(Q27676635)

2

0 references

Antonello Mai

object named as

Antonello Mai

9

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author name string

Anup K Upadhyay

1

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Ji Woong Han

3

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Ruogu Hu

4

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Donatella Labella

6

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Xing Zhang

7

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Young-Sup Yoon

8

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Xiaodong Cheng

Journal of Molecular Biology

10

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language of work or name

English

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publication date

24 February 2012

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published in

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volume

416

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issue

3

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page(s)

319-27

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cites work

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Quantitative High-Throughput Screening Identifies 8-Hydroxyquinolines as Cell-Active Histone Demethylase Inhibitors

20 March 2017

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PHF8 mediates histone H4 lysine 20 demethylation events involved in cell cycle progression

20 March 2017

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Histone H4K20/H3K9 demethylase PHF8 regulates zebrafish brain and craniofacial development

20 March 2017

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Selective Inhibitors of the JMJD2 Histone Demethylases: Combined Nondenaturing Mass Spectrometric Screening and Crystallographic Approaches

20 March 2017

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20 March 2017

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Discovery of a 2,4-Diamino-7-aminoalkoxyquinazoline as a Potent and Selective Inhibitor of Histone Lysine Methyltransferase G9a

20 March 2017

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Structural basis for G9a-like protein lysine methyltransferase inhibition by BIX-01294

20 March 2017

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Specificity and mechanism of JMJD2A, a trimethyllysine-specific histone demethylase

20 March 2017

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The X-linked mental retardation gene SMCX/JARID1C defines a family of histone H3 lysine 4 demethylases

20 March 2017

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Loss-of-function mutations in euchromatin histone methyl transferase 1 (EHMT1) cause the 9q34 subtelomeric deletion syndrome

20 March 2017

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20 March 2017

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20 March 2017

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20 March 2017

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JmjC-domain-containing proteins and histone demethylation

20 March 2017

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Multiparametric scaling of diffraction intensities

7 April 2017

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Targeting Histone Demethylases: A New Avenue for the Fight against Cancer

7 April 2017

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Optimization of cellular activity of G9a inhibitors 7-aminoalkoxy-quinazolines

29 September 2017

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Epigenetic modifications as therapeutic targets

29 September 2017

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Design, synthesis, enzyme-inhibitory activity, and effect on human cancer cells of a novel series of jumonji domain-containing protein 2 histone demethylase inhibitors.

29 September 2017

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Targeting epigenetic enzymes for drug discovery

29 September 2017

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Dual-specificity histone demethylase KIAA1718 (KDM7A) regulates neural differentiation through FGF4.

29 September 2017

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Histone lysine demethylases: emerging roles in development, physiology and disease

29 September 2017

1 reference

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The histone H3K4 demethylase SMCX links REST target genes to X-linked mental retardation.

29 September 2017

1 reference

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Reversal of H3K9me2 by a small-molecule inhibitor for the G9a histone methyltransferase

29 September 2017

1 reference

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ZONE BEHAVIOR OF ENZYMES : ILLUSTRATED BY THE EFFECT OF DISSOCIATION CONSTANT AND DILUTION ON THE SYSTEM CHOLINESTERASE-PHYSOSTIGMINE.

29 September 2017

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KIAA1718 is a histone demethylase that erases repressive histone methyl marks.

2 June 2018

1 reference

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JmjC: cupin metalloenzyme-like domains in jumonji, hairless and phospholipase A2β

27 November 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/22227394

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Evaluation of enzyme inhibitors in drug discovery. A guide for medicinal chemists and pharmacologists

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/22227394