(Q49073474)

18 February 2018

title

Desirability function combining metabolic stability and functionality of peptides (English)

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18 February 2018

author name string

Sylvia Van Dorpe

1

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18 February 2018

Antita Adriaens

2

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Simon Vermeire

3

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18 February 2018

Ingeborgh Polis

4

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18 February 2018

Kathelijne Peremans

5

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Bart De Spiegeleer

6

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18 February 2018

publication date

4 February 2011

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18 February 2018

Journal of Peptide Science

published in

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18 February 2018

volume

17

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18 February 2018

issue

5

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18 February 2018

page(s)

398-404

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18 February 2018

Design of peptide oxytocin antagonists with strikingly higher affinities and selectivities for the human oxytocin receptor than atosiban

cites work

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Development of simplified vasoactive intestinal peptide analogs with receptor selectivity and stability for human vasoactive intestinal peptide/pituitary adenylate cyclase-activating polypeptide receptors

21 January 2018

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Comparison of opioid receptor binding in horse, guinea pig, and rat cerebral cortex and cerebellum

21 January 2018

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Mutagenesis studies of neuropeptide S identify a suitable peptide tracer for neuropeptide S receptor binding studies and peptides selectively activating the I(107) variant of human neuropeptide S receptor

21 January 2018

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Interaction of agonist peptide [3H]Tyr-D-Ala-Phe-Phe-NH2 with mu-opioid receptor in rat brain and CHO-mu/1 cell line

21 January 2018

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Receptor binding and biological activity of the dermorphin analog Tyr-D-Arg(2)-Phe-Sar (TAPS).

21 January 2018

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Josef Rudinger Memorial Lecture 2002. The chemistry of the opioid receptor binding sites

21 January 2018

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Delivery of peptides and proteins through the blood-brain barrier

21 January 2018

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Transport of opioid peptides into the central nervous system.

21 January 2018

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Structure and function of the blood-brain barrier

21 January 2018

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Tight junctions of the blood-brain barrier

21 January 2018

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Differential BBB interactions of three ingestive peptides: obestatin, ghrelin, and adiponectin

21 January 2018

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Evidence that [125I]N-Tyr-delta sleep-inducing peptide crosses the blood-brain barrier by a non-competitive mechanism

21 January 2018

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Radiolabeled peptides in the diagnosis and therapy of oncological diseases

21 January 2018

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Synthesis, radiolabeling and receptor binding of [3H][(1S,2R)ACPC2]endomorphin-2.

21 January 2018

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21 January 2018

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Effect of guanidino modification and proline substitution on the in vitro stability and blood-brain barrier permeability of endomorphin II.

21 January 2018

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Novel glycosylated VIP analogs: synthesis, biological activity, and metabolic stability

21 January 2018

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In vitro metabolism of opioid tetrapeptide agonists in various tissues and subcellular fractions from rats

21 January 2018

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New trends in the development of opioid peptide analogues as advanced remedies for pain relief

21 January 2018

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Synthesis and biological activity of homoarginine-containing opioid peptides

21 January 2018

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In vitro metabolic stability of obestatin: kinetics and identification of cleavage products

21 January 2018

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Analytical characterization and comparison of the blood-brain barrier permeability of eight opioid peptides

21 January 2018

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Hydrophilic interaction LC of peptides: columns comparison and clustering

21 January 2018

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Evolving molecules using multi-objective optimization: applying to ADME/Tox

21 January 2018

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Impurity profiling quality control testing of synthetic peptides using liquid chromatography-photodiode array-fluorescence and liquid chromatography-electrospray ionization-mass spectrometry: the obestatin case

21 January 2018

1 reference

Simultaneous optimization of the resolution and analysis time in micellar liquid chromatography of phenyl thiohydantoin amino acids using Derringer's desirability function

21 January 2018

1 reference

Zyklophin, a systemically active selective kappa opioid receptor peptide antagonist with short duration of action

21 January 2018

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[Dmt1, d-1-Nal3]morphiceptin, a novel opioid peptide analog with high analgesic activity

21 January 2018

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Development of opioid peptide analogs for pain relief

21 January 2018

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Synthesis and pharmacological properties of a new fluorescent opioid peptide analog.

21 January 2018

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21 January 2018

Identifiers

DOI

10.1002/PSC.1323

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18 February 2018

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18 February 2018