(Q70067192)

English

In vivo labelling of rat brain dopamine D-2 receptors. Stereoselective blockade by the D-2 antagonist raclopride and its enantiomer of 3H-spiperone, 3H-N,N-propylnorapomorphine and 3H-raclopride binding in the rat brain

scientific article published on 01 January 1988

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scholarly article

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Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2974879%20AND%20SRC:MED&resulttype=core&format=json

8 October 2019

In vivo labelling of rat brain dopamine D-2 receptors. Stereoselective blockade by the D-2 antagonist raclopride and its enantiomer of 3H-spiperone, 3H-N,N-propylnorapomorphine and 3H-raclopride binding in the rat brain (English)

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2974879%20AND%20SRC:MED&resulttype=core&format=json

8 October 2019

stereoselectivity

1 reference

based on heuristic

inferred from title

1 reference

based on heuristic

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author name string

C Köhler

1

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2974879%20AND%20SRC:MED&resulttype=core&format=json

8 October 2019

G Karlsson-Boethius

2

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2974879%20AND%20SRC:MED&resulttype=core&format=json

8 October 2019

publication date

1 January 1988

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Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2974879%20AND%20SRC:MED&resulttype=core&format=json

8 October 2019

73

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2974879%20AND%20SRC:MED&resulttype=core&format=json

8 October 2019

2

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Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2974879%20AND%20SRC:MED&resulttype=core&format=json

8 October 2019

87-100

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2974879%20AND%20SRC:MED&resulttype=core&format=json

8 October 2019

3H-spiroperidol labels dopamine receptors in pituitary and brain

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

3HN-propylapomorphine and 3Hspiperone binding in brain indicate two states of the D2-dopamine receptor

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Autoradiographic distribution of the D1 agonist [3H]SKF 38393, in the rat brain and spinal cord. Comparison with the distribution of D2 dopamine receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Serotonergic component of neuroleptic receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Heterogeneous distribution of dopamine D2 receptors within the rat striatum as revealed by autoradiography of [3H]N-n-propylnorapomorphine binding sites

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Brain dopamine receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Potential neuroleptic agents. 2,6-Dialkoxybenzamide derivatives with potent dopamine receptor blocking activities

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Autoradiographic study of 14C-sulpiride in monkey

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Differential anatomical location of [3H]-N,n-propylnorapomorphine and [3H]-spiperone binding sites in the striatum and substantia nigra of the rat

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Tracer and maximal specific binding of tritiated spiperone or N-n-propylnorapomorphine to quantify dopamine receptors in rat brain regions in vivo

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Dopamine receptor binding in vivo: The feasibility of autoradiographic studies

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Potential neuroleptic agents. 4. Chemistry, behavioral pharmacology, and inhibition of [3H]spiperone binding of 3,5-disubstituted N-[(1-ethyl-2-pyrrolidinyl)methyl]-6-methoxysalicylamides

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

[3H]Spiroperidol binding to a putative dopaminergic receptor in rat pituitary gland

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Comparisons between the in vitro binding of two substituted benzamides and two butyrophenones to dopamine-D2 receptors in the rat striatum

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Dopamine D2 receptors and dopamine metabolism. Relationship between biochemical and behavioural effects of substituted benzamide drugs.

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Contamination of serotonin-2 binding sites by an alpha-1 adrenergic component in assays with (3H) spiperone

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Differential labelling of dopamine receptors in rat brain in vivo: Comparison of [3H]piribedil, [3H]S 3608 and [3H]N,n-propylnorapomorphine

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Typical and atypical antipsychotic occupancy of D2 and S2 receptors: an autoradiographic analysis in rat brain

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

In vivo stereospecific [3H]spiperone binding in rat brain: characteristics, regional distribution, kinetics and pharmacological properties

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Classification of neuroleptic drugs according to their ability to inhibit apomorphine-induced locomotion and gnawing: Evidence for two different mechanisms of action

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Autoradiographic visualization of dopamine D-2 receptors in the monkey brain using the selective benzamide drug [3H]raclopride

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

In situ molecular size of agonist dopamine D-2 binding sites in rat striatum

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The selective dopamine D2 receptor antagonist raclopride discriminates between dopamine-mediated motor functions.

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Substituted benzamides as ligands for visualization of dopamine receptor binding in the human brain by positron emission tomography

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Regional displacement by sulpiride of [3H]spiperone binding in vivo. Biochemical and behavioural evidence for a preferential action of limbic and nigral dopamine receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Quantification of in vivo spiperone binding in the rat striatum after lesions produced by kainate or decortication

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Studies on the Mechanism of Action of Substituted Benzamide Drugs

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Specific in vivo binding of neuroleptic drugs in rat brain

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

In vivo binding of spiroperidol and bromospiroperidol at low drug loadings

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Regional in vivo binding of [3H]N-propylnorapomorphine in the mouse brain. Evidence for labelling of central dopamine receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Regional blockade by neuroleptic drugs ofin vivo 3H-spiperone binding in the rat brain. Relation to blockade of apomorphine induced hyperactivity and stereotypies

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The substituted benzamides - a novel class of dopamine antagonists

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Regional in vivo binding of the substituted benzamide [3H]eticlopride in the rat brain: evidence for selective labelling of dopamine receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Specific in vitro and in vivo binding of 3H-raclopride. A potent substituted benzamide drug with high affinity for dopamine D-2 receptors in the rat brain

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Characterization of normal and supersensitive dopamine receptors: Effects of ergot drugs and neuropeptides

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Spiperone: a ligand of choice for neuroleptic receptors. 1. Kinetics and characteristics of in vitro binding

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Dopamine receptor binding on intact cells. Absence of a high-affinity agonist-receptor binding state

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Remoxipride, a new potential antipsychotic compound with selective antidopaminergic actions in the rat brain

1 reference

https://pubmed.ncbi.nlm.nih.gov/2974879

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1007/BF01243380

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2974879%20AND%20SRC:MED&resulttype=core&format=json

8 October 2019

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2974879%20AND%20SRC:MED&resulttype=core&format=json

8 October 2019

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