(Q37679402)

English

Covalent inhibitors of human monoacylglycerol lipase: ligand-assisted characterization of the catalytic site by mass spectrometry and mutational analysis

scientific article published on August 2008

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scholarly article

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

Covalent inhibitors of human monoacylglycerol lipase: ligand-assisted characterization of the catalytic site by mass spectrometry and mutational analysis (English)

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

mass spectrometry

0 references

Alexandros Makriyannis

8

object named as

Alexandros Makriyannis

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

1

object named as

Nikolai Zvonok

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

author name string

Lakshmipathi Pandarinathan

2

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

John Williams

3

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

Meghan Johnston

4

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

Ioannis Karageorgos

5

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

David R Janero

6

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

Srinivasan C Krishnan

7

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

publication date

1 August 2008

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

Chemistry and Biology

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

15

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

8

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

854-862

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

describes a project that uses

mass spectrometry

1 reference

based on heuristic

inferred from title

Full mass spectrometric characterization of human monoacylglycerol lipase generated by large-scale expression and single-step purification

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

23 August 2017

Pharmacotherapeutic targeting of the endocannabinoid signaling system: drugs for obesity and the metabolic syndrome.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

23 August 2017

A comprehensive profile of brain enzymes that hydrolyze the endocannabinoid 2-arachidonoylglycerol

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

23 August 2017

Therapeutic potential of endocannabinoid-hydrolysing enzyme inhibitors.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

23 August 2017

Endocannabinoids and the regulation of their levels in health and disease

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

23 August 2017

A second fatty acid amide hydrolase with variable distribution among placental mammals

1 reference

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23 August 2017

The endocannabinoid system as an emerging target of pharmacotherapy

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

23 August 2017

The putative endocannabinoid transport blocker LY2183240 is a potent inhibitor of FAAH and several other brain serine hydrolases

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

23 August 2017

Identification of a high-affinity binding site involved in the transport of endocannabinoids

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

23 August 2017

Inhibition of monoacylglycerol lipase and fatty acid amide hydrolase by analogues of 2-arachidonoylglycerol

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

23 August 2017

CB2 cannabinoid receptor agonists: pain relief without psychoactive effects?

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

23 August 2017

cDNA cloning, tissue distribution, and identification of the catalytic triad of monoglyceride lipase. Evolutionary relationship to esterases, lysophospholipases, and haloperoxidases

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

23 August 2017

Molecular characterization of an enzyme that degrades neuromodulatory fatty-acid amides

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

23 August 2017

Identification of an endogenous 2-monoglyceride, present in canine gut, that binds to cannabinoid receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

23 August 2017

2-Arachidonoylglycerol: a possible endogenous cannabinoid receptor ligand in brain

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

23 August 2017

Isolation and structure of a brain constituent that binds to the cannabinoid receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

23 August 2017

Carbamoyl tetrazoles as inhibitors of endocannabinoid inactivation: a critical revisitation

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

14 September 2017

Identification of a novel endocannabinoid-hydrolyzing enzyme expressed by microglial cells

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

14 September 2017

Comprehensive proteomic mass spectrometric characterization of human cannabinoid CB2 receptor.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

1 September 2018

Fatty acid amide hydrolase inhibitors from virtual screening of the endocannabinoid system.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

1 September 2018

Characterization of the sulfhydryl-sensitive site in the enzyme responsible for hydrolysis of 2-arachidonoyl-glycerol in rat cerebellar membranes

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

1 September 2018

RNA interference suggests a primary role for monoacylglycerol lipase in the degradation of the endocannabinoid 2-arachidonoylglycerol

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

1 September 2018

Subcellular Localization and Some Properties of Monoacyiglycerol Lipase in Rat Adipocytes

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3972761

1 September 2018

Fatty acid sulfonyl fluorides inhibit anandamide metabolism and bind to the cannabinoid receptor

1 reference

https://pubmed.ncbi.nlm.nih.gov/18721756

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Anandamide amidohydrolase reacting with 2-arachidonoylglycerol, another cannabinoid receptor ligand

1 reference

https://pubmed.ncbi.nlm.nih.gov/18721756

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1016/J.CHEMBIOL.2008.06.008

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

ResearchGate publication ID

0 references

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