(Q61066436)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10896108%20AND%20SRC:MED&resulttype=core&format=json

8 November 2019

title

Aziridinyl peptides as inhibitors of cysteine proteases: effect of a free carboxylic acid function on inhibition (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10896108%20AND%20SRC:MED&resulttype=core&format=json

8 November 2019

0 references

0 references

pharmaceutical science

0 references

author

Tanja Schirmeister

series ordinal

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10896108%20AND%20SRC:MED&resulttype=core&format=json

8 November 2019

author name string

M Peric

series ordinal

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10896108%20AND%20SRC:MED&resulttype=core&format=json

8 November 2019

language of work or name

English

0 references

publication date

1 June 2000

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10896108%20AND%20SRC:MED&resulttype=core&format=json

Bioorganic & Medicinal Chemistry

8 November 2019

published in

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10896108%20AND%20SRC:MED&resulttype=core&format=json

8 November 2019

volume

8

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10896108%20AND%20SRC:MED&resulttype=core&format=json

8 November 2019

issue

6

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10896108%20AND%20SRC:MED&resulttype=core&format=json

8 November 2019

page(s)

1281-1291

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10896108%20AND%20SRC:MED&resulttype=core&format=json

Enzyme-substrate interactions in the hydrolysis of peptides by cathepsins B and H from rat liver

8 November 2019

cites work

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Crystal structure of human osteoclast cathepsin K complex with E-64

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

The crystal structure of human cathepsin L complexed with E-64

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Acid sulphydryl protease from calf lymph nodes

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Human cathepsins F and W: A new subgroup of cathepsins

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Cynomolgus monkey (Macaca fascicularis) cathepsin K: cloning, expression, purification, and activation

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Human cathepsin V functional expression, tissue distribution, electrostatic surface potential, enzymatic characterization, and chromosomal localization

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Genomic structure, chromosomal localization, and expression of human cathepsin W.

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Human cathepsin X: a novel cysteine protease of the papain family with a very short proregion and unique insertions

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Cathepsin Z, a novel human cysteine proteinase with a short propeptide domain and a unique chromosomal location

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Effects on Cathepsin B, H, and D in Pectoral Muscle of Dystrophic Chickens (Line 413) of In Vivo Administration of E-64-c (N-[N-(L-3-Transcarboxyoxirane-2-Carbonyl)-L-Leucyl]-3-Methyl-Butylamine)1

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Human cathepsin B and cysteine proteinase inhibitors (CPIs) in inflammatory and metabolic joint diseases

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Mode of activation of the precursor to cathepsin L: implication for matrix degradation in arthritis

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Cathepsin K, but not cathepsins B, L, or S, is abundantly expressed in human osteoclasts

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Aziridine Analogs of [[trans-(Epoxysuccinyl)-L-leucyl]amino]-4-guanidinobutane (E-64) as Inhibitors of Cysteine Proteases

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Aziridine-2,3-dicarboxylic Acid Derivatives as Inhibitors of Papain

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

New Peptidic Cysteine Protease Inhibitors Derived from the Electrophilic α-Amino Acid Aziridine-2,3-dicarboxylic Acid

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Mechanistic studies on the inactivation of papain by epoxysuccinyl inhibitors

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Families of cysteine peptidases.

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Determination of the rate constant of enzyme modification by measuring the substrate reaction in the presence of the modifier.

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

L-trans-Epoxysuccinyl-leucylamido(4-guanidino)butane (E-64) and its analogues as inhibitors of cysteine proteinases including cathepsins B, H and L

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Epoxysuccinyl dipeptides as selective inhibitors of cathepsin B

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

E-64 analogues as inhibitors of cathepsin B. On the role of the absolute configuration of the epoxysuccinyl group

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Crystal structure of a papain-E-64 complex

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Mode of binding of E-64-c, a potent thiol protease inhibitor, to papain as determined by X-ray crystal analysis of the complex

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Crystal structure of cathepsin B inhibited with CA030 at 2.0-A resolution: A basis for the design of specific epoxysuccinyl inhibitors

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Binding mode of CA074, a specific irreversible inhibitor, to bovine cathepsin B as determined by X-ray crystal analysis of the complex

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

Demonstration that 1-trans-epoxysuccinyl-L-leucylamido-(4-guanidino) butane (E-64) is one of the most effective low Mr inhibitors of trypsin-catalysed hydrolysis. Characterization by kinetic analysis and by energy minimization and molecular dynamics

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

The synthesis and properties of peptidylmethylsulphonium salts with two cationic residues as potential inhibitors of prohormone processing

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

The Practice of Peptide Synthesis

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

The refined 2.15 A X-ray crystal structure of human liver cathepsin B: the structural basis for its specificity

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2800%2900058-4

7 January 2021

10.1016/S0968-0896(00)00058-4

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10896108%20AND%20SRC:MED&resulttype=core&format=json

8 November 2019

1 reference