(Q24324741)

GOA release 2020-03-11

author

Jean-Luc Ferrer

4

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Cédric Bauvois

2

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Franck Borel

3

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author name string

Geoffray Labar

1

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Johan Wouters

5

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Didier M Lambert

Development of a potent inhibitor of 2-arachidonoylglycerol hydrolysis with antinociceptive activity in vivo

6

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language of work or name

English

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publication date

25 January 2010

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published in

ChemBioChem

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volume

11

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issue

2

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page(s)

218-27

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cites work

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Disulfiram is an inhibitor of human purified monoacylglycerol lipase, the enzyme regulating 2-arachidonoylglycerol signaling

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2-Arachidonoylglycerol: a possible endogenous cannabinoid receptor ligand in brain

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Crystallization of pancreatic procolipase and of its complex with pancreatic lipase

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Structural investigation of the cofactor-free chloroperoxidases

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Identification of an endogenous 2-monoglyceride, present in canine gut, that binds to cannabinoid receptors

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A new class of inhibitors of 2-arachidonoylglycerol hydrolysis and invasion of prostate cancer cells.

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Characterization of the sulfhydryl-sensitive site in the enzyme responsible for hydrolysis of 2-arachidonoyl-glycerol in rat cerebellar membranes

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A comprehensive profile of brain enzymes that hydrolyze the endocannabinoid 2-arachidonoylglycerol

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Covalent inhibitors of human monoacylglycerol lipase: ligand-assisted characterization of the catalytic site by mass spectrometry and mutational analysis

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Pain and beyond: fatty acid amides and fatty acid amide hydrolase inhibitors in cardiovascular and metabolic diseases

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Carbamoyl tetrazoles as inhibitors of endocannabinoid inactivation: a critical revisitation

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Protective activation of the endocannabinoid system during ischemia in dopamine neurons

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A molecular dynamics study of the pores formed by Escherichia coli OmpF porin in a fully hydrated palmitoyloleoylphosphatidylcholine bilayer

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[27] Maximum-likelihood heavy-atom parameter refinement for multiple isomorphous replacement and multiwavelength anomalous diffraction methods.

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Exon-intron organization and chromosomal localization of the mouse monoglyceride lipase gene

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The 2.46 A resolution structure of the pancreatic lipase-colipase complex inhibited by a C11 alkyl phosphonate

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Structure of human pancreatic lipase-related protein 2 with the lid in an open conformation

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Fatty acid amide hydrolase inhibitors from virtual screening of the endocannabinoid system

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Structure of a cannabinoid receptor and functional expression of the cloned cDNA

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Endogenous cannabinoids mediate retrograde signalling at hippocampal synapses

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A model for interfacial activation in lipases from the structure of a fungal lipase-inhibitor complex

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Molecular characterization of a peripheral receptor for cannabinoids

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A second endogenous cannabinoid that modulates long-term potentiation

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An endocannabinoid mechanism for stress-induced analgesia.

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Selective blockade of 2-arachidonoylglycerol hydrolysis produces cannabinoid behavioral effects

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Targeting the endocannabinoid system: to enhance or reduce?

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2-arachidonoylglycerol, an endogenous cannabinoid receptor ligand, induces rapid actin polymerization in HL-60 cells differentiated into macrophage-like cells

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7 January 2021

Brain monoglyceride lipase participating in endocannabinoid inactivation

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7 January 2021

cDNA cloning, tissue distribution, and identification of the catalytic triad of monoglyceride lipase. Evolutionary relationship to esterases, lysophospholipases, and haloperoxidases

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7 January 2021

Crystal structure of the open form of dog gastric lipase in complex with a phosphonate inhibitor

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7 January 2021

Intestinal Monoacylglycerol Metabolism

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7 January 2021

Automatic processing of rotation diffraction data from crystals of initially unknown symmetry and cell constants

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7 January 2021

Structure of an aryl esterase from Pseudomonas fluorescens.

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7 January 2021

A critical cysteine residue in monoacylglycerol lipase is targeted by a new class of isothiazolinone-based enzyme inhibitors

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7 January 2021

Therapeutic potential of endocannabinoid-hydrolysing enzyme inhibitors.

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7 January 2021

Depolarization-induced retrograde synaptic inhibition in the mouse cerebellar cortex is mediated by 2-arachidonoylglycerol.

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7 January 2021

RNA interference suggests a primary role for monoacylglycerol lipase in the degradation of the endocannabinoid 2-arachidonoylglycerol

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7 January 2021

Structural adaptations in a membrane enzyme that terminates endocannabinoid signaling

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7 January 2021

Isolation and structure of a brain constituent that binds to the cannabinoid receptor

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7 January 2021

Stereoselective esterase from Pseudomonas putida IFO12996 reveals alpha/beta hydrolase folds for D-beta-acetylthioisobutyric acid synthesis

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7 January 2021

2-arachidonoylglycerol, an endogenous cannabinoid receptor ligand, induces the migration of EoL-1 human eosinophilic leukemia cells and human peripheral blood eosinophils

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7 January 2021

Adipose triglyceride lipase and the lipolytic catabolism of cellular fat stores

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7 January 2021

Suppression of nerve growth factor Trk receptors and prolactin receptors by endocannabinoids leads to inhibition of human breast and prostate cancer cell proliferation.

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7 January 2021