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Taking the time to study competitive antagonism
scientific article
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instance of
scholarly article
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review article
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Europe PubMed Central
title
Taking the time to study competitive antagonism
(English)
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author name string
D J A Wyllie
series ordinal
1
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P E Chen
series ordinal
2
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language of work or name
English
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publication date
March 2007
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published in
British Journal of Pharmacology
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volume
150
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issue
5
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page(s)
541-51
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cites work
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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction
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Identification of amino acid residues of the NR2A subunit that control glutamate potency in recombinant NR1/NR2A NMDA receptors
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Some quantitative uses of drug antagonists
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Equilibrium constants for (R)-[(S)-1-(4-bromo-phenyl)-ethylamino]-(2,3-dioxo-1,2,3,4-tetrahydroquinoxalin-5-yl)-methyl]-phosphonic acid (NVP-AAM077) acting at recombinant NR1/NR2A and NR1/NR2B N-methyl-D-aspartate receptors: Implications for studies
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Glutamate receptors at atomic resolution
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Agonist-activated ion channels
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Structural features of the glutamate binding site in recombinant NR1/NR2A N-methyl-D-aspartate receptors determined by site-directed mutagenesis and molecular modeling
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Subunit-specific gating controls rat NR1/NR2A and NR1/NR2B NMDA channel kinetics and synaptic signalling profiles.
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Molecular determinants of agonist discrimination by NMDA receptor subunits: analysis of the glutamate binding site on the NR2B subunit
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28 September 2017
Estimation of competitive antagonist affinity from functional inhibition curves using the Gaddum, Schild and Cheng-Prusoff equations
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28 September 2017
Analysis of competitive agonist-antagonist interactions by nonlinear regression.
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The effects of a series of omega-phosphonic alpha-carboxylic amino acids on electrically evoked and excitant amino acid-induced responses in isolated spinal cord preparations
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pAx and competitive drug antagonism
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Single-channel analysis of a point mutation of a conserved serine residue in the S2 ligand-binding domain of the NR2A NMDA receptor subunit
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Definition and antagonism of histamine H 2 -receptors
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28 November 2018
Identification of subunit- and antagonist-specific amino acid residues in the N-Methyl-D-aspartate receptor glutamate-binding pocket
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28 November 2018
Molecular determinants of ligand discrimination in the glutamate-binding pocket of the NMDA receptor
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Properties of human glycine receptors containing the hyperekplexia mutation alpha1(K276E), expressed in Xenopus oocytes.
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28 November 2018
The Cheng-Prusoff relationship: something lost in the translation.
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28 November 2018
Interaction at End-Plate Receptors between Different Choline Derivatives
1 reference
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reference URL
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retrieved
12 December 2020
based on heuristic
inferred from PubMed ID database lookup
Further concerns over Cheng-Prusoff analysis
1 reference
stated in
PubMed
reference URL
https://pubmed.ncbi.nlm.nih.gov/17245371
retrieved
12 December 2020
based on heuristic
inferred from PubMed ID database lookup
Identifiers
DOI
10.1038/SJ.BJP.0706997
1 reference
stated in
Consolidated OpenCitations Corpus – April 2017
OpenCitations bibliographic resource ID
2208014
OpenCitations bibliographic resource ID
2208014
1 reference
stated in
Consolidated OpenCitations Corpus – April 2017
OpenCitations bibliographic resource ID
2208014
PMC publication ID
2189774
1 reference
stated in
Consolidated OpenCitations Corpus – April 2017
OpenCitations bibliographic resource ID
2208014
PubMed publication ID
17245371
1 reference
stated in
Consolidated OpenCitations Corpus – April 2017
OpenCitations bibliographic resource ID
2208014
ResearchGate publication ID
6558581
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