(Q85225058)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:23079492%20AND%20SRC:MED&resulttype=core&format=json

15 February 2020

title

Discovery and validation of SIRT2 inhibitors based on tenovin-6: use of a ¹H-NMR method to assess deacetylase activity (English)

1 reference

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15 February 2020

3

1 reference

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15 February 2020

Daumantas Matulis

6

1 reference

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15 February 2020

Tomas Lebl

8

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15 February 2020

Nicholas J Westwood

9

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15 February 2020

author name string

Lisa Pirrie

1

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15 February 2020

Anna R McCarthy

2

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15 February 2020

Vaida Morkūnaitė

4

1 reference

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15 February 2020

Asta Zubrienė

5

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15 February 2020

Sonia Lain

7

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15 February 2020

language of work or name

English

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publication date

18 October 2012

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15 February 2020

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15 February 2020

volume

17

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15 February 2020

issue

10

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15 February 2020

page(s)

12206-12224

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Creative Commons Attribution 4.0 International

15 February 2020

copyright license

start time

18 October 2012

1 reference

April 2022 Public Data File from Crossref

copyright status

copyrighted

0 references

cites work

Isoform-selective histone deacetylase inhibitors.

1 reference

12 December 2020

Sirt5 is a NAD-dependent protein lysine demalonylase and desuccinylase

1 reference

12 December 2020

Novel cambinol analogs as sirtuin inhibitors: synthesis, biological evaluation, and rationalization of activity.

1 reference

12 December 2020

Sirtuins inhibitors: the approach to affinity and selectivity

1 reference

12 December 2020

SIRT2 inhibition achieves neuroprotection by decreasing sterol biosynthesis

1 reference

12 December 2020

SRT1720, SRT2183, SRT1460, and resveratrol are not direct activators of SIRT1

1 reference

12 December 2020

Evaluation of fluorescence-based thermal shift assays for hit identification in drug discovery

1 reference

12 December 2020

Design, synthesis, and biological activity of a novel series of human sirtuin-2-selective inhibitors

1 reference

12 December 2020

SIRT2-mediated protein deacetylation: An emerging key regulator in brain physiology and pathology

1 reference

12 December 2020

Thermodynamic stability of carbonic anhydrase: measurements of binding affinity and stoichiometry using ThermoFluor.

1 reference

12 December 2020

The critical role of the class III histone deacetylase SIRT1 in cancer

1 reference

12 December 2020

Mammalian sirtuins: biological insights and disease relevance

1 reference

12 December 2020

Inhibition and binding studies of carbonic anhydrase isozymes I, II and IX with benzimidazo[1,2-c][1,2,3]thiadiazole-7-sulphonamides

1 reference

12 December 2020

SirT2 is a histone deacetylase with preference for histone H4 Lys 16 during mitosis

1 reference

12 December 2020

Activation of p53 by SIRT1 inhibition enhances elimination of CML leukemia stem cells in combination with imatinib

1 reference

12 December 2020

SIRT1 deacetylase promotes acquisition of genetic mutations for drug resistance in CML cells

1 reference

12 December 2020

Synthesis and biological characterisation of sirtuin inhibitors based on the tenovins

1 reference

12 December 2020

Small molecule regulation of Sir2 protein deacetylases

1 reference

12 December 2020

1 reference

12 December 2020

Sirtuin 2 inhibitors rescue alpha-synuclein-mediated toxicity in models of Parkinson's disease

1 reference

12 December 2020

Activation of stress response gene SIRT1 by BCR-ABL promotes leukemogenesis

1 reference

12 December 2020

The Quenching Effect of Flavonoids on 4-Methylumbelliferone, a Potential Pitfall in Fluorimetric Neuraminidase Inhibition Assays

1 reference

12 December 2020

Discovery, in vivo activity, and mechanism of action of a small-molecule p53 activator.

1 reference

12 December 2020

The use of differential scanning fluorimetry to detect ligand interactions that promote protein stability

1 reference

12 December 2020

Characterization of chemical libraries for luciferase inhibitory activity

1 reference

12 December 2020

A quantitative model of thermal stabilization and destabilization of proteins by ligands

1 reference

12 December 2020

Inhibitors of NAD+ dependent histone deacetylases (sirtuins).

1 reference

12 December 2020

High-density miniaturized thermal shift assays as a general strategy for drug discovery

1 reference

12 December 2020

10.3390/MOLECULES171012206

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:23079492%20AND%20SRC:MED&resulttype=core&format=json

15 February 2020

1 reference

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15 February 2020

PubMed publication ID

23079492

1 reference