(Q52877248)

9 May 2018

title

Structure-activity relationships of the inhibition of human placental aromatase by imidazole drugs including ketoconazole (English)

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

5 January 2023

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https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

5 January 2023

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

5 January 2023

author name string

M. Ayub

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A3398530

5 January 2023

M. J. Levell

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A3398530

5 January 2023

language of work or name

English

1 reference

National Center for Biotechnology Information

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/esummary.fcgi?db=pubmed&retmode=json&id=3398530

5 January 2023

publication date

1 July 1988

1 reference

9 May 2018

full work available at URL

https://api.elsevier.com/content/article/PII:0022473188902075?httpAccept=text/xml

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https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

https://api.elsevier.com/content/article/PII:0022473188902075?httpAccept=text/plain

5 January 2023

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

The Journal of Steroid Biochemistry

5 January 2023

published in

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9 May 2018

volume

31

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9 May 2018

page(s)

65-72

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9 May 2018

issue

1

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9 May 2018

In vitro and in vivo effects of the antimycotic drug ketoconazole on sterol synthesis

cites work

4

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Gynecomastia with ketoconazole

5 January 2023

6

1 reference

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Effects of high dose ketoconazole therapy on the main plasma testicular and adrenal steroids in previously untreated prostatic cancer patients

5 January 2023

8

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Imidazole antimycotics: inhibitors of steroid aromatase

5 January 2023

12

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Inhibition of ovarian aromatase by ketoconazole

5 January 2023

13

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Ketoconazole and other imidazole derivatives as inhibitors of steroidogenesis

5 January 2023

14

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Aromatase inhibitors and their potential clinical significance

5 January 2023

16

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Aromatase inhibitors and benign prostatic hyperplasia

5 January 2023

17

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Stereoselective Inhibition of Aromatase by Enantiomers of Aminoglutethimide*

5 January 2023

18

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Inactivation of aromatase in vitro by 4-hydroxy-4-androstene-3,17-dione and 4-acetoxy-4-androstene-3,17-dione and sustained effects in vivo

5 January 2023

19

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Inhibition of testicular 17 alpha-hydroxylase and 17,20-lyase but not 3 beta-hydroxysteroid dehydrogenase-isomerase or 17 beta-hydroxysteroid oxidoreductase by ketoconazole and other imidazole drugs.

5 January 2023

20

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Effect of ketoconazole on placental aromatase, 3 beta-hydroxysteroid dehydrogenase-isomerase and 17 beta-hydroxysteroid dehydrogenase

5 January 2023

21

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Protein measurement with the Folin phenol reagent

5 January 2023

22

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Substrate specificity of the placental microsomal aromatase

5 January 2023

26

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https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Enzymatic androgen assay: some properties of human placental microsomal aromatase

5 January 2023

27

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Inhibition of estrogen synthetase (aromatase) by 4-cyclohexylaniline

5 January 2023

28

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https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

The effect of ketoconazole on adrenal and testicular steroidogenesis in vitro

5 January 2023

30

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Human placental Δ5-3β hydroxysteroid dehydrogenase activity (Δ5-33 HSDH): Intracellular distribution, kinetic properties, retroinhibition and influence of membrane delipidation

5 January 2023

31

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

The influence of 4-hydroxy-4-androstene-3,17-dione on androgen metabolism and action in cultured human foreskin fibroblasts

5 January 2023

32

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Effect of 1,4,6-androstatriene-3,17-dione (ATD), 4-hydroxy-4-androstene-3,17-dione (4-OH-A) and 4-acetoxy-4-androstene-3,17-dione (4-Ac-A) on the 5 alpha-reduction of androgens in the rat prostate

5 January 2023

33

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Effects of 4-hydroxy-4-androstene-3,17-dione and 10-propargylestr-4-ene-3,17-dione on the metabolism of androstenedione in human breast carcinoma and breast adipose tissues

5 January 2023

34

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Effect of a single administration of ketoconazole on total and physiologically free plasma testosterone and 17 beta-oestradiol levels in healthy male volunteers

5 January 2023

35

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Regression of metastatic adrenal carcinoma during palliative ketoconazole treatment

5 January 2023

38

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Adrenal rest tumor of the liver causing Cushing's syndrome: treatment with ketoconazole preceding an apparent surgical cure

5 January 2023

39

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Effects of tioconazole on parturition and serum levels of 17 beta-oestradiol, progesterone, LH and PRL in the rat

5 January 2023

41

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Imidazole antifungal agents reduce production of 17 beta-oestradiol by rat ovaries in vitro

5 January 2023

42

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Site of Action of Low Dose Ketoconazole on Androgen Biosynthesis in Men*

5 January 2023

44

57

732

Santen

1983

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Long-term experience with high dose ketoconazole therapy in patients with stage D2 prostatic carcinoma.

5 January 2023

45

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Ketoconazole therapy for advanced prostatic cancer: feasibility and treatment results

5 January 2023

46

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Ketoconazole in the management of precocious puberty not responsive to LHRH-analogue therapy

5 January 2023

47

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Gonadotropin-independent precocious puberty ("testotoxicosis"): influence of maturational status on response to ketoconazole

5 January 2023

48

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https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Ketoconazole for hirsutism

5 January 2023

49

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https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Hepatic reactions associated with ketoconazole in the United Kingdom

5 January 2023

50

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Action of imidazole-containing antifungal drugs

5 January 2023

51

1 reference

https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

Mechanism of action of antifungal drugs, with special reference to the imidazole derivatives.

5 January 2023

52

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https://api.crossref.org/works/10.1016/0022-4731(88)90207-5

5 January 2023

Identifiers

1 reference

9 May 2018

1 reference

9 May 2018