(Q48397096)

11 February 2018

title

Synthesis and characterization of two PET radioligands for the metabotropic glutamate 1 (mGlu1) receptor (English)

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11 February 2018

author name string

Yiyun Huang

1

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Rajesh Narendran

2

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Francois Bischoff

3

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Ningning Guo

4

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Sung A Bae

5

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Dah-Ren Hwang

6

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Anne S Lesage

7

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Marc Laruelle

8

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publication date

29 September 2012

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11 February 2018

published in

Synapse

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volume

66

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issue

12

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page(s)

1002-1014

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PET studies of binding competition between endogenous dopamine and the D1 radiotracer [11C]NNC 756.

cites work

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21 January 2018

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Characterization of 1-(2-[18F] fluoro-3-pyridyl)-4-(2-isopropyl-1-oxo- isoindoline-5-yl)-5-methyl-1H-1,2,3-triazole, a PET ligand for imaging the metabotropic glutamate receptor type 1 in rat and monkey brains

21 January 2018

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Synthesis and evaluation of novel radioligands for positron emission tomography imaging of metabotropic glutamate receptor subtype 1 (mGluR1) in rodent brain

21 January 2018

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Evaluation of ultrafiltration for the free-fraction determination of single photon emission computed tomography (SPECT) radiotracers: beta-CIT, IBF, and iomazenil

21 January 2018

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[(3)H]-M-MPEP, a potent, subtype-selective radioligand for the metabotropic glutamate receptor subtype 5.

21 January 2018

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2-Methyl-6-(phenylethynyl)-pyridine (MPEP), a potent, selective and systemically active mGlu5 receptor antagonist

21 January 2018

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Synthesis, characterization, and monkey PET studies of [¹⁸F]MK-1312, a PET tracer for quantification of mGluR1 receptor occupancy by MK-5435.

21 January 2018

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A positron emission tomography radioligand for the in vivo labeling of metabotropic glutamate 1 receptor: (3-ethyl-2-[11C]methyl-6-quinolinyl)(cis- 4-methoxycyclohexyl)methanone

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LY341495 is a nanomolar potent and selective antagonist of group II metabotropic glutamate receptors

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21 January 2018

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21 January 2018

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Characterization of [(3)H]Quisqualate binding to recombinant rat metabotropic glutamate 1a and 5a receptors and to rat and human brain sections

21 January 2018

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21 January 2018

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21 January 2018

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Synthesis, in vitro and in vivo evaluation of [11C]MMTP: a potential PET ligand for mGluR1 receptors

21 January 2018

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21 January 2018

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21 January 2018

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Imaging for metabotropic glutamate receptor subtype 1 in rat and monkey brains using PET with [18F]FITM.

21 January 2018

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Radiosynthesis and preliminary evaluation of 4-[18F]fluoro-N-[4-[6-(isopropylamino)pyrimidin-4-yl]-1,3-thiazol-2-yl]-N-methylbenzamide as a new positron emission tomography ligand for metabotropic glutamate receptor subtype 1.

21 January 2018

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21 January 2018

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21 January 2018

Identifiers

DOI

10.1002/SYN.21606

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11 February 2018

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11 February 2018