(Q27685477)

English

Discovery of epigenetic regulator I-BET762: lead optimization to afford a clinical candidate inhibitor of the BET bromodomains

scientific article

Statements

Discovery of epigenetic regulator I-BET762: lead optimization to afford a clinical candidate inhibitor of the BET bromodomains (English)
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Romain Gosmini
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Jérôme Toum
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Catherine A Clément
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Mélanie Barnathan
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Jean-Marie Brusq
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Jacqueline E Mordaunt
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Richard M Grimes
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Miriam Crowe
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Olivier Pineau
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Myriam Ajakane
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Alain Daugan
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Phillip Jeffrey
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Leanne Cutler
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Andrea C Haynes
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Nicholas N Smithers
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Chun-wa Chung
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Antonia Lewis
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Jason Witherington
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Nigel Parr
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Rab K Prinjha
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Edwige Nicodème
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10 October 2013
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56
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7501-15
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19
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