(Q70162862)

English

Correlation between the negative inotropic potency and binding parameters of 1,4-dihydropyridine and phenylalkylamine calcium channel blockers in cat heart

scientific article published on 01 November 1986

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scholarly article

1 reference

Europe PubMed Central

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:3027587%20AND%20SRC:MED&resulttype=core&format=json

9 October 2019

Correlation between the negative inotropic potency and binding parameters of 1,4-dihydropyridine and phenylalkylamine calcium channel blockers in cat heart (English)

1 reference

Europe PubMed Central

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:3027587%20AND%20SRC:MED&resulttype=core&format=json

9 October 2019

Hartmut H. Glossmann

2

1 reference

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9 October 2019

author name string

A Goll

1

1 reference

Europe PubMed Central

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9 October 2019

R Mannhold

3

1 reference

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9 October 2019

publication date

1 November 1986

1 reference

Europe PubMed Central

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9 October 2019

Naunyn-Schmiedeberg's Archives of Pharmacology

1 reference

Europe PubMed Central

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9 October 2019

334

1 reference

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9 October 2019

303-312

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9 October 2019

3

1 reference

Europe PubMed Central

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9 October 2019

https://scigraph.springernature.com/pub.10.1007/bf00508786

0 references

High affinity specific [3H] (+)PN 200-110 binding to dihydropyridine receptors associated with calcium channels in rat cerebral cortex and heart

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Comparative pharmacology of calcium antagonists: Nifedipine, verapamil and diltiazem

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Relationship between the stereoselective negative inotropic effects of verapamil enantiomers and their binding to putative calcium channels in human heart

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Nitrendipine block of cardiac calcium channels: high-affinity binding to the inactivated state

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Calculating the dissociation constant of an unlabeled compound from the concentration required to displace radiolabel binding by 50%

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Specific Pharmacology of Calcium in Myocardium, Cardiac Pacemakers, and Vascular Smooth Muscle

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The effects of nimodipine, its optical isomers and metabolites on isolated vascular smooth muscle

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Mechanism of calcium channel blockade by verapamil, D600, diltiazem and nitrendipine in single dialysed heart cells

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Simultaneous analysis of families of sigmoidal curves: application to bioassay, radioligand assay, and physiological dose-response curves

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Modulation of calcium ion influx by the 1,4-dihydropyridines nifedipine and BAY K 8644

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Target size analysis and molecular properties of Ca2+ channels labelled with [3H]verapamil.

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Diltiazem potentiates the negative inotropic action of nimodipine in heart

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Different modes of Ca channel gating behaviour favoured by dihydropyridine Ca agonists and antagonists

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Molecular pharmacology of the calcium channel: evidence for subtypes, multiple drug-receptor sites, channel subunits, and the development of a radioiodinated 1,4-dihydropyridine calcium channel label, [125I]iodipine.

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Temperature-dependent modulation of [3H]nitrendipine binding by the calcium channel antagonists verapamil and diltiazem in rat brain synaptosomes.

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Characterization of the binding sites for nimodipine and (-)-desmethoxyverapamil in bovine cardiac sarcolemma

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Binding of [3H]nimodipine to cardiac and smooth muscle membranes

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Characterization of binding of the Ca++ channel antagonist, [3H]nitrendipine, to guinea-pig ileal smooth muscle

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identification of putative calcium channels in skeletal muscle microsomes.

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Characterization of verapamil binding sites in cardiac membrane vesicles

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Principles and practice of Hansch analysis: a guide to structure-activity correlation for the medicinal chemist

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

[3H]diltiazem binding to calcium channel antagonists recognition sites in rat cerebral cortex.

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Voltage-dependent block of calcium channel current in the calf cardiac Purkinje fiber by dihydropyridine calcium channel antagonists

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identification of Voltage Operated Calcium Channels by Binding Studies: Differentiation of Subclasses of Calcium Antagonist Drugs with3H-Nimodipine Radioligand Binding

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

(-)-[3H]Desmethoxyverapamil, a novel Ca2+ channel probe. Binding characteristics and target size analysis of its receptor in skeletal muscle

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Temperature‐dependent regulation of d‐cis‐[3H]diltiazem binding to Ca2+ channels by 1,4‐dihydropyridine channel agonists and antagonists

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

(?)-3H-desmethoxyverapamil labelling of putative calcium channels in brain: autoradiographic distribution and allosteric coupling to 1,4-dihydropyridine and diltiazem binding sites

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The optical isomers of the 1,4-dihydropyridine BAY K 8644 show opposite effects on Ca channels

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Calcium antagonists. Some chemical-pharmacologic aspects

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Stereoselective and non-stereoselective effects of D 600 (methoxyverapamil) in smooth muscle preparations.

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Protein measurement with the Folin phenol reagent

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Calcium channels and calcium channel drugs: recent biochemical and biophysical findings

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Calcium-antagonist drugs. Receptor interactions that clarify therapeutic effects

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Evidence of multiple receptor sites within the putative calcium channel.

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Assessment of "Ca2+ -antagonist" effects of drugs in K+ -depolarized smooth muscle. Differentiation of antagonist subgroups.

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

[3H]-Nitrendipine, a potent calcium antagonist, binds with high affinity to cardiac membranes.

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Differential labelling of putative skeletal muscle calcium channels by [3H]-nifedipine, [3H]-nitrendipine, [3H]-nimodipine and [3H]-PN 200 110

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The influence of aromatic substitution on the negative inotropic action of verapamil in the isolated cat papillary muscle

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Mechanism of Action of Calcium-Channel-Blocking Agents

1 reference

https://pubmed.ncbi.nlm.nih.gov/3027587

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1007/BF00508786

1 reference

Europe PubMed Central

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:3027587%20AND%20SRC:MED&resulttype=core&format=json

9 October 2019

1 reference

Europe PubMed Central

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:3027587%20AND%20SRC:MED&resulttype=core&format=json

9 October 2019

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