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Utilization of NMR-derived fragment leads in drug design
scientific article published on 01 January 2005
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1 reference
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Europe PubMed Central
PubMed publication ID
15808237
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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:15808237%20AND%20SRC:MED&resulttype=core&format=json
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10 January 2020
title
Utilization of NMR-derived fragment leads in drug design
(English)
1 reference
stated in
Europe PubMed Central
PubMed publication ID
15808237
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:15808237%20AND%20SRC:MED&resulttype=core&format=json
retrieved
10 January 2020
author name string
Jeffrey R Huth
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1
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Europe PubMed Central
PubMed publication ID
15808237
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:15808237%20AND%20SRC:MED&resulttype=core&format=json
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10 January 2020
Chaohong Sun
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2
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Europe PubMed Central
PubMed publication ID
15808237
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:15808237%20AND%20SRC:MED&resulttype=core&format=json
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10 January 2020
Daryl R Sauer
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3
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Europe PubMed Central
PubMed publication ID
15808237
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:15808237%20AND%20SRC:MED&resulttype=core&format=json
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10 January 2020
Philip J Hajduk
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4
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Europe PubMed Central
PubMed publication ID
15808237
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10 January 2020
publication date
1 January 2005
1 reference
stated in
Europe PubMed Central
PubMed publication ID
15808237
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:15808237%20AND%20SRC:MED&resulttype=core&format=json
retrieved
10 January 2020
published in
Methods in Enzymology
1 reference
stated in
Europe PubMed Central
PubMed publication ID
15808237
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:15808237%20AND%20SRC:MED&resulttype=core&format=json
retrieved
10 January 2020
volume
394
1 reference
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Europe PubMed Central
PubMed publication ID
15808237
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:15808237%20AND%20SRC:MED&resulttype=core&format=json
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10 January 2020
page(s)
549-571
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Europe PubMed Central
PubMed publication ID
15808237
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10 January 2020
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The SHAPES strategy: an NMR-based approach for lead generation in drug discovery.
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Novel inhibitors of Erm methyltransferases from NMR and parallel synthesis.
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NMR-based screening in drug discovery
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Identification of novel inhibitors of urokinase via NMR-based screening
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NMR-based modification of matrix metalloproteinase inhibitors with improved bioavailability
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Utility of NMR in lead optimization: fragment-based approaches
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Spin labels as a tool to identify and characterize protein-ligand interactions by NMR spectroscopy
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Applications of SHAPES screening in drug discovery.
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The inter-ligand Overhauser effect: a powerful new NMR approach for mapping structural relationships of macromolecular ligands
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based on heuristic
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Identifiers
DOI
10.1016/S0076-6879(05)94023-8
1 reference
stated in
Europe PubMed Central
PubMed publication ID
15808237
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:15808237%20AND%20SRC:MED&resulttype=core&format=json
retrieved
10 January 2020
PubMed publication ID
15808237
1 reference
stated in
Europe PubMed Central
PubMed publication ID
15808237
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:15808237%20AND%20SRC:MED&resulttype=core&format=json
retrieved
10 January 2020
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