(Q27705339)

English

Discovery of (S)-1-(1-(4-Chloro-3-fluorophenyl)-2-hydroxyethyl)-4-(2-((1-methyl-1H-pyrazol-5-yl)amino)pyrimidin-4-yl)pyridin-2(1H)-one (GDC-0994), an Extracellular Signal-Regulated Kinase 1/2 (ERK1/2) Inhibitor in Early Clinical Development

scientific article

Statements

Discovery of (S)-1-(1-(4-Chloro-3-fluorophenyl)-2-hydroxyethyl)-4-(2-((1-methyl-1H-pyrazol-5-yl)amino)pyrimidin-4-yl)pyridin-2(1H)-one (GDC-0994), an Extracellular Signal-Regulated Kinase 1/2 (ERK1/2) Inhibitor in Early Clinical Development (English)
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James F Blake
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Michael Burkard
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Jocelyn Chan
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Huifen Chen
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Kang-Jye Chou
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Dolores Diaz
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Danette A Dudley
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John J Gaudino
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Jonas Grina
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Thomas Hunsaker
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Lichuan Liu
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Matthew Martinson
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David Moreno
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Lars Mueller
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Christine Orr
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Patricia Pacheco
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Ann Qin
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Kevin Rasor
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Li Ren
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Kirk Robarge
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Sheerin Shahidi-Latham
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Jeffrey Stults
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Francis Sullivan
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Weiru Wang
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Jianping Yin
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Aihe Zhou
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Marcia Belvin
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Mark Merchant
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John Moffat
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Jacob B Schwarz
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23 June 2016
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59
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12
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5650-60
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