(Q44827536)

6 December 2017

Binding of (-)-[3H]-CGP12177 at two sites in recombinant human beta 1-adrenoceptors and interaction with beta-blockers (English)

1 reference

6 December 2017

3

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6 December 2017

Shirin S Joseph

1

1 reference

PubMed ID

15060759

6 December 2017

James A Lynham

series ordinal

2

1 reference

PubMed ID

15060759

6 December 2017

Alberto J Kaumann

series ordinal

4

1 reference

6 December 2017

2 April 2004

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Naunyn-Schmiedeberg's Archives of Pharmacology

6 December 2017

1 reference

6 December 2017

369

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6 December 2017

5

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6 December 2017

525-532

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https://scigraph.springernature.com/pub.10.1007/s00210-004-0884-y

6 December 2017

0 references

cites work

A gain-of-function polymorphism in a G-protein coupling domain of the human beta1-adrenergic receptor

1 reference

12 December 2020

Beta 1- and beta 2-adrenergic-receptor subpopulations in nonfailing and failing human ventricular myocardium: coupling of both receptor subtypes to muscle contraction and selective beta 1-receptor down-regulation in heart failure

1 reference

12 December 2020

Cardiac beta receptors--experimental aspects

1 reference

12 December 2020

The affinity of (-)-propranolol for beta 1- and beta 2-adrenoceptors of human heart. Differential antagonism of the positive inotropic effects and adenylate cyclase stimulation by (-)-noradrenaline and (-)-adrenaline

1 reference

12 December 2020

Tight control of gene expression in mammalian cells by tetracycline-responsive promoters

1 reference

12 December 2020

Decreased Catecholamine Sensitivity and β-Adrenergic-Receptor Density in Failing Human Hearts

1 reference

12 December 2020

(--)-Timolol is a more potent antagonist of the positive inotropic effects of (--)-adrenaline than of those of (--)-noradrenaline in human atrium

1 reference

12 December 2020

beta1-adrenergic receptors mediate beta3-adrenergic-independent effects of CGP 12177 in brown adipose tissue

1 reference

12 December 2020

(-)-CGP 12177 causes cardiostimulation and binds to cardiac putative beta 4-adrenoceptors in both wild-type and beta 3-adrenoceptor knockout mice.

1 reference

12 December 2020

Comparison of the affinity of beta-blockers for two states of the beta 1-adrenoceptor in ferret ventricular myocardium

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12 December 2020

Differences between the third cardiac beta-adrenoceptor and the colonic beta 3-adrenoceptor in the rat.

1 reference

12 December 2020

Stimulant and blocking effects of optical isomers of pindolol on the sinoatrial node and trachea of guinea pig. Role of ?-adrenoceptor subtypes in the dissociation between blockade and stimulation

1 reference

12 December 2020

Is there a third heart beta-adrenoceptor?

1 reference

12 December 2020

Putative beta 4-adrenoceptors in rat ventricle mediate increases in contractile force and cell Ca2+: comparison with atrial receptors and relationship to (-)-[3H]-CGP 12177 binding

1 reference

12 December 2020

(-)-CGP 12177 increases contractile force and hastens relaxation of human myocardial preparations through a propranolol-resistant state of the beta 1-adrenoceptor

1 reference

12 December 2020

An initial characterization of human heart beta-adrenoceptors and their mediation of the positive inotropic effects of catecholamines

1 reference

12 December 2020

Validity of (-)-[3H]-CGP 12177A as a radioligand for the 'putative beta4-adrenoceptor' in rat atrium

1 reference

12 December 2020

The putative beta4-adrenergic receptor is a novel state of the beta1-adrenergic receptor

1 reference

12 December 2020

Mode of action of (-)-pindolol on feline and human myocardium

1 reference

12 December 2020

Comparative pharmacology of human beta-adrenergic receptor subtypes--characterization of stably transfected receptors in CHO cells

1 reference

12 December 2020

CGP-12177. A hydrophilic beta-adrenergic receptor radioligand reveals high affinity binding of agonists to intact cells.

1 reference

12 December 2020

Desensitization and resensitization of beta 1- and putative beta 4-adrenoceptor mediated responses occur in parallel in a rat model of cardiac failure

1 reference

12 December 2020

Stimulation of cyclic AMP-dependent protein kinase in rat atria by (-)-CGP 12177 through an atypical beta-adrenoceptor

1 reference

12 December 2020

Agonist actions of "beta-blockers" provide evidence for two agonist activation sites or conformations of the human beta1-adrenoceptor

1 reference

12 December 2020

Action potential shortening through the putative beta4-adrenoceptor in ferret ventricle: comparison with beta1- and beta2-adrenoceptor-mediated effects

1 reference

12 December 2020

Blockade of putative beta4- and beta1-adrenoceptors by carvedilol in ferret myocardium

1 reference

12 December 2020

Anomalous behavior of CGP 12177A on beta 1-adrenergic receptors

1 reference

12 December 2020

Contribution of beta 1- and beta 2-adrenoceptors of human atrium and ventricle to the effects of noradrenaline and adrenaline as assessed with (-)-atenolol

1 reference

12 December 2020

Intrinsic sympathomimetic activity of (-)-pindolol mediated through a (-)-propranolol-resistant site of the beta1-adrenoceptor in human atrium and recombinant receptors

1 reference

12 December 2020

(-)-CGP 12177-induced increase of human atrial contraction through a putative third beta-adrenoceptor

1 reference

12 December 2020

Abolition of (-)-CGP 12177-evoked cardiostimulation in double beta1/beta2-adrenoceptor knockout mice. Obligatory role of beta1-adrenoceptors for putative beta4-adrenoceptor pharmacology

1 reference

12 December 2020

10.1007/S00210-004-0884-Y

Identifiers

DOI

1 reference

6 December 2017

1 reference

PubMed ID

15060759