(Q27658211)

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Identification of a brain penetrant PDE9A inhibitor utilizing prospective design and chemical enablement as a rapid lead optimization strategy

scientific article

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Identification of a brain penetrant PDE9A inhibitor utilizing prospective design and chemical enablement as a rapid lead optimization strategy (English)
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Patrick R Verhoest
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Caroline Proulx-Lafrance
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Michael Corman
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Lois Chenard
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Christopher J Helal
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Xinjun Hou
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Eric Marr
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Frank S Menniti
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Christopher J Schmidt
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Michelle Vanase-Frawley
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Anne W Schmidt
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Robert D Williams
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Frederick R Nelson
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Kari R Fonseca
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Spiros Liras
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24 December 2009
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52
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24
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7946-9
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