(Q74623160)

English

Irreversible inhibition of epidermal growth factor receptor tyrosine kinase with in vivo activity by N-[4-[(3-bromophenyl)amino]-6-quinazolinyl]-2-butynamide (CL-387,785)

scientific article published on 01 April 1999

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12 November 2019

Irreversible inhibition of epidermal growth factor receptor tyrosine kinase with in vivo activity by N-[4-[(3-bromophenyl)amino]-6-quinazolinyl]-2-butynamide (CL-387,785) (English)

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12 November 2019

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ChEBI release 2020-05-28

Douglas B. Kitchen

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12 November 2019

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C M Discafani

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12 November 2019

M L Carroll

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12 November 2019

M B Floyd

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12 November 2019

I J Hollander

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12 November 2019

Z Husain

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12 November 2019

B D Johnson

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12 November 2019

M K May

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12 November 2019

M S Malo

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12 November 2019

A A Minnick

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12 November 2019

R Nilakantan

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12 November 2019

R Shen

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12 November 2019

Y F Wang

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12 November 2019

A Wissner

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12 November 2019

L M Greenberger

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12 November 2019

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1 April 1999

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12 November 2019

Biochemical Pharmacology

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12 November 2019

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12 November 2019

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12 November 2019

917-925

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12 November 2019

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Human epidermal growth factor receptor cDNA sequence and aberrant expression of the amplified gene in A431 epidermoid carcinoma cells

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Tyrosine kinase inhibitors. 11. Soluble analogues of pyrrolo- and pyrazoloquinazolines as epidermal growth factor receptor inhibitors: synthesis, biological evaluation, and modeling of the mode of binding

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10.1016/S0006-2952(98)00356-6

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12 November 2019

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12 November 2019

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