(Q44416588)

English

Imidazole derivatives as a novel class of hybrid compounds with inhibitory histamine N-methyltransferase potencies and histamine hH3 receptor affinities

scientific article published in May 2003

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scholarly article

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Imidazole derivatives as a novel class of hybrid compounds with inhibitory histamine N-methyltransferase potencies and histamine hH3 receptor affinities (English)

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

3

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2 December 2017

author name string

Sven Grassmann

1

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Europe PubMed Central

PubMed publication ID

2 December 2017

Joachim Apelt

2

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Europe PubMed Central

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2 December 2017

Xavier Ligneau

4

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Europe PubMed Central

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2 December 2017

Heinz H Pertz

5

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Europe PubMed Central

PubMed publication ID

2 December 2017

Yuan Hui Zhao

6

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Europe PubMed Central

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2 December 2017

Jean Michel Arrang

7

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Europe PubMed Central

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2 December 2017

C Robin Ganellin

8

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Europe PubMed Central

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2 December 2017

Jean Charles Schwartz

9

1 reference

Europe PubMed Central

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2 December 2017

Walter Schunack

10

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Europe PubMed Central

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2 December 2017

Holger Stark

11

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Europe PubMed Central

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2 December 2017

language of work or name

0 references

publication date

1 May 2003

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Europe PubMed Central

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2 December 2017

Bioorganic & Medicinal Chemistry

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Europe PubMed Central

PubMed publication ID

2 December 2017

11

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Europe PubMed Central

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2 December 2017

10

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2 December 2017

2163-2174

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Europe PubMed Central

PubMed publication ID

2 December 2017

Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

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Histaminergic transmission in the mammalian brain

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The physiology of brain histamine.

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Catabolism of 3H-histamine in the rat brain after intracisternal administration

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Highly potent and selective ligands for histamine H3-receptors

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Molecular cloning and characterization of a new human histamine receptor, HH4R

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Cloning and functional expression of the human histamine H3 receptor

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Immunological identification of the mammalian H3 histamine receptor in the mouse brain

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Cloning and cerebral expression of the guinea pig histamine H3 receptor: evidence for two isoforms

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Different antagonist binding properties of human and rat histamine H3 receptors

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Autoregulation of histamine release in brain by presynaptic H3-receptors

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Autoinhibition of histamine synthesis mediated by presynaptic H3-receptors

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Inhibition of histamine versus acetylcholine metabolism as a mechanism of tacrine activity.

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Therapeutic potential of histamine H3 receptor agonists and antagonists.

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Effects of thioperamide, a histamine H3-receptor antagonist, on a scopolamine-induced learning deficit using an elevated plus-maze test in mice

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Inhibition of cortical acetylcholine release and cognitive performance by histamine H3 receptor activation in rats

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Improvement by FUB 181, a novel histamine H3-receptor antagonist, of learning and memory in the elevated plus-maze test in mice

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A Highly Sensitive Assay for Histamine Using Ion-Pair HPLC Coupled with Postcolumn Fluorescent Derivatization: Its Application to Biological Specimens

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Development of a new class of nonimidazole histamine H(3) receptor ligands with combined inhibitory histamine N-methyltransferase activity

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9-Amino-1,2,3,4-tetrahydroacridine is a potent inhibitor of histamine N-methyltransferase

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Two Polymorphic Forms of Human Histamine Methyltransferase

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Inhibition of histamine-N-methyltransferase (HNMT) by fragments of 9-amino-1,2,3,4-tetrahydroacridine (tacrine) and by beta-carbolines

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Novel carbamates as potent histamine H3 receptor antagonists with high in vitro and oral in vivo activity

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The Use of Diethyl Azodicarboxylate and Triphenylphosphine in Synthesis and Transformation of Natural Products

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Development of FUB 181, a selective histamine H3-receptor antagonist of high oral in vivo potency with 4-(omega-(arylalkyloxy)alkyl)-1H-imidazole structure.

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Design, synthesis, and structure-activity relationships of acetylene-based histamine H3 receptor antagonists.

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Distinct pharmacology of rat and human histamine H(3) receptors: role of two amino acids in the third transmembrane domain

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Identifiers

10.1016/S0968-0896(03)00120-2

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

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