(Q27642528)

English

Requirements for Specific Binding of Low Affinity Inhibitor Fragments to the SH2 Domain ofpp60Src Are Identical to Those for High Affinity Binding of Full Length Inhibitors

scientific article published on November 20, 2003

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scholarly article

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Requirements for specific binding of low affinity inhibitor fragments to the SH2 domain of (pp60)Src are identical to those for high affinity binding of full length inhibitors (English)

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Requirements for Specific Binding of Low Affinity Inhibitor Fragments to the SH2 Domain ofpp60Src Are Identical to Those for High Affinity Binding of Full Length Inhibitors (English)

1 reference

10.1021/JM020970S

https://api.crossref.org/works/10.1021/JM020970S

31 March 2024

molecular medicine

1 reference

10.1021/JM020970S

https://api.crossref.org/works/10.1021/JM020970S

31 March 2024

Jean-Pierre Marquette

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author name string

Gudrun Lange

1

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Dominique Lesuisse

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Pierre Deprez

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Bernard Schoot

4

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Petra Loenze

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Didier Bénard

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Pierre Broto

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Edoardo Sarubbi

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Eliane Mandine

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language of work or name

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publication date

20 November 2003

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full work available at URL

https://pubs.acs.org/doi/pdf/10.1021/jm020970s

1 reference

10.1021/JM020970S

https://api.crossref.org/works/10.1021/JM020970S

31 March 2024

Journal of Medicinal Chemistry

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46

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24

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5184-95

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Targeted disruption of the c-src proto-oncogene leads to osteopetrosis in mice

1 reference

24 May 2022

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A geometric approach to macromolecule-ligand interactions

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A fast flexible docking method using an incremental construction algorithm.

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Comparative computer graphics and solution studies of the DNA interaction of substituted anthraquinones based on doxorubicin and mitoxantrone

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Discovering high-affinity ligands for proteins: SAR by NMR

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NMR-based discovery of phosphotyrosine mimetics that bind to the Lck SH2 domain

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Discovering novel ligands for macromolecules using X-ray crystallographic screening

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SAR and X-ray. A new approach combining fragment-based screening and rational drug design: application to the discovery of nanomolar inhibitors of Src SH2.

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Binding of a high affinity phosphotyrosyl peptide to the Src SH2 domain: crystal structures of the complexed and peptide-free forms

11

1 reference

10.1021/JM020970S

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31 March 2024

Bioorganic & Medicinal Chemistry Letters

12

12

1298

author name string

Deprez P.

publication date

2002

1 reference

10.1021/JM020970S

https://api.crossref.org/works/10.1021/JM020970S

31 March 2024

Bioorganic & Medicinal Chemistry Letters

13

12

1294

author name string

Deprez P.

publication date

2002

1 reference

10.1021/JM020970S

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31 March 2024

Discovery of thioazepinone ligands for Src SH2: from non-specific to specific binding

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1 reference

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Principles governing the binding of a class of non-peptidic inhibitors to the SH2 domain of src studied by X-ray analysis

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10.1021/JM020970S

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Automatic processing of rotation diffraction data from crystals of initially unknown symmetry and cell constants

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Direct phase determination for the molecular envelope of tryptophanyl-tRNA synthetase from Bacillus stearothermophilus by X-ray contrast variation

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The Protein Data Bank

20

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A novel phosphotyrosine mimetic 4'-carboxymethyloxy-3'-phosphonophenylalanine (Cpp): exploitation in the design of nonpeptide inhibitors of pp60(Src) SH2 domain

22

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Structure-based design of an osteoclast-selective, nonpeptide src homology 2 inhibitor with in vivo antiresorptive activity

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1 reference

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Proceedings of the National Academy of Sciences of the United States of America

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97

2424

author name string

Maly D. J.

publication date

2000

1 reference

10.1021/JM020970S

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Characterization of SH2-ligand interactions via library affinity selection with mass spectrometric detection

25

1 reference

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Journal of Medicinal Chemistry

26

43

3447

author name string

Hajduk P. J.

publication date

2000

1 reference

10.1021/JM020970S

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Thioformaldehyde S-sulfide (Thiosulfine)

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1 reference

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Peptide ligands of pp60(c-src) SH2 domains: a thermodynamic and structural study

29

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10.1021/JM020970S

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Electrostatic contributions to protein-protein interactions: fast energetic filters for docking and their physical basis

32

1 reference

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Proceedings of the National Academy of Sciences of the United States of America

34

95

5864

author name string

Schultz J.

publication date

1998

1 reference

10.1021/JM020970S

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31 March 2024

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10.1021/JM020970S

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