(Q74818932)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11665576%20AND%20SRC:MED&resulttype=core&format=json

13 November 2019

title

Considerations in the evaluation of inverse agonism and protean agonism at G protein-coupled receptors (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11665576%20AND%20SRC:MED&resulttype=core&format=json

G protein-coupled receptor

13 November 2019

main subject

1 reference

Peter Chidiac

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11665576%20AND%20SRC:MED&resulttype=core&format=json

13 November 2019

publication date

1 January 2002

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11665576%20AND%20SRC:MED&resulttype=core&format=json

13 November 2019

published in

Methods in Enzymology

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11665576%20AND%20SRC:MED&resulttype=core&format=json

13 November 2019

volume

343

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11665576%20AND%20SRC:MED&resulttype=core&format=json

13 November 2019

page(s)

3-16

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11665576%20AND%20SRC:MED&resulttype=core&format=json

Inverse agonism at G protein-coupled receptors: (patho)physiological relevance and implications for drug discovery

13 November 2019

cites work

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

Regulation of the cellular localization and signaling properties of the alpha(1B)- and alpha(1D)-adrenoceptors by agonists and inverse agonists.

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

Regulation of peripheral cannabinoid receptor CB2 phosphorylation by the inverse agonist SR 144528. Implications for receptor biological responses

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

Labelling of recombinant human and native rat serotonin 5-HT1A receptors by a novel, selective radioligand, [3H]-S 15535: definition of its binding profile using agonists, antagonists and inverse agonists

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

Fluorescent labeling of purified beta 2 adrenergic receptor. Evidence for ligand-specific conformational changes

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

The mammalian beta 2-adrenergic receptor: reconstitution of functional interactions between pure receptor and pure stimulatory nucleotide binding protein of the adenylate cyclase system

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

Modulation of forskolin-mediated adenylyl cyclase activation by constitutively active G(S)-coupled receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

Constitutive activity of the histamine H(1) receptor reveals inverse agonism of histamine H(1) receptor antagonists

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

Modulation of basal intracellular calcium by inverse agonists and phorbol myristate acetate in rat-1 fibroblasts stably expressing alpha1d-adrenoceptors.

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

A Selective Inverse Agonist for Central Cannabinoid Receptor Inhibits Mitogen-activated Protein Kinase Activation Stimulated by Insulin or Insulin-like Growth Factor 1

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

Inverse agonist activities of beta-adrenoceptor antagonists in rat myocardium

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

Pharmacology of muscarinic receptor subtypes constitutively activated by G proteins

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

Receptor-effector coupling by G proteins

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

A three-state receptor model of agonist action

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

Sodium dependency of constitutive activity at 5-HT1D alpha/1D beta receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

Role of phosphorylation in desensitization of the beta-adrenoceptor

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

Constitutive activation of the human bradykinin B2 receptor induced by mutations in transmembrane helices III and VI.

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

Spontaneous human B2 bradykinin receptor activity determines the action of partial agonists as agonists or inverse agonists. Effect of basal desensitization

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

Agonist efficacy and allosteric models of receptor action.

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

The role of receptor kinases and arrestins in G protein-coupled receptor regulation

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

Membrane organization in G-protein mechanisms.

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

Switching of the coupling of the beta2-adrenergic receptor to different G proteins by protein kinase A.

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

Beta-arrestin-dependent formation of beta2 adrenergic receptor-Src protein kinase complexes

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2802%2943124-2

7 January 2021

10.1016/S0076-6879(02)43124-2

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11665576%20AND%20SRC:MED&resulttype=core&format=json

13 November 2019

1 reference