(Q27649007)

2

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Emilia Caselli

3

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Brian K Shoichet

4

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Fabio Prati

Bioorganic & Medicinal Chemistry

5

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language of work or name

English

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publication date

1 February 2008

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published in

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volume

16

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issue

3

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page(s)

1195-205

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cites work

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The crystal structure of phosphonate-inhibited D-Ala-D-Ala peptidase reveals an analogue of a tetrahedral transition state

20 March 2017

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Nanomolar inhibitors of AmpC beta-lactamase

20 March 2017

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Structural milestones in the reaction pathway of an amide hydrolase: substrate, acyl, and product complexes of cephalothin with AmpC beta-lactamase

20 March 2017

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Structures of ceftazidime and its transition-state analogue in complex with AmpC beta-lactamase: implications for resistance mutations and inhibitor design

20 March 2017

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Energetic, structural, and antimicrobial analyses of beta-lactam side chain recognition by beta-lactamases

20 March 2017

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Structure-based design guides the improved efficacy of deacylation transition state analogue inhibitors of TEM-1 beta-Lactamase(,)

20 March 2017

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The complexed structure and antimicrobial activity of a non-β-lactam inhibitor of AmpC β-lactamase

20 March 2017

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Three-dimensional structure of AmpC beta-lactamase from Escherichia coli bound to a transition-state analogue: possible implications for the oxyanion hypothesis and for inhibitor design

20 March 2017

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Crystallographic structure of a phosphonate derivative of the Enterobacter cloacae P99 cephalosporinase: mechanistic interpretation of a beta-lactamase transition-state analog

20 March 2017

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7 April 2017

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29 September 2017

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Hydrogen bonding and biological specificity analysed by protein engineering

29 September 2017

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A quick method for the determination of inhibition constants

29 September 2017

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Contribution of conformer focusing to the uncertainty in predicting free energies for protein-ligand binding.

2 June 2018

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Inhibitor specificity via protein dynamics: insights from the design of antibacterial agents targeted against thymidylate synthase

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An Improved Preparation of Arylboronates: Application in One-Pot Suzuki Biaryl Synthesis†

27 November 2018

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27 November 2018

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27 November 2018

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Spatial localization of the K+ channel selectivity filter by mutant cycle-based structure analysis.

27 November 2018

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27 November 2018

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A new protocol for the one-pot synthesis of symmetrical biaryls

27 November 2018

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12 December 2020

Ester and orthoester formation in the alcoholysis of iminoester hydrochlorides; a proposed mechanism

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12 December 2020

Processing of X-ray diffraction data collected in oscillation mode

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12 December 2020

Reversible enzyme inhibitors as mechanistic probes

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