(Q48166685)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22539833%20AND%20SRC:MED&resulttype=core&format=json

30 January 2020

title

Benzodiazepines modulate GABAA receptors by regulating the preactivation step after GABA binding (English)

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30 January 2020

1

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30 January 2020

author name string

Michael J Lumb

series ordinal

2

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22539833%20AND%20SRC:MED&resulttype=core&format=json

30 January 2020

Trevor G Smart

series ordinal

3

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30 January 2020

language of work or name

English

0 references

publication date

1 April 2012

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30 January 2020

published in

Journal of Neuroscience

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30 January 2020

volume

32

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30 January 2020

issue

17

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30 January 2020

page(s)

5707-5715

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Allosteric modulators affect the efficacy of partial agonists for recombinant GABA(A) receptors

30 January 2020

cites work

1 reference

12 December 2020

Agonist Trapping by GABAA Receptor Channels.

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12 December 2020

Drug interactions at GABA(A) receptors

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12 December 2020

Mapping of the benzodiazepine recognition site on GABA(A) receptors

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12 December 2020

Comparative modeling of GABA(A) receptors: limits, insights, future developments.

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12 December 2020

Activation of single heteromeric GABA(A) receptor ion channels by full and partial agonists

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12 December 2020

Techniques: Use of concatenated subunits for the study of ligand-gated ion channels.

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12 December 2020

Benzodiazepines affect channel opening of GABA A receptors induced by either agonist binding site

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12 December 2020

Classic benzodiazepines modulate the open-close equilibrium in alpha1beta2gamma2L gamma-aminobutyric acid type A receptors

1 reference

12 December 2020

Benzodiazepine modulation of partial agonist efficacy and spontaneously active GABA(A) receptors supports an allosteric model of modulation

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12 December 2020

Modes and models of GABA(A) receptor gating

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12 December 2020

A GABA(A) receptor of defined subunit composition and positioning: concatenation of five subunits.

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12 December 2020

Mechanism of action of benzodiazepines on GABAA receptors

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12 December 2020

Tandem couture: Cys-loop receptor concatamer insights and caveats

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12 December 2020

X-ray structure of a prokaryotic pentameric ligand-gated ion channel

1 reference

12 December 2020

On the nature of partial agonism in the nicotinic receptor superfamily

1 reference

12 December 2020

X-ray structure of a pentameric ligand-gated ion channel in an apparently open conformation

1 reference

12 December 2020

Detection and trapping of intermediate states priming nicotinic receptor channel opening

1 reference

12 December 2020

Use of concatamers to study GABAA receptor architecture and function: application to delta-subunit-containing receptors and possible pitfalls

1 reference

12 December 2020

The activation mechanism of alpha1beta2gamma2S and alpha3beta3gamma2S GABAA receptors

1 reference

12 December 2020

Binding, activation and modulation of Cys-loop receptors.

1 reference

12 December 2020

Distinct activities of GABA agonists at synaptic- and extrasynaptic-type GABAA receptors.

1 reference

12 December 2020

The short splice variant of the gamma 2 subunit acts as an external modulator of GABA(A) receptor function

1 reference

12 December 2020

Diversity of structure and function of alpha1alpha6beta3delta GABAA receptors: comparison with alpha1beta3delta and alpha6beta3delta receptors

1 reference

12 December 2020

Occupation of either site for the neurosteroid allopregnanolone potentiates the opening of the GABAA receptor induced from either transmitter binding site

1 reference

12 December 2020

Beyond classical benzodiazepines: novel therapeutic potential of GABAA receptor subtypes

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12 December 2020

Differential regulation of gamma-aminobutyric acid receptor channels by diazepam and phenobarbital

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12 December 2020

Diazepam and (--)-pentobarbital: fluctuation analysis reveals different mechanisms for potentiation of gamma-aminobutyric acid responses in cultured central neurons

1 reference

12 December 2020

GABAA receptor needs two homologous domains of the beta-subunit for activation by GABA but not by pentobarbital.

1 reference

12 December 2020

Benzodiazepine and beta-carboline regulation of single GABAA receptor channels of mouse spinal neurones in culture.

1 reference

12 December 2020

Structure and pharmacology of vertebrate GABAA receptor subtypes.

1 reference

12 December 2020

10.1523/JNEUROSCI.5663-11.2012

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22539833%20AND%20SRC:MED&resulttype=core&format=json

30 January 2020

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30 January 2020

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