of mu-opioid agonists to activate Galpha(i/o) proteins containing a pertussis toxin-insensitive mutation

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

Functional impact of allosteric agonist activity of selective positive allosteric modulators of metabotropic glutamate receptor subtype 5 in regulating central nervous system function.

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

Subtype-selective allosteric modulators of muscarinic receptors for the treatment of CNS disorders

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

The narcotic antagonist naloxone enhances clinical pain

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

Functional selectivity and biased receptor signaling.

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

Specific G protein activation and mu-opioid receptor internalization caused by morphine, DAMGO and endomorphin I

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

μ-opioid receptors: correlation of agonist efficacy for signalling with ability to activate internalization

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

Endomorphin-2: a biased agonist at the μ-opioid receptor.

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

A G protein-biased ligand at the μ-opioid receptor is potently analgesic with reduced gastrointestinal and respiratory dysfunction compared with morphine

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

Differential regulation of muscarinic M1 receptors by orthosteric and allosteric ligands

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

Receptor activation involving positive allosteric modulation, unlike full agonism, does not result in GABAB receptor desensitization

1 reference

https://api.crossref.org/works/10.1177%2F1087057114542975

21 January 2018

Identifiers

10.1177/1087057114542975

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

ResearchGate publication ID

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