(Q28207222)

Okadaic acid: the archetypal serine/threonine protein phosphatase inhibitor

31 March 2020

1 reference

Vibrio alginolyticus, a tetrodotoxin-producing bacterium, in the intestines of the fish Fugu vermicularis vermicularis

31 March 2020

1 reference

Ernest Guenther award in chemistry of natural products. Amphibian skin: a remarkable source of biologically active arthropod alkaloids

31 March 2020

1 reference

Broad-spectrum, non-opioid analgesic activity by selective modulation of neuronal nicotinic acetylcholine receptors

31 March 2020

1 reference

Nicotinic acetylcholine receptor regulation of spinal norepinephrine release

31 March 2020

1 reference

Purification and sequence of a presynaptic peptide toxin from Conus geographus venom

31 March 2020

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Novel omega-conotoxins from Conus catus discriminate among neuronal calcium channel subtypes

31 March 2020

1 reference

Isolation and characterization of a cone snail protease with homology to CRISP proteins of the pathogenesis-related protein superfamily

31 March 2020

1 reference

Synthesis, structure elucidation, in vitro biological activity, toxicity, and Caco-2 cell permeability of lipophilic analogues of alpha-conotoxin MII.

31 March 2020

1 reference

The voltage-gated potassium channels and their relatives

31 March 2020

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The principle of gating charge movement in a voltage-dependent K+ channel

31 March 2020

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X-ray structure of a voltage-dependent K+ channel

31 March 2020

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Functional analysis of an archaebacterial voltage-dependent K+ channel

31 March 2020

1 reference

Helical structure of the COOH terminus of S3 and its contribution to the gating modifier toxin receptor in voltage-gated ion channels

31 March 2020

1 reference

Solution structure of hanatoxin1, a gating modifier of voltage-dependent K(+) channels: common surface features of gating modifier toxins

31 March 2020

1 reference

The molecular basis of voltage-gated Ca2+ channel diversity: is it time for T?

31 March 2020

1 reference

Pharmacological dissection of multiple types of Ca2+ channel currents in rat cerebellar granule neurons

31 March 2020

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Identification of functionally distinct isoforms of the N-type Ca2+ channel in rat sympathetic ganglia and brain

31 March 2020

1 reference

Neuronal calcium channel antagonists. Discrimination between calcium channel subtypes using omega-conotoxin from Conus magus venom

31 March 2020

1 reference

Inhibition of N- and L-type Ca2+ channels by the spider venom toxin omega-Aga-IIIA.

31 March 2020

1 reference

P-type calcium channels blocked by the spider toxin ω-Aga-IVA

31 March 2020

1 reference

Selective peptide antagonist of the class E calcium channel from the venom of the tarantula Hysterocrates gigas

31 March 2020

1 reference

Discovery and structure of a potent and highly specific blocker of insect calcium channels

31 March 2020

1 reference

Calciseptine, a peptide isolated from black mamba venom, is a specific blocker of the L-type calcium channel

31 March 2020

1 reference

Localization of N-type Ca2+ channels in the rat spinal cord following chronic constrictive nerve injury

31 March 2020

1 reference

Upregulation of dorsal root ganglion (alpha)2(delta) calcium channel subunit and its correlation with allodynia in spinal nerve-injured rats.

31 March 2020

1 reference

Effect of continuous intrathecal infusion of omega-conopeptides, N-type calcium-channel blockers, on behavior and antinociception in the formalin and hot-plate tests in rats

31 March 2020

1 reference

Interactions of intrathecally administered ziconotide, a selective blocker of neuronal N-type voltage-sensitive calcium channels, with morphine on nociception in rats

31 March 2020

1 reference

Structure-activity relationships of omega-conotoxins at N-type voltage-sensitive calcium channels

31 March 2020

1 reference

Omega-conotoxin CVID inhibits a pharmacologically distinct voltage-sensitive calcium channel associated with transmitter release from preganglionic nerve terminals

31 March 2020

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The novel N-type calcium channel blocker, AM336, produces potent dose-dependent antinociception after intrathecal dosing in rats and inhibits substance P release in rat spinal cord slices

31 March 2020

1 reference

Actions of intrathecal omega-conotoxins CVID, GVIA, MVIIA, and morphine in acute and neuropathic pain in the rat.

31 March 2020

1 reference

Nomenclature of voltage-gated sodium channels

31 March 2020

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A tetrodotoxin-resistant voltage-gated sodium channel expressed by sensory neurons

31 March 2020

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A tetrodotoxin-resistant voltage-gated sodium channel from human dorsal root ganglia, hPN3/SCN10A

31 March 2020

1 reference

A comparison of the potential role of the tetrodotoxin-insensitive sodium channels, PN3/SNS and NaN/SNS2, in rat models of chronic pain

31 March 2020

1 reference

Redistribution of Na(V)1.8 in uninjured axons enables neuropathic pain.

31 March 2020

1 reference

Modification of sodium channel gating and kinetics by versutoxin from the Australian funnel-web spider Hadronyche versuta.

31 March 2020

1 reference

Three-dimensional structure analysis of mu-agatoxins: further evidence for common motifs among neurotoxins with diverse ion channel specificities

31 March 2020

1 reference

Binding of sea anemone toxin to receptor sites associated with gating system of sodium channel in synaptic nerve endings in vitro

31 March 2020

1 reference

Structure and structure-function relationships of sea anemone proteins that interact with the sodium channel

31 March 2020

1 reference

Scorpion toxins specific for Na+-channels

31 March 2020

1 reference

mu-Conotoxin PIIIA, a new peptide for discriminating among tetrodotoxin-sensitive Na channel subtypes.

31 March 2020

1 reference

Isolation of a tarantula toxin specific for a class of proton-gated Na+ channels.

31 March 2020

1 reference

Discrimination of muscle and neuronal Na-channel subtypes by binding competition between [3H]saxitoxin and mu-conotoxins

31 March 2020

1 reference

Reconstitution of IKATP: an inward rectifier subunit plus the sulfonylurea receptor

31 March 2020

1 reference

K(+) channels as therapeutic drug targets

31 March 2020

1 reference

Terminally alkylated polyamine analogues as chemotherapeutic agents.

31 March 2020

1 reference

Therapeutic strategies for prevention of sickle cell dehydration

31 March 2020

1 reference

Correolide and derivatives are novel immunosuppressants blocking the lymphocyte Kv1.3 potassium channels

31 March 2020

1 reference

Potassium channels: from scorpion venoms to high-resolution structure

31 March 2020

1 reference

Subunit composition of brain voltage-gated potassium channels determined by hongotoxin-1, a novel peptide derived from Centruroides limbatus venom

31 March 2020

1 reference

Selective blockers of voltage-gated K+ channels depolarize human T lymphocytes: mechanism of the antiproliferative effect of charybdotoxin

31 March 2020

1 reference

Charybdotoxin inhibits proliferation and interleukin 2 production in human peripheral blood lymphocytes

31 March 2020

1 reference

ShK-Dap22, a potent Kv1.3-specific immunosuppressive polypeptide

31 March 2020

1 reference

A novel fluorescent toxin to detect and investigate Kv1.3 channel up-regulation in chronically activated T lymphocytes

31 March 2020

1 reference

Selective blockade of T lymphocyte K(+) channels ameliorates experimental autoimmune encephalomyelitis, a model for multiple sclerosis

31 March 2020

1 reference

The voltage-gated Kv1.3 K(+) channel in effector memory T cells as new target for MS

31 March 2020

1 reference

Oncogenic potential of EAG K(+) channels

31 March 2020

1 reference

Isolation of a long-lasting eag-related gene-type K+ current in MMQ lactotrophs and its accommodating role during slow firing and prolactin release.

31 March 2020

1 reference

New binding site on common molecular scaffold provides HERG channel specificity of scorpion toxin BeKm-1

31 March 2020

1 reference

APETx1, a new toxin from the sea anemone Anthopleura elegantissima, blocks voltage-gated human ether-a-go-go-related gene potassium channels.

31 March 2020

1 reference

Purification and characterization of chlorotoxin, a chloride channel ligand from the venom of the scorpion

31 March 2020

1 reference

Chlorotoxin‐sensitive Ca2+‐activated Cl− channel in type R2 reactive astrocytes from adult rat brain

31 March 2020

1 reference

Chlorotoxin inhibits glioma cell invasion via matrix metalloproteinase-2

31 March 2020

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Chlorotoxin does not inhibit volume-regulated, calcium-activated and cyclic AMP-activated chloride channels

31 March 2020

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Chlorotoxin, a scorpion-derived peptide, specifically binds to gliomas and tumors of neuroectodermal origin

31 March 2020

1 reference

Molecular determinants by which a long chain toxin from snake venom interacts with the neuronal alpha 7-nicotinic acetylcholine receptor

31 March 2020

1 reference

Conus peptides targeted to specific nicotinic acetylcholine receptor subtypes

31 March 2020

1 reference

Synthesis and Structure-Activity Relationships of Neuromuscular Blocking Agents

31 March 2020

1 reference

A novel alpha-conotoxin identified by gene sequencing is active in suppressing the vascular response to selective stimulation of sensory nerves in vivo.

31 March 2020

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Prevention and management of chronic heart failure in patients at risk

31 March 2020

1 reference

A new natriuretic peptide in porcine brain

31 March 2020

1 reference

Natriuretic peptide receptors and neutral endopeptidase in mediating the renal actions of a new therapeutic synthetic natriuretic peptide dendroaspis natriuretic peptide

31 March 2020

1 reference

Cell attachment activity of fibronectin can be duplicated by small synthetic fragments of the molecule

31 March 2020

1 reference

Non-peptide fibrinogen receptor antagonists. 1. Discovery and design of exosite inhibitors

31 March 2020

1 reference

Novel platelet inhibitors

31 March 2020

1 reference

Cost-effectiveness of ancrod treatment of acute ischaemic stroke: results from the Stroke Treatment with Ancrod Trial (STAT).

31 March 2020

1 reference

A family of textilinin genes, two of which encode proteins with antihaemorrhagic properties.

31 March 2020

1 reference

Two new classes of conopeptides inhibit the alpha1-adrenoceptor and noradrenaline transporter

31 March 2020

1 reference

Allosteric alpha 1-adrenoreceptor antagonism by the conopeptide rho-TIA.

31 March 2020

1 reference

Identification of a peptide toxin from Grammostola spatulata spider venom that blocks cation-selective stretch-activated channels

31 March 2020

1 reference

Solution structure of peptide toxins that block mechanosensitive ion channels

31 March 2020

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Tarantula peptide inhibits atrial fibrillation

31 March 2020

1 reference

Role of norepinephrine in the pathophysiology and treatment of mood disorders

31 March 2020

1 reference

Descending control of pain

31 March 2020

1 reference

Advances in the pharmacological control of the bladder

31 March 2020

1 reference

Isolation and characterization of a novel conus peptide with apparent antinociceptive activity

31 March 2020

1 reference

chi-Conopeptide MrIA partially overlaps desipramine and cocaine binding sites on the human norepinephrine transporter

31 March 2020

1 reference

Inhibition of the norepinephrine transporter by the venom peptide chi-MrIA. Site of action, Na+ dependence, and structure-activity relationship

31 March 2020

1 reference

Determination of the solution structures of conantokin-G and conantokin-T by CD and NMR spectroscopy

31 March 2020

1 reference

Structure-activity studies of conantokins as human N-methyl-D-aspartate receptor modulators

31 March 2020

1 reference

Spermine modulation of the glutamate(NMDA) receptor is differentially responsive to conantokins in normal and Alzheimer's disease human cerebral cortex

31 March 2020

1 reference

Conantokin-L, a new NMDA receptor antagonist: determinants for anticonvulsant potency.

31 March 2020

1 reference

Powerful antinociceptive effects of the cone snail venom-derived subtype-selective NMDA receptor antagonists conantokins G and T.

31 March 2020

1 reference

Contulakin-G, an O-glycosylated invertebrate neurotensin

31 March 2020

1 reference

Black widow spider alpha-latrotoxin: a presynaptic neurotoxin that shares structural homology with the glucagon-like peptide-1 family of insulin secretagogic hormones

31 March 2020

1 reference

The glucagon-like peptides: a new genre in therapeutic targets for intervention in Alzheimer's disease.

31 March 2020

1 reference

Isolation, structure, and activity of GID, a novel alpha 4/7-conotoxin with an extended N-terminal sequence

31 March 2020

1 reference

Solution structure of ShK toxin, a novel potassium channel inhibitor from a sea anemone

31 March 2020

1 reference

NMR sequential assignments and solution structure of chlorotoxin, a small scorpion toxin that blocks chloride channels

31 March 2020

1 reference

Determination of the three-dimensional structure of margatoxin by 1H, 13C, 15N triple-resonance nuclear magnetic resonance spectroscopy

31 March 2020

1 reference

Structural determinants of the blockade of N-type calcium channels by a peptide neurotoxin

31 March 2020

1 reference

A mu-conotoxin-insensitive Na+ channel mutant: possible localization of a binding site at the outer vestibule

31 March 2020

1 reference

Molecular mechanisms of nociception

31 March 2020

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31 March 2020

1 reference

Crystal structure of an ACh-binding protein reveals the ligand-binding domain of nicotinic receptors

31 March 2020

1 reference

Experimentally based model of a complex between a snake toxin and the alpha 7 nicotinic receptor

31 March 2020

1 reference

Alpha-conotoxins PnIA and [A10L]PnIA stabilize different states of the alpha7-L247T nicotinic acetylcholine receptor.

31 March 2020

1 reference

Structure of the BgK-Kv1.1 complex based on distance restraints identified by double mutant cycles. Molecular basis for convergent evolution of Kv1 channel blockers

31 March 2020

1 reference

Crystal structure of rhodopsin: A G protein-coupled receptor

31 March 2020

1 reference

X-ray structure of a ClC chloride channel at 3.0 A reveals the molecular basis of anion selectivity

31 March 2020

1 reference

Mechanisms of activation, inhibition and specificity: crystal structures of the NMDA receptor NR1 ligand-binding core

31 March 2020

1 reference

Rational design of a CD4 mimic that inhibits HIV-1 entry and exposes cryptic neutralization epitopes

31 March 2020

1 reference

Angiotensin-converting enzyme inhibitors from the venom of Bothrops jararaca. Isolation, elucidation of structure, and synthesis

31 March 2020

1 reference

Design of angiotensin converting enzyme inhibitors

31 March 2020

1 reference

Design of potent competitive inhibitors of angiotensin-converting enzyme. Carboxyalkanoyl and mercaptoalkanoyl amino acids

31 March 2020

1 reference

Crystal structure of the human angiotensin-converting enzyme-lisinopril complex

31 March 2020

1 reference

Defibrinogenating enzymes

31 March 2020

1 reference