(Q73390518)

English

Three-dimensional quantitative structure-activity relationships study on HIV-1 reverse transcriptase inhibitors in the class of dipyridodiazepinone derivatives, using comparative molecular field analysis

scientific article published on 01 December 2000

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scholarly article

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Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11155314%20AND%20SRC:MED&resulttype=core&format=json

3 November 2019

Three-dimensional quantitative structure-activity relationships study on HIV-1 reverse transcriptase inhibitors in the class of dipyridodiazepinone derivatives, using comparative molecular field analysis (English)

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11155314%20AND%20SRC:MED&resulttype=core&format=json

3 November 2019

Supa Hannongbua

2

1 reference

Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11155314%20AND%20SRC:MED&resulttype=core&format=json

3 November 2019

author name string

Pungpo P

1

1 reference

Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11155314%20AND%20SRC:MED&resulttype=core&format=json

3 November 2019

publication date

1 December 2000

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11155314%20AND%20SRC:MED&resulttype=core&format=json

3 November 2019

Journal of Molecular Graphics & Modelling

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11155314%20AND%20SRC:MED&resulttype=core&format=json

3 November 2019

18

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Europe PubMed Central

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3 November 2019

6

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Europe PubMed Central

PubMed publication ID

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3 November 2019

581-90, 601

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11155314%20AND%20SRC:MED&resulttype=core&format=json

3 November 2019

Inhibition of HIV-1 Replication by a Nonnucleoside Reverse Transcriptase Inhibitor

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

Crystal structure at 3.5 A resolution of HIV-1 reverse transcriptase complexed with an inhibitor

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

Structure of the binding site for nonnucleoside inhibitors of the reverse transcriptase of human immunodeficiency virus type 1

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

A novel dipyridodiazepinone inhibitor of HIV-1 reverse transcriptase acts through a nonsubstrate binding site

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

Human immunodeficiency virus type 1 mutants resistant to nonnucleoside inhibitors of reverse transcriptase arise in tissue culture

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

A check on rational drug design: molecular simulation of the allosteric inhibition of HIV-1 reverse transcriptase

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

Human immunodeficiency virus 1 (HIV-1)-specific reverse transcriptase (RT) inhibitors may suppress the replication of specific drug-resistant (E138K)RT HIV-1 mutants or select for highly resistant (Y181C-->C181I)RT HIV-1 mutants

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

Non-nucleoside reverse transcriptase inhibitors (NNRTIs) for the treatment of human immunodeficiency virus type 1 (HIV-1) infections: strategies to overcome drug resistance development

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

Urea-PETT compounds as a new class of HIV-1 reverse transcriptase inhibitors. 3. Synthesis and further structure-activity relationship studies of PETT analogues

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

High resolution structures of HIV-1 RT from four RT-inhibitor complexes

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

Structure of HIV-1 RT/TIBO R 86183 complex reveals similarity in the binding of diverse nonnucleoside inhibitors

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

Crystal structures of 8-Cl and 9-Cl TIBO complexed with wild-type HIV-1 RT and 8-Cl TIBO complexed with the Tyr181Cys HIV-1 RT drug-resistant mutant

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

Locations of anti-AIDS drug binding sites and resistance mutations in the three-dimensional structure of HIV-1 reverse transcriptase. Implications for mechanisms of drug inhibition and resistance

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

Structure of HIV-1 reverse transcriptase in a complex with the non-nucleoside inhibitor alpha-APA R 95845 at 2.8 A resolution

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

Structures of Tyr188Leu mutant and wild-type HIV-1 reverse transcriptase complexed with the non-nucleoside inhibitor HBY 097: inhibitor flexibility is a useful design feature for reducing drug resistance

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

Novel non-nucleoside inhibitors of human immunodeficiency virus type 1 (HIV-1) reverse transcriptase. 4. 2-Substituted dipyridodiazepinones as potent inhibitors of both wild-type and cysteine-181 HIV-1 reverse transcriptase enzymes

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

Novel non-nucleoside inhibitors of human immunodeficiency virus type 1 reverse transcriptase. 5. 4-Substituted and 2,4-disubstituted analogs of nevirapine.

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

Novel non-nucleoside inhibitors of human immunodeficiency virus type 1 reverse transcriptase. 6. 2-Indol-3-yl- and 2-azaindol-3-yl-dipyridodiazepinones

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

Structure-activity correlation study of HIV-1 inhibitors: electronic and molecular parameters

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

Quantitative structure-activity relationships and comparative molecular field analysis of TIBO derivatised HIV-1 reverse transcriptase inhibitors

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

Comparative molecular field analysis (CoMFA). 1. Effect of shape on binding of steroids to carrier proteins

1 reference

https://api.crossref.org/works/10.1016%2FS1093-3263%2800%2900053-X

7 January 2021

based on heuristic

inferred from DOI database lookup

Identifiers

10.1016/S1093-3263(00)00053-X

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11155314%20AND%20SRC:MED&resulttype=core&format=json

3 November 2019

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11155314%20AND%20SRC:MED&resulttype=core&format=json

3 November 2019

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