(Q73599332)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12837541%20AND%20SRC:MED&resulttype=core&format=json

5 November 2019

title

Synthesis and analysis of potential prodrugs of coenzyme A analogues for the inhibition of the histone acetyltransferase p300 (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12837541%20AND%20SRC:MED&resulttype=core&format=json

5 November 2019

1

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5 November 2019

author name string

Cheol M Kim

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12837541%20AND%20SRC:MED&resulttype=core&format=json

5 November 2019

Paul R Thompson

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12837541%20AND%20SRC:MED&resulttype=core&format=json

5 November 2019

Matthew Daugherty

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12837541%20AND%20SRC:MED&resulttype=core&format=json

5 November 2019

Philip A Cole

5

1 reference

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5 November 2019

language of work or name

English

0 references

publication date

1 July 2003

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12837541%20AND%20SRC:MED&resulttype=core&format=json

Bioorganic & Medicinal Chemistry

5 November 2019

published in

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12837541%20AND%20SRC:MED&resulttype=core&format=json

5 November 2019

volume

11

1 reference

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5 November 2019

issue

15

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5 November 2019

page(s)

3307-3313

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12837541%20AND%20SRC:MED&resulttype=core&format=json

Conditions for the self-catalysed inactivation of carnitine acetyltransferase. A novel form of enzyme inhibition

5 November 2019

cites work

1 reference

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7 January 2021

S-(2-oxopentadecyl)-CoA, a nonhydrolyzable analogue of myristoyl-CoA, is a potent inhibitor of myristoyl-CoA:protein N-myristoyltransferase

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7 January 2021

A Potent Inhibitor of the Melatonin Rhythm Enzyme

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7 January 2021

Mechanism-based inhibition of the melatonin rhythm enzyme: pharmacologic exploitation of active site functional plasticity

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7 January 2021

The structural basis of ordered substrate binding by serotonin N-acetyltransferase: enzyme complex at 1.8 A resolution with a bisubstrate analog

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7 January 2021

Bisubstrate ketone analogues as serotonin N-acetyltransferase inhibitors

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7 January 2021

X-ray crystallographic studies of serotonin N-acetyltransferase catalysis and inhibition

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7 January 2021

Serotonin N-acetyltransferase: mechanism and inhibition

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7 January 2021

HATs off: selective synthetic inhibitors of the histone acetyltransferases p300 and PCAF.

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7 January 2021

p300/CBP-associated factor histone acetyltransferase processing of a peptide substrate. Kinetic analysis of the catalytic mechanism

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7 January 2021

Transcriptional coactivator protein p300. Kinetic characterization of its histone acetyltransferase activity

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7 January 2021

Structure of the GCN5 histone acetyltransferase bound to a bisubstrate inhibitor

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7 January 2021

Epigenetic codes for heterochromatin formation and silencing: rounding up the usual suspects

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7 January 2021

Activator-dependent transcription from chromatin in vitro involving targeted histone acetylation by p300.

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7 January 2021

Chromatin-dependent cooperativity between constitutive and inducible activation domains in CREB.

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7 January 2021

Acetylation of nucleosomal histones by p300 facilitates transcription from tax-responsive human T-cell leukemia virus type 1 chromatin template

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7 January 2021

CBP/p300 and muscle differentiation: no HAT, no muscle

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7 January 2021

DNA damage-dependent acetylation of p73 dictates the selective activation of apoptotic target genes.

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7 January 2021

The biosynthesis of coenzyme A in bacteria

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7 January 2021

Pantothenic acid in health and disease.

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7 January 2021

Complete reconstitution of the human coenzyme A biosynthetic pathway via comparative genomics

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7 January 2021

Membrane-permeant esters of phosphatidylinositol 3,4,5-trisphosphate

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7 January 2021

Evidence for acyloxymethyl esters of pyrimidine 5'-deoxyribonucleotides as extracellular sources of active 5'-deoxyribonucleotides in cultured cells

1 reference

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7 January 2021

Synthesis and antitumor evaluation of bis[(pivaloyloxy)methyl] 2'-deoxy-5-fluorouridine 5'-monophosphate (FdUMP): a strategy to introduce nucleotides into cells

1 reference

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7 January 2021

Synthesis, in vitro antiviral evaluation, and stability studies of bis(S-acyl-2-thioethyl) ester derivatives of 9-[2-(phosphonomethoxy)ethyl]adenine (PMEA) as potential PMEA prodrugs with improved oral bioavailability

1 reference

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7 January 2021

The Role of 4-phosphonodifluoromethyl- and 4-phosphono-phenylalanine in the selectivity and cellular uptake of SH2 domain ligands

1 reference

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7 January 2021

Cellular delivery of nucleoside diphosphates: a prodrug approach

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7 January 2021

Synthesis and biological activity of bis(pivaloyloxymethyl) ester of 2'-azido-2'-deoxyuridine 5'-monophosphate

1 reference

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7 January 2021

Crystal structure of a GCN5-related N-acetyltransferase: Serratia marcescens aminoglycoside 3-N-acetyltransferase

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2803%2900265-7

7 January 2021

Structure of histone acetyltransferases

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2803%2900265-7

7 January 2021

The acetyltransferase activity of CBP stimulates transcription

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2803%2900265-7

7 January 2021

S-Ethyl-coenzyme A and acetonyldethio-coenzyme A. Interactions with pyruvate carboxylase and phosphotransacetylase

1 reference

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7 January 2021

10.1016/S0968-0896(03)00265-7

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12837541%20AND%20SRC:MED&resulttype=core&format=json

5 November 2019

1 reference