(Q44376093)

2 December 2017

title

Novel indole-based inhibitors of IMPDH: introduction of hydrogen bond acceptors at indole C-3. (English)

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2 December 2017

Scott H Watterson

1

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2 December 2017

T G Murali Dhar

2

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2 December 2017

Shelley K Ballentine

3

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2 December 2017

Zhongqi Shen

4

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2 December 2017

Joel C Barrish

5

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2 December 2017

Daniel Cheney

6

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2 December 2017

Catherine A Fleener

7

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2 December 2017

Katherine A Rouleau

8

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2 December 2017

Robert Townsend

9

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2 December 2017

Diane L Hollenbaugh

10

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2 December 2017

Edwin J Iwanowicz

11

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2 December 2017

language of work or name

English

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publication date

1 April 2003

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Bioorganic & Medicinal Chemistry Letters

2 December 2017

published in

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2 December 2017

volume

13

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2 December 2017

issue

7

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2 December 2017

page(s)

1273-1276

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Inosine-5'-monophosphate dehydrogenase: regulation of expression and role in cellular proliferation and T lymphocyte activation.

2 December 2017

cites work

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900109-4

7 January 2021

IMP dehydrogenase, an enzyme linked with proliferation and malignancy

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900109-4

7 January 2021

The structure of inosine 5'-monophosphate dehydrogenase and the design of novel inhibitors

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900109-4

7 January 2021

Synthesis and modeling studies with monocyclic analogues of mycophenolic acid

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900109-4

7 January 2021

Synthesis and immunosuppressive activity of some side-chain variants of mycophenolic acid

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900109-4

7 January 2021

Enterohepatic recirculation: a powerful incentive for drug discovery in the inosine monophosphate dehydrogenase field

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900109-4

7 January 2021

The acyl glucuronide metabolite of mycophenolic acid inhibits the proliferation of human mononuclear leukocytes

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900109-4

7 January 2021

Discovery of N-[2-[2-[[3-methoxy-4-(5-oxazolyl)phenyl]amino]-5-oxazolyl]phenyl]-N-methyl-4- morpholineacetamide as a novel and potent inhibitor of inosine monophosphate dehydrogenase with excellent in vivo activity.

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900109-4

7 January 2021

VX-497: a novel, selective IMPDH inhibitor and immunosuppressive agent

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900109-4

7 January 2021

Novel amide-based inhibitors of inosine 5'-monophosphate dehydrogenase

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900109-4

7 January 2021

Novel guanidine-based inhibitors of inosine monophosphate dehydrogenase.

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900109-4

7 January 2021

Novel diamide-based inhibitors of IMPDH.

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900109-4

7 January 2021

Rapid synthesis of triazine inhibitors of inosine monophosphate dehydrogenase

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900109-4

7 January 2021

Novel inhibitors of IMPDH: a highly potent and selective quinolone-based series

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900109-4

7 January 2021

Quinolone-based IMPDH inhibitors: introduction of basic residues on ring D and SAR of the corresponding mono, di and benzofused analogues

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900109-4

7 January 2021

A convenient synthesis of acetylenes: catalytic substitutions of acetylenic hydrogen with bromoalkenes, iodoarenes and bromopyridines

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900109-4

7 January 2021

Versatile Indole Synthesis by a 5-endo-dig Cyclization Mediated by Potassium or Cesium Bases We thank the DFG (Leibniz-Programm) and the Fonds der Chemischen Industrie for generous financial support. A.L.R. and C. K. thank the Humboldt-Foundation an

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900109-4

7 January 2021

10.1016/S0960-894X(03)00109-4

Identifiers

DOI

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2 December 2017

1 reference