(Q44557212)
Statements
1 reference
Fluorine substitution can block CYP3A4 metabolism-dependent inhibition: identification of (S)-N-[1-(4-fluoro-3- morpholin-4-ylphenyl)ethyl]-3- (4-fluorophenyl)acrylamide as an orally bioavailable KCNQ2 opener devoid of CYP3A4 metabolism-dependent in (English)
1 reference
Yong-Jin Wu
1 reference
Carl D Davis
1 reference
Steven Dworetzky
1 reference
William C Fitzpatrick
1 reference
David Harden
1 reference
Huan He
1 reference
Ronald J Knox
1 reference
Amy E Newton
1 reference
Thomas Philip
1 reference
Craig Polson
1 reference
Digavalli V Sivarao
1 reference
Li-Qiang Sun
1 reference
Svetlana Tertyshnikova
1 reference
David Weaver
1 reference
Suresh Yeola
1 reference
Mary Zoeckler
1 reference
Michael W Sinz
1 reference
1 August 2003
1 reference
1 reference
46
1 reference
18
1 reference
3778-3781
1 reference
Identifiers
1 reference
1 reference