(Q24595919)

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Discovery of a series of 2-phenyl-N-(2-(pyrrolidin-1-yl)phenyl)acetamides as novel molecular switches that modulate modes of K(v)7.2 (KCNQ2) channel pharmacology: identification of (S)-2-phenyl-N-(2-(pyrrolidin-1-yl)phenyl)butanamide (ML252) as a potent, brain penetrant K(v)7.2 channel inhibitor (English)
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Yiu-Yin Cheung
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Haibo Yu
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Kaiping Xu
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Beiyan Zou
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Meng Wu
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Owen B McManus
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Min Li
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Corey R Hopkins
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9 August 2012
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55
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15
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6975-9
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